JP2011500801A5 - - Google Patents

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JP2011500801A5
JP2011500801A5 JP2010530989A JP2010530989A JP2011500801A5 JP 2011500801 A5 JP2011500801 A5 JP 2011500801A5 JP 2010530989 A JP2010530989 A JP 2010530989A JP 2010530989 A JP2010530989 A JP 2010530989A JP 2011500801 A5 JP2011500801 A5 JP 2011500801A5
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optionally substituted
independently
heteroaryl
optionally
group
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JP2010530989A
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JP2011500801A (ja
JP5635909B2 (ja
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Priority claimed from PCT/US2007/089178 external-priority patent/WO2009054864A1/en
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JP2010530989A 2007-10-26 2007-12-29 Axl阻害剤として有用な多環アリール置換トリアゾール及び多環ヘテロアリール置換トリアゾール Expired - Fee Related JP5635909B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US98310707P 2007-10-26 2007-10-26
US60/983,107 2007-10-26
PCT/US2007/089178 WO2009054864A1 (en) 2007-10-26 2007-12-29 Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as axl inhibitors

Publications (3)

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JP2011500801A JP2011500801A (ja) 2011-01-06
JP2011500801A5 true JP2011500801A5 (https=) 2012-09-06
JP5635909B2 JP5635909B2 (ja) 2014-12-03

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JP2010530989A Expired - Fee Related JP5635909B2 (ja) 2007-10-26 2007-12-29 Axl阻害剤として有用な多環アリール置換トリアゾール及び多環ヘテロアリール置換トリアゾール

Country Status (7)

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US (2) US7935693B2 (https=)
EP (1) EP2205592B1 (https=)
JP (1) JP5635909B2 (https=)
CA (1) CA2704052C (https=)
ES (1) ES2424259T3 (https=)
SI (1) SI2205592T1 (https=)
WO (1) WO2009054864A1 (https=)

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EP2079736B1 (en) 2006-12-29 2017-10-18 Rigel Pharmaceuticals, Inc. Substituted triazoles useful as axl inhibitors
EP2078010B1 (en) 2006-12-29 2014-01-29 Rigel Pharmaceuticals, Inc. Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
WO2008083353A1 (en) * 2006-12-29 2008-07-10 Rigel Pharmaceuticals, Inc. Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as axl inhibitors
WO2009054864A1 (en) * 2007-10-26 2009-04-30 Rigel Pharmaceuticals, Inc. Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as axl inhibitors
US8309566B2 (en) 2008-02-15 2012-11-13 Rigel Pharmaceuticals, Inc. Pyrimidine-2-amine compounds and their use as inhibitors of JAK kinases
US8431594B2 (en) 2008-07-09 2013-04-30 Rigel Pharmaceuticals, Inc. Bridged bicyclic heteroaryl substituted triazoles useful as AXL inhibitors
CA2730231C (en) 2008-07-09 2016-10-18 Rigel Pharmaceuticals, Inc. Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
JP4644273B2 (ja) * 2008-07-15 2011-03-02 本田技研工業株式会社 車両周辺監視装置
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JP7156287B2 (ja) 2017-08-23 2022-10-19 小野薬品工業株式会社 Axl阻害剤を有効成分として含むがん治療剤
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US20230183379A1 (en) 2018-11-20 2023-06-15 INSERM (Institut National de la Santé et de la Recherche Médicale) Bispecific antibody targeting transferrin receptor 1 and soluble antigen
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WO2021048292A1 (en) 2019-09-11 2021-03-18 INSERM (Institut National de la Santé et de la Recherche Médicale) Methods and compositions for treating melanoma
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WO2021148581A1 (en) 2020-01-22 2021-07-29 Onxeo Novel dbait molecule and its use
US20230072528A1 (en) 2020-02-05 2023-03-09 INSERM (Institut National de la Santé et de la Recherche Médicale) Methods for discontinuing a treatment with a tyrosine kinase inhibitor (tki)
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WO2021204713A1 (en) 2020-04-08 2021-10-14 Bergenbio Asa Axl inhibitors for antiviral therapy
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WO2024051667A1 (zh) * 2022-09-05 2024-03-14 南京正大天晴制药有限公司 具有axl抑制活性的取代三唑化合物
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