JP2010534722A5 - - Google Patents

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Publication number
JP2010534722A5
JP2010534722A5 JP2010520074A JP2010520074A JP2010534722A5 JP 2010534722 A5 JP2010534722 A5 JP 2010534722A5 JP 2010520074 A JP2010520074 A JP 2010520074A JP 2010520074 A JP2010520074 A JP 2010520074A JP 2010534722 A5 JP2010534722 A5 JP 2010534722A5
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JP
Japan
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agent
drugs
drug
pharmaceutically acceptable
diastereomers
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JP2010520074A
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English (en)
Japanese (ja)
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JP2010534722A (ja
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Priority claimed from PCT/US2008/070962 external-priority patent/WO2009018065A2/en
Publication of JP2010534722A publication Critical patent/JP2010534722A/ja
Publication of JP2010534722A5 publication Critical patent/JP2010534722A5/ja
Withdrawn legal-status Critical Current

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JP2010520074A 2007-07-27 2008-07-24 新規グルコキナーゼ活性化薬およびその使用方法 Withdrawn JP2010534722A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US95227307P 2007-07-27 2007-07-27
PCT/US2008/070962 WO2009018065A2 (en) 2007-07-27 2008-07-24 Novel glucokinase activators and methods of using same

Publications (2)

Publication Number Publication Date
JP2010534722A JP2010534722A (ja) 2010-11-11
JP2010534722A5 true JP2010534722A5 (enExample) 2011-09-01

Family

ID=39811513

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010520074A Withdrawn JP2010534722A (ja) 2007-07-27 2008-07-24 新規グルコキナーゼ活性化薬およびその使用方法

Country Status (6)

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US (2) US7812048B2 (enExample)
EP (1) EP2173717B9 (enExample)
JP (1) JP2010534722A (enExample)
CN (1) CN101808995A (enExample)
ES (1) ES2408384T3 (enExample)
WO (1) WO2009018065A2 (enExample)

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US8222285B2 (en) 2007-06-11 2012-07-17 Bristol-Myers Squibb Company 1,3-dihydroxy substituted phenylamide glucokinase activators
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US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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CN109715637B (zh) 2016-07-22 2022-04-05 百时美施贵宝公司 葡萄糖激酶激活剂及其使用方法
US11872221B2 (en) * 2020-01-31 2024-01-16 Hua Medicine (Shanghai) Ltd. Treating untreated or treatment-resistant diabetes with glucokinase activator
US11857536B2 (en) * 2020-06-04 2024-01-02 Hua Medicine (Shanghai) Ltd. Glucokinase activator for treating diabetes with renal impairment

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