JP2010526777A5 - - Google Patents

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Publication number
JP2010526777A5
JP2010526777A5 JP2010506388A JP2010506388A JP2010526777A5 JP 2010526777 A5 JP2010526777 A5 JP 2010526777A5 JP 2010506388 A JP2010506388 A JP 2010506388A JP 2010506388 A JP2010506388 A JP 2010506388A JP 2010526777 A5 JP2010526777 A5 JP 2010526777A5
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JP
Japan
Prior art keywords
adamantan
butyramide
dichloro
phenoxy
hydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2010506388A
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English (en)
Japanese (ja)
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JP2010526777A (ja
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Publication date
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Priority claimed from PCT/US2008/059903 external-priority patent/WO2008134221A1/en
Publication of JP2010526777A publication Critical patent/JP2010526777A/ja
Publication of JP2010526777A5 publication Critical patent/JP2010526777A5/ja
Ceased legal-status Critical Current

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JP2010506388A 2007-04-24 2008-04-10 置換アミドの医薬用途 Ceased JP2010526777A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07106828 2007-04-24
US92692407P 2007-04-30 2007-04-30
PCT/US2008/059903 WO2008134221A1 (en) 2007-04-24 2008-04-10 Pharmaceutical use of substituted amides

Publications (2)

Publication Number Publication Date
JP2010526777A JP2010526777A (ja) 2010-08-05
JP2010526777A5 true JP2010526777A5 (cg-RX-API-DMAC7.html) 2011-05-12

Family

ID=39926028

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010506388A Ceased JP2010526777A (ja) 2007-04-24 2008-04-10 置換アミドの医薬用途

Country Status (10)

Country Link
US (1) US8383683B2 (cg-RX-API-DMAC7.html)
EP (1) EP2150109B1 (cg-RX-API-DMAC7.html)
JP (1) JP2010526777A (cg-RX-API-DMAC7.html)
CN (1) CN101711106B (cg-RX-API-DMAC7.html)
AR (1) AR066293A1 (cg-RX-API-DMAC7.html)
CA (1) CA2685036A1 (cg-RX-API-DMAC7.html)
CL (1) CL2008001197A1 (cg-RX-API-DMAC7.html)
ES (1) ES2393230T3 (cg-RX-API-DMAC7.html)
TW (1) TWI374871B (cg-RX-API-DMAC7.html)
WO (1) WO2008134221A1 (cg-RX-API-DMAC7.html)

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TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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CN102838505B (zh) * 2011-06-24 2016-02-17 上海医药工业研究院 酰胺类化合物、其制备方法及应用
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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JP2009530346A (ja) * 2006-03-21 2009-08-27 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー メタボリックシンドロームの治療用のアダマンタン誘導体
KR20090014347A (ko) * 2006-04-07 2009-02-10 하이 포인트 파마슈티칼스, 엘엘씨 11β-히드록시스테로이드 탈수소효소 타입 1 활성 화합물
JP2009539937A (ja) 2006-06-16 2009-11-19 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー 置換型ピペリジンカルボキサミドの医薬的使用
EP1878721A1 (en) 2006-07-13 2008-01-16 Novo Nordisk A/S 4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors
EP2129652A2 (en) 2007-02-23 2009-12-09 High Point Pharmaceuticals, LLC N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
US20110003856A1 (en) * 2007-02-23 2011-01-06 Soren Ebdrup N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
JP5243455B2 (ja) * 2007-02-23 2013-07-24 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー 新規化合物
JP2010519239A (ja) * 2007-02-23 2010-06-03 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー １１−ベータ−ヒドロキシステロイドデヒドロゲナーゼの阻害因子としてのｎ−アドマンチルベンザミド
CN101652359A (zh) * 2007-03-09 2010-02-17 高点制药有限责任公司 作为羟类固醇脱氢酶抑制剂的吲哚-和苯并咪唑酰胺类
JP2010522766A (ja) * 2007-03-28 2010-07-08 ハイ ポイント ファーマシューティカルズ，リミティド ライアビリティ カンパニー １１ベータ−ｈｓｄ１活性化合物
ES2399912T3 (es) * 2007-04-11 2013-04-04 High Point Pharmaceuticals, Llc Nuevos compuestos
WO2010059618A1 (en) * 2008-11-21 2010-05-27 High Point Pharmaceuticals, Llc Adamantyl benzamide compounds

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