DE602004025220D1 - Pharmazeutische verwendungen von kondensierten 1,2,4-triazolen - Google Patents

Pharmazeutische verwendungen von kondensierten 1,2,4-triazolen

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Publication number
DE602004025220D1
DE602004025220D1 DE602004025220T DE602004025220T DE602004025220D1 DE 602004025220 D1 DE602004025220 D1 DE 602004025220D1 DE 602004025220 T DE602004025220 T DE 602004025220T DE 602004025220 T DE602004025220 T DE 602004025220T DE 602004025220 D1 DE602004025220 D1 DE 602004025220D1
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DE
Germany
Prior art keywords
triazolene
condensed
11βhsd1
activity
pharmaceutical uses
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE602004025220T
Other languages
English (en)
Inventor
Henrik Sune Andersen
Gita Camilla Kampen
Inge Thoger Christensen
John Patrick Mogensen
Annette Rosendal Larsen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
vTv Therapeutics LLC
Original Assignee
High Point Pharnaceuticals LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by High Point Pharnaceuticals LLC filed Critical High Point Pharnaceuticals LLC
Publication of DE602004025220D1 publication Critical patent/DE602004025220D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

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WO2004089380A2 (en) 2004-10-21
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