JP2010523559A5 - - Google Patents
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- Publication number
- JP2010523559A5 JP2010523559A5 JP2010502079A JP2010502079A JP2010523559A5 JP 2010523559 A5 JP2010523559 A5 JP 2010523559A5 JP 2010502079 A JP2010502079 A JP 2010502079A JP 2010502079 A JP2010502079 A JP 2010502079A JP 2010523559 A5 JP2010523559 A5 JP 2010523559A5
- Authority
- JP
- Japan
- Prior art keywords
- phenoxy
- polymorph
- diethylamine
- chloro
- propyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US92196407P | 2007-04-05 | 2007-04-05 | |
| US92578607P | 2007-04-23 | 2007-04-23 | |
| PCT/US2008/003325 WO2008123914A1 (en) | 2007-04-05 | 2008-03-12 | Crystalline forms i and ii of [3-(4-{2-butyl-1-[4-(4-chloro-phenoxy)-phenyl]-1h-imidazol-4-yl}-phenoxy)-propyl]-diethyl-amine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010523559A JP2010523559A (ja) | 2010-07-15 |
| JP2010523559A5 true JP2010523559A5 (https=) | 2011-03-31 |
Family
ID=39469930
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010502079A Pending JP2010523559A (ja) | 2007-04-05 | 2008-03-12 | [3−(4−{2−ブチル−1−[4−(4−クロロ−フェノキシ)−フェニル]−1h−イミダゾール−4−イル}−フェノキシ)−プロピル]−ジエチルアミンの結晶形態 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US7884219B2 (https=) |
| EP (1) | EP2144883A1 (https=) |
| JP (1) | JP2010523559A (https=) |
| AR (1) | AR065896A1 (https=) |
| CA (1) | CA2681864A1 (https=) |
| CL (1) | CL2008000987A1 (https=) |
| PA (1) | PA8775601A1 (https=) |
| PE (1) | PE20090808A1 (https=) |
| TW (1) | TW200900384A (https=) |
| UY (1) | UY31004A1 (https=) |
| WO (1) | WO2008123914A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010523559A (ja) * | 2007-04-05 | 2010-07-15 | トランス テック ファーマ,インコーポレイテッド | [3−(4−{2−ブチル−1−[4−(4−クロロ−フェノキシ)−フェニル]−1h−イミダゾール−4−イル}−フェノキシ)−プロピル]−ジエチルアミンの結晶形態 |
| ES2467923T3 (es) | 2009-09-30 | 2014-06-13 | Transtech Pharma, Llc | Derivados de imidazol substituidos para el tratamiento de la enfermedad de Alzheimer |
| US9717710B2 (en) * | 2012-10-05 | 2017-08-01 | Vtv Therapeutics Llc | Treatment of mild and moderate Alzheimer's disease |
| HK1207004A1 (zh) * | 2012-10-05 | 2016-01-22 | Vtv治疗有限责任公司 | 治療輕度和中度阿爾茨海默病的方法 |
| CN103726005A (zh) * | 2012-10-16 | 2014-04-16 | 深圳富泰宏精密工业有限公司 | 珐琅涂层的制造方法及其制品 |
| WO2019190822A1 (en) * | 2018-03-28 | 2019-10-03 | Vtv Therapeutics Llc | Crystalline forms of [3-(4- {2-butyl-1-[4-(4-chloro-phenoxy)-phenyl]-1h-imidazol-4-yl} -phenoxy)-propyl]-diethyl-amine |
| WO2019190823A1 (en) | 2018-03-28 | 2019-10-03 | Vtv Therapeutics Llc | Pharmaceutically acceptable salts of [3-(4- {2-butyl-1-[4-(4-chlorophenoxy)-phenyl]-1h-imidazol-4-yl} -phenoxy)-propyl]-diethyl-amine |
| JP7464591B2 (ja) * | 2018-10-10 | 2024-04-09 | ブイティーブイ・セラピューティクス・エルエルシー | [3-(4-{2-ブチル-1-[4-(4-クロロ-フェノキシ)-フェニル]-1h-イミダゾール-4-イル}-フェノキシ)-プロピル]-ジエチル-アミンの代謝産物 |
| WO2020086388A1 (en) | 2018-10-22 | 2020-04-30 | Vtv Therapeutics Llc | Glucokinase activator compositions for the treatment of cognitive impairment |
| US11648235B1 (en) | 2022-12-30 | 2023-05-16 | Cantex Pharmaceuticals, Inc. | Treatment of glioblastoma |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4481011B2 (ja) | 2002-03-05 | 2010-06-16 | トランス テック ファーマ,インコーポレイテッド | リガンドのrageとの相互作用を阻害する単環式および二環式アゾール誘導体 |
| EP1635823A1 (en) * | 2003-05-20 | 2006-03-22 | TransTech Pharma Inc. | Rage antagonists as agents to reverse amyloidosis and diseases associated therewith |
| JP2010523559A (ja) * | 2007-04-05 | 2010-07-15 | トランス テック ファーマ,インコーポレイテッド | [3−(4−{2−ブチル−1−[4−(4−クロロ−フェノキシ)−フェニル]−1h−イミダゾール−4−イル}−フェノキシ)−プロピル]−ジエチルアミンの結晶形態 |
-
2008
- 2008-03-12 JP JP2010502079A patent/JP2010523559A/ja active Pending
- 2008-03-12 EP EP08726789A patent/EP2144883A1/en not_active Withdrawn
- 2008-03-12 CA CA002681864A patent/CA2681864A1/en not_active Withdrawn
- 2008-03-12 WO PCT/US2008/003325 patent/WO2008123914A1/en not_active Ceased
- 2008-03-12 US US12/046,872 patent/US7884219B2/en active Active
- 2008-03-19 TW TW097109673A patent/TW200900384A/zh unknown
- 2008-03-31 AR ARP080101342A patent/AR065896A1/es unknown
- 2008-04-04 PA PA20088775601A patent/PA8775601A1/es unknown
- 2008-04-04 PE PE2008000616A patent/PE20090808A1/es not_active Application Discontinuation
- 2008-04-04 UY UY31004A patent/UY31004A1/es not_active Application Discontinuation
- 2008-04-04 CL CL200800987A patent/CL2008000987A1/es unknown
-
2010
- 2010-12-30 US US12/982,775 patent/US8372988B2/en active Active
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