JP2010521529A5 - - Google Patents
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- Publication number
- JP2010521529A5 JP2010521529A5 JP2010500190A JP2010500190A JP2010521529A5 JP 2010521529 A5 JP2010521529 A5 JP 2010521529A5 JP 2010500190 A JP2010500190 A JP 2010500190A JP 2010500190 A JP2010500190 A JP 2010500190A JP 2010521529 A5 JP2010521529 A5 JP 2010521529A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- compound
- linear
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 CC(C*N(*)*)C(C)(*)N(*)S(*)=O Chemical compound CC(C*N(*)*)C(C)(*)N(*)S(*)=O 0.000 description 13
- PFLAVJKHIKGGHK-UHFFFAOYSA-N CCCON(C(CCN(C(c1ccccc11)=O)C1=O)C(NO)=O)S(=O)=O Chemical compound CCCON(C(CCN(C(c1ccccc11)=O)C1=O)C(NO)=O)S(=O)=O PFLAVJKHIKGGHK-UHFFFAOYSA-N 0.000 description 3
- FFRUPWBMVNXTRM-UHFFFAOYSA-N CN(C(C1)=O)C1=O Chemical compound CN(C(C1)=O)C1=O FFRUPWBMVNXTRM-UHFFFAOYSA-N 0.000 description 2
- KYEACNNYFNZCST-UHFFFAOYSA-N CN(C(CC1)=O)C1=O Chemical compound CN(C(CC1)=O)C1=O KYEACNNYFNZCST-UHFFFAOYSA-N 0.000 description 2
- VUYOLIKWIVQHBC-UHFFFAOYSA-N CN(C(CCC1)=O)C1=O Chemical compound CN(C(CCC1)=O)C1=O VUYOLIKWIVQHBC-UHFFFAOYSA-N 0.000 description 2
- ZXLYYQUMYFHCLQ-UHFFFAOYSA-N CN(C(c1ccccc11)=O)C1=O Chemical compound CN(C(c1ccccc11)=O)C1=O ZXLYYQUMYFHCLQ-UHFFFAOYSA-N 0.000 description 2
- QOEUNLQGZBSTBB-UHFFFAOYSA-N CN(CC1)C1=O Chemical compound CN(CC1)C1=O QOEUNLQGZBSTBB-UHFFFAOYSA-N 0.000 description 2
- SECXISVLQFMRJM-UHFFFAOYSA-N CN(CCC1)C1=O Chemical compound CN(CCC1)C1=O SECXISVLQFMRJM-UHFFFAOYSA-N 0.000 description 2
- GGYVTHJIUNGKFZ-UHFFFAOYSA-N CN(CCCC1)C1=O Chemical compound CN(CCCC1)C1=O GGYVTHJIUNGKFZ-UHFFFAOYSA-N 0.000 description 2
- WTFDPWXGUAWAFA-UHFFFAOYSA-N CCC(N1CCN(CCOCCON(C(CCN)C(NO)=O)S(=O)=O)CC1)=O Chemical compound CCC(N1CCN(CCOCCON(C(CCN)C(NO)=O)S(=O)=O)CC1)=O WTFDPWXGUAWAFA-UHFFFAOYSA-N 0.000 description 1
- GSOPZZSRFOGOGH-CQSZACIVSA-N CCCON(C)[C@H](CCNC(Cc1ccccc1)=O)C(NO)=O Chemical compound CCCON(C)[C@H](CCNC(Cc1ccccc1)=O)C(NO)=O GSOPZZSRFOGOGH-CQSZACIVSA-N 0.000 description 1
- GJHOOTVKVTXDQV-UHFFFAOYSA-N CCCON(CCCNC(OCc1ccccc1)=O)S(=O)=O Chemical compound CCCON(CCCNC(OCc1ccccc1)=O)S(=O)=O GJHOOTVKVTXDQV-UHFFFAOYSA-N 0.000 description 1
- UQVYNEKSBAKUEY-LJQANCHMSA-N CCCON([C@H](CCN)C(NO)=O)S(c(cc1)ccc1-c(cc1)ccc1OC)(=O)=O Chemical compound CCCON([C@H](CCN)C(NO)=O)S(c(cc1)ccc1-c(cc1)ccc1OC)(=O)=O UQVYNEKSBAKUEY-LJQANCHMSA-N 0.000 description 1
- DXLKWOUSKQECHN-XMMPIXPASA-N CCCON([C@H](CCNC(c1ccccc1)=O)C(NO)=O)S(c(cc1)ccc1-c1ccccc1)(=O)=O Chemical compound CCCON([C@H](CCNC(c1ccccc1)=O)C(NO)=O)S(c(cc1)ccc1-c1ccccc1)(=O)=O DXLKWOUSKQECHN-XMMPIXPASA-N 0.000 description 1
- UZICUEAGGHJDRC-WJOKGBTCSA-N COc(cc1)ccc1-c(cc1)ccc1S(N([C@H](CCNC(OCc1ccccc1)=O)C(O)=O)OCCOCCN1CCNCC1)(=O)=O Chemical compound COc(cc1)ccc1-c(cc1)ccc1S(N([C@H](CCNC(OCc1ccccc1)=O)C(O)=O)OCCOCCN1CCNCC1)(=O)=O UZICUEAGGHJDRC-WJOKGBTCSA-N 0.000 description 1
- ASDVEJMGKRLMQT-UHFFFAOYSA-N ONC(C(CCNC(OCc1ccccc1)=O)N(OCCOCCN1CCNCC1)S(=O)=O)=O Chemical compound ONC(C(CCNC(OCc1ccccc1)=O)N(OCCOCCN1CCNCC1)S(=O)=O)=O ASDVEJMGKRLMQT-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07104393A EP1972617A1 (en) | 2007-03-19 | 2007-03-19 | Compounds having aryl-sulphonamidic structure useful as metalloproteases inhibitors |
| PCT/EP2008/053078 WO2008113756A2 (en) | 2007-03-19 | 2008-03-14 | Compounds having aryl-sulphonamidic structure useful as metalloproteases inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010521529A JP2010521529A (ja) | 2010-06-24 |
| JP2010521529A5 true JP2010521529A5 (enExample) | 2011-04-28 |
Family
ID=38626433
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010500190A Pending JP2010521529A (ja) | 2007-03-19 | 2008-03-14 | メタロプロテアーゼ阻害剤として有用なアリール−スルホンアミド構造を有する化合物 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8329751B2 (enExample) |
| EP (2) | EP1972617A1 (enExample) |
| JP (1) | JP2010521529A (enExample) |
| KR (1) | KR20090121329A (enExample) |
| CN (1) | CN101610997A (enExample) |
| AU (1) | AU2008228260B2 (enExample) |
| CA (1) | CA2680239A1 (enExample) |
| IL (1) | IL200951A0 (enExample) |
| MX (1) | MX2009009409A (enExample) |
| RU (1) | RU2488580C2 (enExample) |
| WO (1) | WO2008113756A2 (enExample) |
| ZA (1) | ZA200905263B (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2149568A1 (en) | 2008-07-22 | 2010-02-03 | Bracco Imaging S.p.A | Aryl-sulphonamidic dimers as metalloproteases inhibitors |
| EP2147684A1 (en) * | 2008-07-22 | 2010-01-27 | Bracco Imaging S.p.A | Diagnostic Agents Selective Against Metalloproteases |
| US20240207415A1 (en) | 2022-11-08 | 2024-06-27 | Montelino Therapeutics, Inc. | Bi-functional compounds and methods for targeted ubiquitination of androgen receptor |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5058026A (enExample) * | 1973-09-26 | 1975-05-20 | ||
| IL137465A0 (en) * | 1998-02-04 | 2001-07-24 | Novartis Ag | Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases |
| HUP0102196A3 (en) * | 1998-04-03 | 2002-12-28 | Sankyo Company Ltd Chuo Ku | Sulfonamide derivatives |
| WO2006101828A1 (en) * | 2005-03-15 | 2006-09-28 | Bayer Cropscience Ag | Insecticidal alkylamino phenyl sulfonamide derivatives |
-
2007
- 2007-03-19 EP EP07104393A patent/EP1972617A1/en not_active Withdrawn
-
2008
- 2008-03-14 KR KR1020097019222A patent/KR20090121329A/ko not_active Ceased
- 2008-03-14 RU RU2009138346/04A patent/RU2488580C2/ru not_active IP Right Cessation
- 2008-03-14 CN CNA200880004727XA patent/CN101610997A/zh active Pending
- 2008-03-14 EP EP08717820A patent/EP2121590A2/en not_active Withdrawn
- 2008-03-14 MX MX2009009409A patent/MX2009009409A/es active IP Right Grant
- 2008-03-14 WO PCT/EP2008/053078 patent/WO2008113756A2/en not_active Ceased
- 2008-03-14 JP JP2010500190A patent/JP2010521529A/ja active Pending
- 2008-03-14 CA CA002680239A patent/CA2680239A1/en not_active Abandoned
- 2008-03-14 AU AU2008228260A patent/AU2008228260B2/en not_active Ceased
- 2008-03-14 US US12/531,119 patent/US8329751B2/en not_active Expired - Fee Related
-
2009
- 2009-07-05 ZA ZA200905263A patent/ZA200905263B/xx unknown
- 2009-09-15 IL IL200951A patent/IL200951A0/en unknown