JP2010520307A - エストロゲン関連受容体−アルファモジュレーターとしての置換フェノキシｎ−アルキル置換チアゾリジンジオン - Google Patents
エストロゲン関連受容体−アルファモジュレーターとしての置換フェノキシｎ−アルキル置換チアゾリジンジオン Download PDFInfo
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- JP2010520307A JP2010520307A JP2009552883A JP2009552883A JP2010520307A JP 2010520307 A JP2010520307 A JP 2010520307A JP 2009552883 A JP2009552883 A JP 2009552883A JP 2009552883 A JP2009552883 A JP 2009552883A JP 2010520307 A JP2010520307 A JP 2010520307A
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- ethyl
- phenoxy
- thiazolidine
- benzonitrile
- dioxo
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Classifications
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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Landscapes
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| PCT/US2008/056018 WO2008109731A2 (en) | 2007-03-07 | 2008-03-06 | Substituted phenoxy n-alkylated thiazoledinedione as estrogen related receptor-alpha modulators |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2021534254A (ja) * | 2018-08-22 | 2021-12-09 | ザ ジェイ． デビッド グラッドストーン インスティテューツ、 ア テスタメンタリー トラスト エスタブリッシュド アンダー ザ ウィル オブ ジェイ． デビッド グラッドストーン | 心臓弁疾患を治療するための方法 |
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| AR059898A1 (es) | 2006-03-15 | 2008-05-07 | Janssen Pharmaceutica Nv | Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2 |
| TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
| TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
| CN101679322A (zh) * | 2007-03-07 | 2010-03-24 | 詹森药业有限公司 | 用作雌激素相关性受体-α调节剂的取代苯氧基噻唑烷二酮类化合物 |
| BRPI0817101A2 (pt) | 2007-09-14 | 2017-05-09 | Addex Pharmaceuticals Sa | 4-(aril-x-fenil)-1h-piridin-2-onas 1,3-dissubstituídas |
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| JP2021534254A (ja) * | 2018-08-22 | 2021-12-09 | ザ ジェイ． デビッド グラッドストーン インスティテューツ、 ア テスタメンタリー トラスト エスタブリッシュド アンダー ザ ウィル オブ ジェイ． デビッド グラッドストーン | 心臓弁疾患を治療するための方法 |
| JP7476198B2 (ja) | 2018-08-22 | 2024-04-30 | ザ ジェイ． デビッド グラッドストーン インスティテューツ、 ア テスタメンタリー トラスト エスタブリッシュド アンダー ザ ウィル オブ ジェイ． デビッド グラッドストーン | 心臓弁疾患を治療するための医薬組成物 |
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| RS52247B (sr) | 2012-10-31 |
| CY1112778T1 (el) | 2016-02-10 |
| DK2132188T3 (da) | 2012-02-27 |
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| BRPI0808662B1 (pt) | 2020-09-29 |
| TW200902507A (en) | 2009-01-16 |
| WO2008109731A3 (en) | 2008-11-27 |
| KR20090118103A (ko) | 2009-11-17 |
| PT2132188E (pt) | 2012-02-13 |
| ZA200906953B (en) | 2010-12-29 |
| CN101679326A (zh) | 2010-03-24 |
| IL200758A0 (en) | 2010-05-17 |
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| SI2132188T1 (sl) | 2012-04-30 |
| US9034852B2 (en) | 2015-05-19 |
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| CA2679965A1 (en) | 2008-09-12 |
| ATE537157T1 (de) | 2011-12-15 |
| NZ579418A (en) | 2012-01-12 |
| AU2008222749A1 (en) | 2008-09-12 |
| BRPI0808662B8 (pt) | 2021-05-25 |
| MX2009009519A (es) | 2009-11-18 |
| PL2132188T3 (pl) | 2012-05-31 |
| BRPI0808662A2 (pt) | 2014-08-26 |
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| US20080286265A1 (en) | 2008-11-20 |
| US8119669B2 (en) | 2012-02-21 |
| CN101679326B (zh) | 2012-12-12 |
| US20120108571A1 (en) | 2012-05-03 |
| WO2008109731A2 (en) | 2008-09-12 |
| HRP20120160T1 (hr) | 2012-03-31 |
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