JP2010518094A5 - - Google Patents

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JP2010518094A5
JP2010518094A5 JP2009549133A JP2009549133A JP2010518094A5 JP 2010518094 A5 JP2010518094 A5 JP 2010518094A5 JP 2009549133 A JP2009549133 A JP 2009549133A JP 2009549133 A JP2009549133 A JP 2009549133A JP 2010518094 A5 JP2010518094 A5 JP 2010518094A5
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Japan
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alkanyl
aryl
alkynyl
alkenyl
heteroaryl
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JP2009549133A
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JP5511390B2 (ja
JP2010518094A (ja
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Priority claimed from PCT/US2008/001762 external-priority patent/WO2008100453A1/en
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Publication of JP2010518094A5 publication Critical patent/JP2010518094A5/ja
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JP2009549133A 2007-02-09 2008-02-07 ヘキソースおよびｎ−アセチルヘキソサミンの置換体を有する糖模倣体の使用方法 Expired - Fee Related JP5511390B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US90039807P 2007-02-09 2007-02-09
US60/900,398 2007-02-09
US93277907P 2007-05-31 2007-05-31
US60/932,779 2007-05-31
PCT/US2008/001762 WO2008100453A1 (en) 2007-02-09 2008-02-07 Methods of use of glycomimetics with replacements for hexoses and n-acetyl hexosamines

Publications (3)

Publication Number Publication Date
JP2010518094A JP2010518094A (ja) 2010-05-27
JP2010518094A5 true JP2010518094A5 (enExample) 2012-03-15
JP5511390B2 JP5511390B2 (ja) 2014-06-04

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JP2009549133A Expired - Fee Related JP5511390B2 (ja) 2007-02-09 2008-02-07 ヘキソースおよびｎ−アセチルヘキソサミンの置換体を有する糖模倣体の使用方法

Country Status (7)

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US (2) US8026222B2 (enExample)
EP (2) EP2117561A1 (enExample)
JP (1) JP5511390B2 (enExample)
AU (1) AU2008216794A1 (enExample)
CA (1) CA2677747A1 (enExample)
NZ (1) NZ598863A (enExample)
WO (1) WO2008100453A1 (enExample)

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JP2019524791A (ja) 2016-08-08 2019-09-05 グリコミメティクス， インコーポレイテッド Ｅ−セレクチンの阻害剤もしくはｃｘｃｒ４の阻害剤との、またはｅ−セレクチンおよびｃｘｃｒ４両方のヘテロ二機能性阻害剤とのｔ細胞チェックポイント阻害剤の組み合わせ
CN109890421B (zh) 2016-10-07 2023-10-20 糖模拟物有限公司 高效的多聚体e-选择蛋白拮抗剂
US11197877B2 (en) 2017-03-15 2021-12-14 Glycomimetics. Inc. Galactopyranosyl-cyclohexyl derivauves as E-selectin antagonists
US11712446B2 (en) 2017-11-30 2023-08-01 Glycomimetics, Inc. Methods of mobilizing marrow infiltrating lymphocytes and uses thereof
EP3732186A1 (en) 2017-12-29 2020-11-04 GlycoMimetics, Inc. Heterobifunctional inhibitors of e-selectin and galectin-3
KR20200128025A (ko) 2018-03-05 2020-11-11 글리코미메틱스, 인크. 급성 골수성 백혈병 및 관련 병태의 치료 방법
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