JP2010503695A5 - - Google Patents

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Publication number
JP2010503695A5
JP2010503695A5 JP2009528434A JP2009528434A JP2010503695A5 JP 2010503695 A5 JP2010503695 A5 JP 2010503695A5 JP 2009528434 A JP2009528434 A JP 2009528434A JP 2009528434 A JP2009528434 A JP 2009528434A JP 2010503695 A5 JP2010503695 A5 JP 2010503695A5
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JP
Japan
Prior art keywords
benzonitrile
dioxo
pyrimidin
piperidin
ylmethyl
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JP2009528434A
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English (en)
Japanese (ja)
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JP5791228B2 (ja
JP2010503695A (ja
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Priority claimed from PCT/US2006/035958 external-priority patent/WO2007033350A1/en
Application filed filed Critical
Priority claimed from PCT/US2007/078177 external-priority patent/WO2008033851A2/en
Publication of JP2010503695A publication Critical patent/JP2010503695A/ja
Publication of JP2010503695A5 publication Critical patent/JP2010503695A5/ja
Application granted granted Critical
Publication of JP5791228B2 publication Critical patent/JP5791228B2/ja
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JP2009528434A 2006-09-13 2007-09-11 2−6−(3−アミノ−ピペリジン−1−イル)−3−メチル−2,4−ジオキソ−3,4−ジヒドロ−2h−ピリミジン−1−イルメチル−4−フルオロ−ベンゾニトリルの使用 Active JP5791228B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
PCT/US2006/035958 WO2007033350A1 (en) 2005-09-14 2006-09-13 Dipeptidyl peptidase inhibitors for treating diabetes
USPCT/US2006/035958 2006-09-13
US89462807P 2007-03-13 2007-03-13
US60/894,628 2007-03-13
PCT/US2007/078177 WO2008033851A2 (en) 2006-09-13 2007-09-11 Use of 2-6- (3-amino-piperidin-l-yl) -3-methyl-2, 4-dioxo-3, 4-dihydr0-2h-pyrimidin-1-ylmet hyl-4-fluoro-benzonitrile

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015020882A Division JP2015129143A (ja) 2006-09-13 2015-02-05 2−6−(3−アミノ−ピペリジン−1−イル)−3−メチル−2,4−ジオキソ−3,4−ジヒドロ−2h−ピリミジン−1−イルメチル−4−フルオロ−ベンゾニトリルの使用

Publications (3)

Publication Number Publication Date
JP2010503695A JP2010503695A (ja) 2010-02-04
JP2010503695A5 true JP2010503695A5 (enExample) 2010-10-28
JP5791228B2 JP5791228B2 (ja) 2015-10-07

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Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009528434A Active JP5791228B2 (ja) 2006-09-13 2007-09-11 2−6−(3−アミノ−ピペリジン−1−イル)−3−メチル−2,4−ジオキソ−3,4−ジヒドロ−2h−ピリミジン−1−イルメチル−4−フルオロ−ベンゾニトリルの使用
JP2015020882A Pending JP2015129143A (ja) 2006-09-13 2015-02-05 2−6−(3−アミノ−ピペリジン−1−イル)−3−メチル−2,4−ジオキソ−3,4−ジヒドロ−2h−ピリミジン−1−イルメチル−4−フルオロ−ベンゾニトリルの使用

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JP2015020882A Pending JP2015129143A (ja) 2006-09-13 2015-02-05 2−6−(3−アミノ−ピペリジン−1−イル)−3−メチル−2,4−ジオキソ−3,4−ジヒドロ−2h−ピリミジン−1−イルメチル−4−フルオロ−ベンゾニトリルの使用

Country Status (34)

Country Link
US (2) US20080287476A1 (enExample)
EP (1) EP2073810B1 (enExample)
JP (2) JP5791228B2 (enExample)
KR (4) KR20150032590A (enExample)
CN (2) CN101616673A (enExample)
AR (2) AR062760A1 (enExample)
AT (1) ATE522216T1 (enExample)
AU (1) AU2007296556B2 (enExample)
BR (1) BRPI0716971A2 (enExample)
CA (1) CA2663279C (enExample)
CL (1) CL2007002649A1 (enExample)
CO (1) CO6160321A2 (enExample)
CY (1) CY1112292T1 (enExample)
DK (1) DK2073810T3 (enExample)
EA (1) EA017799B1 (enExample)
EC (1) ECSP099250A (enExample)
ES (1) ES2370873T3 (enExample)
GE (1) GEP20125701B (enExample)
HR (1) HRP20110800T1 (enExample)
IL (1) IL197502A (enExample)
JO (1) JO2755B1 (enExample)
MA (1) MA30725B1 (enExample)
MX (1) MX2009002772A (enExample)
MY (1) MY145447A (enExample)
NO (1) NO342004B1 (enExample)
NZ (1) NZ575521A (enExample)
PE (1) PE20081150A1 (enExample)
PL (1) PL2073810T3 (enExample)
PT (1) PT2073810E (enExample)
RS (1) RS51965B (enExample)
SI (1) SI2073810T1 (enExample)
TN (1) TN2009000079A1 (enExample)
TW (1) TWI434838B (enExample)
WO (1) WO2008033851A2 (enExample)

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CN103816158A (zh) 2008-08-15 2014-05-28 勃林格殷格翰国际有限公司 用于治疗fab-相关疾病的嘌呤衍生物
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