JP2009542678A5 - - Google Patents

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Publication number
JP2009542678A5
JP2009542678A5 JP2009518301A JP2009518301A JP2009542678A5 JP 2009542678 A5 JP2009542678 A5 JP 2009542678A5 JP 2009518301 A JP2009518301 A JP 2009518301A JP 2009518301 A JP2009518301 A JP 2009518301A JP 2009542678 A5 JP2009542678 A5 JP 2009542678A5
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JP
Japan
Prior art keywords
disintegrant
api
ratio
tablet
dissolution rate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009518301A
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English (en)
Japanese (ja)
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JP2009542678A (ja
JP5116764B2 (ja
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Application filed filed Critical
Priority claimed from PCT/US2007/015168 external-priority patent/WO2008005353A2/en
Publication of JP2009542678A publication Critical patent/JP2009542678A/ja
Publication of JP2009542678A5 publication Critical patent/JP2009542678A5/ja
Application granted granted Critical
Publication of JP5116764B2 publication Critical patent/JP5116764B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2009518301A 2006-06-30 2007-06-29 トロンビン受容体拮抗薬の即放性錠剤製剤 Expired - Fee Related JP5116764B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81782106P 2006-06-30 2006-06-30
US60/817,821 2006-06-30
PCT/US2007/015168 WO2008005353A2 (en) 2006-06-30 2007-06-29 Immediate-release tablet formulations of a thrombin receptor antagonist

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012082021A Division JP2012126752A (ja) 2006-06-30 2012-03-30 トロンビン受容体拮抗薬の即放性錠剤製剤

Publications (3)

Publication Number Publication Date
JP2009542678A JP2009542678A (ja) 2009-12-03
JP2009542678A5 true JP2009542678A5 (https=) 2010-05-13
JP5116764B2 JP5116764B2 (ja) 2013-01-09

Family

ID=38895141

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009518301A Expired - Fee Related JP5116764B2 (ja) 2006-06-30 2007-06-29 トロンビン受容体拮抗薬の即放性錠剤製剤
JP2012082021A Withdrawn JP2012126752A (ja) 2006-06-30 2012-03-30 トロンビン受容体拮抗薬の即放性錠剤製剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012082021A Withdrawn JP2012126752A (ja) 2006-06-30 2012-03-30 トロンビン受容体拮抗薬の即放性錠剤製剤

Country Status (18)

Country Link
US (2) US20080031943A1 (https=)
EP (2) EP2491922B1 (https=)
JP (2) JP5116764B2 (https=)
KR (1) KR20090023670A (https=)
CN (2) CN104922054A (https=)
AR (1) AR061790A1 (https=)
AU (1) AU2007269733B2 (https=)
BR (1) BRPI0713935A2 (https=)
CA (1) CA2656395C (https=)
CL (1) CL2007001923A1 (https=)
CO (1) CO6150126A2 (https=)
ES (2) ES2616405T3 (https=)
MX (1) MX2009000131A (https=)
NO (1) NO20090467L (https=)
PE (1) PE20080376A1 (https=)
TW (1) TWI367112B (https=)
WO (1) WO2008005353A2 (https=)
ZA (1) ZA200900350B (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI343262B (en) * 2006-09-26 2011-06-11 Schering Corp Rapidly disintegrating lyophilized oral formulations of a thrombin receptor antagonist
EP2120879A2 (en) * 2006-12-22 2009-11-25 Schering Corporation Disintegration promoters in solid dose wet granulation formulations
US8624050B2 (en) * 2007-06-22 2014-01-07 General Electric Company Solution process for transparent conductive oxide coatings
WO2009078999A1 (en) 2007-12-17 2009-06-25 Janssen Pharmaceutica N.V. Imidazolo-, oxazolo-, and thiazolopyrimidine modulators of trpv1
EP2438060B1 (en) 2009-06-04 2013-10-02 Merck Sharp & Dohme Corp. Active metabolite of a thrombin receptor antagonist
JP2012529431A (ja) 2009-06-08 2012-11-22 メルク・シャープ・アンド・ドーム・コーポレーション トロンビン受容体アンタゴニストおよびクロピドグレルの固定用量錠剤
CN102442965B (zh) * 2010-09-30 2013-12-11 天津药物研究院 用于治疗血栓性疾病的par-1拮抗剂及其制备方法和用途
WO2017134200A1 (en) 2016-02-05 2017-08-10 Sanovel Ilac Sanayi Ve Ticaret A.S. A novel pharmaceutical composition of vorapaxar and metoprolol
TR201601548A2 (tr) 2016-02-05 2018-03-21 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Vorapaksar ve metoprololün bi̇r farmasöti̇k kompozi̇syonu
MX2020008137A (es) * 2018-02-02 2020-10-19 Eustralis Pharmaceuticals Ltd Trading As Pressura Neuro Formulaciones orales y usos de las mismas.

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61137813A (ja) * 1984-12-07 1986-06-25 Sawai Seiyaku Kk 持続性セフラジン製剤
JPS63162620A (ja) * 1986-12-25 1988-07-06 Teisan Seiyaku Kk 遅溶性顆粒及びそれを用いた持続性複合顆粒
GB9414045D0 (en) * 1994-07-12 1994-08-31 Berwind Pharma Service Moisture barrier film coating composition, method, and coated form
US20010003588A1 (en) * 1996-09-12 2001-06-14 Smithkline Beecham Corporation Controlled release dosage form of [R-(Z)]-alpha-(methoxyimino)-alpha-(1-azabicyclo[2.2.2.]oct-3-yl)acetonitrile monohydrochloride
JPH10130142A (ja) * 1996-10-31 1998-05-19 Zensei Yakuhin Kogyo Kk 放出持続型圧縮製剤
JPH10298062A (ja) * 1997-04-24 1998-11-10 Pfizer Pharmaceut Co Ltd 口腔内速溶型錠剤
CZ298578B6 (cs) * 1997-11-25 2007-11-14 Schering Corporation Heterocyklickou skupinou substituovaná tricyklická sloucenina a farmaceutický prostredek ji obsahující
US6063847A (en) * 1997-11-25 2000-05-16 Schering Corporation Thrombin receptor antagonists
WO2001000656A2 (en) 1999-06-29 2001-01-04 Ortho-Mcneil Pharmaceutical, Inc. Novel indazole peptidomimetics as thrombin receptor antagonists
US6630451B1 (en) 1999-06-29 2003-10-07 Orthomcneil Pharmaceutical, Inc. Benzimidazolone peptidometics as thrombin receptor antagonist
US6858577B1 (en) 1999-06-29 2005-02-22 Ortho-Mcneil Pharmaceutical, Inc. Indole peptidomimetics as thrombin receptor antagonists
US7488742B2 (en) 2000-06-15 2009-02-10 Schering Corporation Thrombin receptor antagonists
AU6690001A (en) * 2000-06-15 2001-12-24 Schering Corp Thrombin receptor antagonists
US7235567B2 (en) * 2000-06-15 2007-06-26 Schering Corporation Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
US20040192753A1 (en) * 2000-06-15 2004-09-30 Samuel Chackalamannil Methods of use of thrombin receptor antagonists
WO2002068425A1 (en) * 2001-02-23 2002-09-06 Ortho-Mcneil Pharmaceutical, Inc. Aminomethyl-pyrroloquinazoline compounds as thrombin receptor antagonists
EP1394152A4 (en) 2001-04-19 2005-02-02 Eisai Co Ltd 2-IMINOIMIDAZOLE DERIVATIVES (1)
KR100960170B1 (ko) * 2001-10-18 2010-05-26 쉐링 코포레이션 트롬빈 수용체 길항제로서의 힘바신 동족체
BRPI0309309B8 (pt) * 2002-04-16 2021-05-25 Merck Sharp & Dohme antagonistas de receptor de trombina tricíclicos
DE10317816A1 (de) * 2003-04-16 2004-11-04 Claas Selbstfahrende Erntemaschinen Gmbh Feldhäcksler mit positionierbarer Fahrerkabine
CZ300438B6 (cs) * 2003-11-25 2009-05-20 Pliva Hrvatska D.O.O. Zpusob prípravy orální pevné lékové formy s okamžitým uvolnováním úcinné látky obsahující jako úcinnou látku polymorfní formu finasteridu
JP2009521472A (ja) * 2005-12-22 2009-06-04 シェーリング コーポレイション 心肺手術の合併症の予防としてのトロンビンレセプターアンタゴニスト
TW200812619A (en) * 2006-04-06 2008-03-16 Schering Corp TRA combination therapies
US20080026050A1 (en) * 2006-06-30 2008-01-31 Rajan Gupta Solid dose formulations of a thrombin receptor antagonist
TWI343262B (en) * 2006-09-26 2011-06-11 Schering Corp Rapidly disintegrating lyophilized oral formulations of a thrombin receptor antagonist
EP2120879A2 (en) * 2006-12-22 2009-11-25 Schering Corporation Disintegration promoters in solid dose wet granulation formulations
BRPI0809095A2 (pt) * 2007-03-23 2014-09-09 Schering Corp Redução de eventos adversos após intervenção percutânea através de uso de um antagonista de receptor de trombina

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