|
US20100137330A1
(en)
*
|
2007-03-08 |
2010-06-03 |
Ratan Bhat |
Use
|
|
WO2010054398A1
(en)
|
2008-11-10 |
2010-05-14 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
AU2009327357C1
(en)
|
2008-12-19 |
2017-02-02 |
Vertex Pharmaceuticals Incorporated |
Pyrazine derivatives useful as inhibitors of ATR kinase
|
|
WO2011089416A1
(en)
*
|
2010-01-19 |
2011-07-28 |
Astrazeneca Ab |
Pyrazine derivatives
|
|
WO2011143399A1
(en)
|
2010-05-12 |
2011-11-17 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
WO2011143423A2
(en)
|
2010-05-12 |
2011-11-17 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
MX2012013081A
(es)
|
2010-05-12 |
2013-05-09 |
Vertex Pharma |
Compuestos utiles como inhibidores de cinasa atr.
|
|
JP2013526540A
(ja)
|
2010-05-12 |
2013-06-24 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Atrキナーゼ阻害剤として有用な化合物
|
|
WO2011143422A1
(en)
|
2010-05-12 |
2011-11-17 |
Vertex Pharmaceuticals Incorporated |
2 -aminopyridine derivatives useful as inhibitors of atr kinase
|
|
US8962631B2
(en)
|
2010-05-12 |
2015-02-24 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
|
US8623869B2
(en)
|
2010-06-23 |
2014-01-07 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
|
MX2013011450A
(es)
|
2011-04-05 |
2014-02-03 |
Vertex Pharma |
Compuestos de aminopirazina utiles como inhibidores de la cinasa ataxia telangiectasia mutada y rad3 relacionados (atr).
|
|
PL2714677T3
(pl)
*
|
2011-05-23 |
2019-02-28 |
Merck Patent Gmbh |
Pochodne pirydynowe i pirazynowe
|
|
JP2014517079A
(ja)
|
2011-06-22 |
2014-07-17 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Atrキナーゼ阻害剤として有用な化合物
|
|
WO2012178123A1
(en)
|
2011-06-22 |
2012-12-27 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
US9096602B2
(en)
|
2011-06-22 |
2015-08-04 |
Vertex Pharmaceuticals Incorporated |
Substituted pyrrolo[2,3-B]pyrazines as ATR kinase inhibitors
|
|
EP2751088B1
(en)
|
2011-09-30 |
2016-04-13 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
RS59337B1
(sr)
|
2011-09-30 |
2019-10-31 |
Vertex Pharma |
Postupak za izradu jedinjenja, korisnih kao inhibitori atr kinaze
|
|
EP2751099B1
(en)
|
2011-09-30 |
2017-06-14 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
SG11201401095YA
(en)
|
2011-09-30 |
2014-04-28 |
Vertex Pharma |
Treating pancreatic cancer and non-small cell lung cancer with atr inhibitors
|
|
WO2013049720A1
(en)
|
2011-09-30 |
2013-04-04 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
US8846917B2
(en)
|
2011-11-09 |
2014-09-30 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
|
EP2776419B1
(en)
|
2011-11-09 |
2016-05-11 |
Vertex Pharmaceuticals Incorporated |
Pyrazine compounds useful as inhibitors of atr kinase
|
|
US8841450B2
(en)
|
2011-11-09 |
2014-09-23 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of ATR kinase
|
|
EP2776429A1
(en)
|
2011-11-09 |
2014-09-17 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
WO2013071090A1
(en)
|
2011-11-09 |
2013-05-16 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
ES2654670T3
(es)
|
2012-04-05 |
2018-02-14 |
Vertex Pharmaceuticals Incorporated |
Compuestos útiles como inhibidores de la cinasa ATR y terapias de combinación de los mismos
|
|
WO2014055756A1
(en)
|
2012-10-04 |
2014-04-10 |
Vertex Pharmaceuticals Incorporated |
Method for measuring atr inhibition mediated increases in dna damage
|
|
EP2909202A1
(en)
|
2012-10-16 |
2015-08-26 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of atr kinase
|
|
PT4190786T
(pt)
|
2012-12-07 |
2025-05-29 |
Vertex Pharma |
Compostos úteis como inibidores da quinase atr
|
|
CA3184040A1
(en)
|
2013-03-14 |
2014-10-02 |
The Brigham And Women's Hospital, Inc. |
Compositions and methods for epithelial stem cell expansion comprising a wnt agonist and a histone deacetylase inhibitor
|
|
EP2970286A1
(en)
|
2013-03-15 |
2016-01-20 |
Vertex Pharmaceuticals Inc. |
Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase
|
|
CA2932757C
(en)
|
2013-12-06 |
2023-10-31 |
Vertex Pharmaceuticals Incorporated |
2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, its preparation, different solid forms and radiolabelled derivatives thereof
|
|
CN103804312B
(zh)
*
|
2014-02-17 |
2016-04-20 |
四川百利药业有限责任公司 |
一类氮杂环化合物及其制备方法和用途
|
|
KR102575125B1
(ko)
|
2014-06-05 |
2023-09-07 |
버텍스 파마슈티칼스 인코포레이티드 |
Atr 키나제의 저해제로서 유용한 2-아미노-6-플루오로-n-[5-플루오로-피리딘-3-일]-피라졸로[1,5-a]피리미딘-3-카복스아미드 화합물의 방사성표지된 유도체, 상기 화합물의 제조 및 이의 다양한 고체 형태
|
|
RU2736219C2
(ru)
|
2014-06-17 |
2020-11-12 |
Вертекс Фармасьютикалз Инкорпорейтед |
Способ лечения рака с использованием комбинации ингибиторов снк1 и atr
|
|
WO2016037016A1
(en)
|
2014-09-03 |
2016-03-10 |
The Brigham And Women's Hospital, Inc. |
Compositions, systems, and methods for generating inner ear hair cells for treatment of hearing loss
|
|
AU2016331955B2
(en)
|
2015-09-30 |
2022-07-21 |
Vertex Pharmaceuticals Incorporated |
Method for treating cancer using a combination of DNA damaging agents and ATR inhibitors
|
|
AU2017205194A1
(en)
|
2016-01-08 |
2018-07-19 |
Massachusetts Institute Of Technology |
Production of differentiated enteroendocrine cells and insulin producing cells
|
|
US11260130B2
(en)
|
2016-03-02 |
2022-03-01 |
Frequency Therapeutics, Inc. |
Solubilized compositions for controlled proliferation of stem cells / generating inner ear hair cells using a GSK3 inhibitor: IV
|
|
US10201540B2
(en)
|
2016-03-02 |
2019-02-12 |
Frequency Therapeutics, Inc. |
Solubilized compositions for controlled proliferation of stem cells / generating inner ear hair cells using GSK3 inhibitors: I
|
|
US10213511B2
(en)
|
2016-03-02 |
2019-02-26 |
Frequency Therapeutics, Inc. |
Thermoreversible compositions for administration of therapeutic agents
|
|
CN110392686A
(zh)
|
2016-12-30 |
2019-10-29 |
频率治疗公司 |
1h-吡咯-2,5-二酮化合物以及使用它们来诱导干/祖支持细胞自我更新的方法
|
|
US11162071B2
(en)
|
2018-08-17 |
2021-11-02 |
Frequency Therapeutics, Inc. |
Compositions and methods for generating hair cells by upregulating JAG-1
|
|
WO2020037326A1
(en)
|
2018-08-17 |
2020-02-20 |
Frequency Therapeutics, Inc. |
Compositions and methods for generating hair cells by downregulating foxo
|
|
JP2022520671A
(ja)
|
2019-02-08 |
2022-03-31 |
フリークエンシー・セラピューティクス・インコーポレイテッド |
耳障害を治療するためのバルプロ酸化合物及びwnt作動薬
|
|
AU2024294424A1
(en)
*
|
2023-07-14 |
2025-11-20 |
Jazz Pharmaceuticals Therapeutics, Inc. |
Methods of use of a liposomal composition comprising an atr inhibitor
|