JP2008525513A5 - - Google Patents

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Publication number
JP2008525513A5
JP2008525513A5 JP2007548747A JP2007548747A JP2008525513A5 JP 2008525513 A5 JP2008525513 A5 JP 2008525513A5 JP 2007548747 A JP2007548747 A JP 2007548747A JP 2007548747 A JP2007548747 A JP 2007548747A JP 2008525513 A5 JP2008525513 A5 JP 2008525513A5
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JP
Japan
Prior art keywords
substituted
unsubstituted
compound
formula
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007548747A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008525513A (ja
Filing date
Publication date
Priority claimed from EP04380279A external-priority patent/EP1676844A1/en
Application filed filed Critical
Publication of JP2008525513A publication Critical patent/JP2008525513A/ja
Publication of JP2008525513A5 publication Critical patent/JP2008525513A5/ja
Pending legal-status Critical Current

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JP2007548747A 2004-12-28 2005-12-27 5−ht7受容体拮抗薬 Pending JP2008525513A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04380279A EP1676844A1 (en) 2004-12-28 2004-12-28 5-HT7 receptor antagonists
US11/048,992 US7345057B2 (en) 2004-12-28 2005-02-02 5-HT7 receptor antagonists
PCT/EP2005/014046 WO2006069776A1 (en) 2004-12-28 2005-12-27 5-ht7 receptor antagonists

Publications (2)

Publication Number Publication Date
JP2008525513A JP2008525513A (ja) 2008-07-17
JP2008525513A5 true JP2008525513A5 (enExample) 2009-02-12

Family

ID=34931894

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007548747A Pending JP2008525513A (ja) 2004-12-28 2005-12-27 5−ht7受容体拮抗薬

Country Status (11)

Country Link
US (1) US7345057B2 (enExample)
EP (2) EP1676844A1 (enExample)
JP (1) JP2008525513A (enExample)
KR (1) KR20070091040A (enExample)
CN (1) CN101090898A (enExample)
AU (1) AU2005321463A1 (enExample)
BR (1) BRPI0519792A2 (enExample)
CA (1) CA2590666A1 (enExample)
MX (1) MX2007007894A (enExample)
RU (1) RU2007128926A (enExample)
WO (1) WO2006069776A1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2005274927B2 (en) 2004-07-15 2011-11-03 Albany Molecular Research, Inc. Aryl-and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
WO2008064329A1 (en) * 2006-11-21 2008-05-29 University Of Tennessee Research Foundation Therapeutic tetrahydroisoquinoline-based compositions for cancer therapy
DK2155717T3 (da) * 2007-05-11 2012-11-19 Lilly Co Eli 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl-pyraziner og -pyridiner og 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl-pyridiner som 5-ht7-receptorantagonister
US9156812B2 (en) 2008-06-04 2015-10-13 Bristol-Myers Squibb Company Crystalline form of 6-[(4S)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine
EP2375899B1 (en) * 2009-01-12 2015-02-25 Array Biopharma Inc. Piperidine-containing compounds and use thereof in the treatment of diabetes
US8802696B2 (en) * 2009-05-12 2014-08-12 Albany Molecular Research, Inc. 7-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydroisoqu inoli and use thereof
WO2010132487A1 (en) 2009-05-12 2010-11-18 Bristol-Myers Squibb Company CRYSTALLINE FORMS OF (S)-7-([1,2,4]TRIAZOLO[1,5-a]PYRIDIN-6-YL)-4-(3,4-DICHLOROHPHENYL)-1,2,3,4-TETRAHYDROISOQUINOLINE AND USE THEREOF
CN102458123A (zh) * 2009-05-12 2012-05-16 阿尔巴尼分子研究公司 芳基、杂芳基和杂环取代的四氢异喹啉及其用途
GB201209587D0 (en) 2012-05-30 2012-07-11 Takeda Pharmaceutical Therapeutic compounds
US10208016B2 (en) 2013-06-21 2019-02-19 Takeda Pharmaceutical Company Limited 1-sulfonyl piperidine derivatives as modulators of prokineticin receptors
GB201420095D0 (en) 2014-11-12 2014-12-24 Takeda Pharmaceutical New use
US11505529B2 (en) * 2017-03-03 2022-11-22 National Taiwan University 8-phenyl-isoquinolines and pharmaceutical composition thereof used in the treatment of irritable bowel syndrome
WO2018165520A1 (en) 2017-03-10 2018-09-13 Vps-3, Inc. Metalloenzyme inhibitor compounds
WO2021021979A2 (en) 2019-07-30 2021-02-04 Eikonizo Therapapeutics, Inc. Hdac6 inhibitors and uses thereof
CN112083107B (zh) * 2020-09-28 2022-07-05 中国计量科学研究院 检测蜂蜜基质中磺胺类药物葡萄糖醛酸结合物的方法
EP4504190A4 (en) 2022-04-08 2026-03-25 Eikonizo Therapeutics Inc OXADIAZOLE HDAC6 INHIBITORS AND THEIR USES

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ193654A (en) 1979-05-16 1984-08-24 Wuelfing Johann A Naphthalene sulphonamido-alkyl-piperidines,pyrrolidines or piperazines and pharmaceutical compositions
EP0076072B1 (en) 1981-09-24 1987-05-13 BEECHAM - WUELFING GmbH & Co. KG Sulphonamides
WO1997029097A1 (en) 1996-02-09 1997-08-14 Smithkline Beecham Plc Sulfonamide derivatives as 5ht7 receptor antagonists
GB9612884D0 (en) 1996-06-20 1996-08-21 Smithkline Beecham Plc Novel compounds
WO1997049695A1 (en) * 1996-06-25 1997-12-31 Smithkline Beecham P.L.C. Sulfonamide derivatives as 5ht7 receptor antagonists
AU1558899A (en) 1997-11-10 1999-05-31 F. Hoffmann-La Roche Ag Isoquinoline derivatives for use against cns disorders
WO2000000472A1 (en) * 1998-06-30 2000-01-06 Du Pont Pharmaceuticals Company 5-ht7 receptor antagonists
GB0128885D0 (en) 2001-12-03 2002-01-23 Merck Sharp & Dohme Therapeutic agents

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