JP2008525502A5 - - Google Patents

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Publication number
JP2008525502A5
JP2008525502A5 JP2007548611A JP2007548611A JP2008525502A5 JP 2008525502 A5 JP2008525502 A5 JP 2008525502A5 JP 2007548611 A JP2007548611 A JP 2007548611A JP 2007548611 A JP2007548611 A JP 2007548611A JP 2008525502 A5 JP2008525502 A5 JP 2008525502A5
Authority
JP
Japan
Prior art keywords
phenyl
pyrazol
urea
dichlorophenyl
oxoethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2007548611A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008525502A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/047597 external-priority patent/WO2006081034A2/en
Publication of JP2008525502A publication Critical patent/JP2008525502A/ja
Publication of JP2008525502A5 publication Critical patent/JP2008525502A5/ja
Abandoned legal-status Critical Current

Links

JP2007548611A 2004-12-23 2005-12-23 抗炎症薬 Abandoned JP2008525502A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63898704P 2004-12-23 2004-12-23
PCT/US2005/047597 WO2006081034A2 (en) 2004-12-23 2005-12-23 Anti-inflammatory medicaments

Publications (2)

Publication Number Publication Date
JP2008525502A JP2008525502A (ja) 2008-07-17
JP2008525502A5 true JP2008525502A5 (https=) 2009-01-29

Family

ID=36740941

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007548611A Abandoned JP2008525502A (ja) 2004-12-23 2005-12-23 抗炎症薬

Country Status (6)

Country Link
US (1) US20090312349A1 (https=)
EP (1) EP1836173A4 (https=)
JP (1) JP2008525502A (https=)
AU (1) AU2005325676A1 (https=)
CA (1) CA2592116A1 (https=)
WO (1) WO2006081034A2 (https=)

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US20110189167A1 (en) * 2007-04-20 2011-08-04 Flynn Daniel L Methods and Compositions for the Treatment of Myeloproliferative Diseases and other Proliferative Diseases
EA019524B1 (ru) 2007-05-04 2014-04-30 Айрм Ллк СОЕДИНЕНИЯ И КОМПОЗИЦИИ КАК ИНГИБИТОРЫ КИНАЗЫ с-kit И PDGFR
US8293757B2 (en) 2007-08-22 2012-10-23 Irm Llc 5-(4-(haloalkoxy)phenyl) pyrimidine-2-amine compounds and compositions as kinase inhibitors
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GB0905955D0 (en) 2009-04-06 2009-05-20 Respivert Ltd Novel compounds
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US8461179B1 (en) 2012-06-07 2013-06-11 Deciphera Pharmaceuticals, Llc Dihydronaphthyridines and related compounds useful as kinase inhibitors for the treatment of proliferative diseases
WO2014078417A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
RS55593B1 (sr) 2012-11-13 2017-06-30 Array Biopharma Inc Jedinjenja biciklične uree, tiouree, guanidina i cijanoguanidina korisna za lečenje bola
WO2014078331A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(arylalkyl)-n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9822118B2 (en) 2012-11-13 2017-11-21 Array Biopharma Inc. Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
WO2014078325A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(monocyclic aryl),n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9981959B2 (en) 2012-11-13 2018-05-29 Array Biopharma Inc. Thiazolyl and oxazolyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
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MX374242B (es) 2012-11-13 2025-03-05 Array Biopharma Inc Compuestos de n-pirrolidinil, n' -pirazolil-urea, tiourea, guanidina y cianoguanidina como inhibidores de trka cinasa.
MA40434B1 (fr) 2014-05-15 2019-09-30 Array Biopharma Inc 1-((3s,4r)-4-(3-fluorophényl)-1-(2-méthoxyéthyl)pyrrolidin-3-yl)-3-(4-méthyl-3-(2-méthylpyrimidin-5-yl)-1-phényl-1h-pyrazol-5-yl)urée comme inhibiteur de la kinase trka
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CN118416236A (zh) 2018-01-31 2024-08-02 德西费拉制药有限责任公司 治疗胃肠道间质瘤的组合疗法
IL276398B2 (en) 2018-01-31 2026-03-01 Deciphera Pharmaceuticals Llc Combination therapy for mastocytosis
WO2019241311A1 (en) * 2018-06-11 2019-12-19 Northeastern University Selective ligands for modulation of girk channels
CN109134451A (zh) * 2018-09-10 2019-01-04 遵义医学院 1,3-二取代脲类与硫脲类衍生物及其应用
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CN109456280B (zh) * 2018-12-24 2020-11-10 锦州医科大学 含有脲结构的4-苯基噻唑-2-胺类衍生物及其制备方法与应用
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CN114641466B (zh) 2019-06-12 2025-09-30 诺瑟拉有限公司 磺酰脲衍生物及其用途
CA3140017A1 (en) 2019-07-19 2021-01-28 Aurore HICK Polyaromatic urea derivatives and their use in the treatment of muscle diseases
TWI878335B (zh) 2019-08-12 2025-04-01 美商迪賽孚爾製藥有限公司 治療胃腸道基質瘤方法
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MX2022008103A (es) 2019-12-30 2022-09-19 Deciphera Pharmaceuticals Llc Formulaciones de inhibidores de la cinasa amorfa y metodos de estas.
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