JP2008514655A5 - - Google Patents

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Publication number
JP2008514655A5
JP2008514655A5 JP2007533891A JP2007533891A JP2008514655A5 JP 2008514655 A5 JP2008514655 A5 JP 2008514655A5 JP 2007533891 A JP2007533891 A JP 2007533891A JP 2007533891 A JP2007533891 A JP 2007533891A JP 2008514655 A5 JP2008514655 A5 JP 2008514655A5
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JP
Japan
Prior art keywords
diyl
atoms
hal
ocoor
ocon
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007533891A
Other languages
English (en)
Japanese (ja)
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JP2008514655A (ja
Filing date
Publication date
Priority claimed from DE102004047254A external-priority patent/DE102004047254A1/de
Application filed filed Critical
Publication of JP2008514655A publication Critical patent/JP2008514655A/ja
Publication of JP2008514655A5 publication Critical patent/JP2008514655A5/ja
Pending legal-status Critical Current

Links

JP2007533891A 2004-09-29 2005-09-01 凝固因子Xaの阻害剤として用いられるカルボニル化合物 Pending JP2008514655A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004047254A DE102004047254A1 (de) 2004-09-29 2004-09-29 Carbonylverbindungen
PCT/EP2005/009418 WO2006034769A1 (de) 2004-09-29 2005-09-01 Carbonylverbindungen verwendbar als inhibitoren des koagulationsfaktors xa

Publications (2)

Publication Number Publication Date
JP2008514655A JP2008514655A (ja) 2008-05-08
JP2008514655A5 true JP2008514655A5 (https=) 2008-10-16

Family

ID=35395743

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007533891A Pending JP2008514655A (ja) 2004-09-29 2005-09-01 凝固因子Xaの阻害剤として用いられるカルボニル化合物

Country Status (13)

Country Link
US (1) US20080081814A1 (https=)
EP (1) EP1797071A1 (https=)
JP (1) JP2008514655A (https=)
KR (1) KR20070057878A (https=)
CN (1) CN101031561A (https=)
AU (1) AU2005289164A1 (https=)
BR (1) BRPI0515577A (https=)
CA (1) CA2581732A1 (https=)
DE (1) DE102004047254A1 (https=)
MX (1) MX2007003470A (https=)
RU (1) RU2007116036A (https=)
WO (1) WO2006034769A1 (https=)
ZA (1) ZA200703443B (https=)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE50453E1 (en) 2006-04-07 2025-06-10 Vertex Pharmaceuticals Incorporated Indole derivatives as CFTR modulators
US10022352B2 (en) 2006-04-07 2018-07-17 Vertex Pharmaceuticals Incorporated Modulators of ATP-binding cassette transporters
US7645789B2 (en) 2006-04-07 2010-01-12 Vertex Pharmaceuticals Incorporated Indole derivatives as CFTR modulators
EP2674428B1 (en) 2006-04-07 2016-04-06 Vertex Pharmaceuticals Incorporated Modulators of ATP-binding cassette transporters
US8563573B2 (en) 2007-11-02 2013-10-22 Vertex Pharmaceuticals Incorporated Azaindole derivatives as CFTR modulators
US8673920B2 (en) 2009-05-06 2014-03-18 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
US8802868B2 (en) 2010-03-25 2014-08-12 Vertex Pharmaceuticals Incorporated Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide
MX353408B (es) 2010-04-22 2018-01-11 Vertex Pharma Proceso para producir compuestos de cicloalquilcarboxamido-indol.
WO2012058116A1 (en) 2010-10-27 2012-05-03 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2632464B1 (en) 2010-10-29 2015-04-29 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
AU2012299227A1 (en) 2011-08-19 2014-02-20 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
WO2013039802A1 (en) 2011-09-16 2013-03-21 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2771004B1 (en) 2011-10-25 2016-05-18 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
US8999990B2 (en) 2011-10-25 2015-04-07 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2773206B1 (en) 2011-10-31 2018-02-21 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
WO2013066714A1 (en) 2011-10-31 2013-05-10 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2773351B1 (en) 2011-10-31 2017-08-23 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2790511B1 (en) 2011-12-16 2016-09-14 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
JP5903499B2 (ja) 2011-12-22 2016-04-13 ノバルティス アーゲー ジヒドロ−ベンゾ−オキサジンおよびジヒドロ−ピリド−オキサジン誘導体
AR092857A1 (es) 2012-07-16 2015-05-06 Vertex Pharma Composiciones farmaceuticas de (r)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-il)-n-(1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il)-1h-indol-5-il)ciclopropancarboxamida y administracion de las mismas
AR092031A1 (es) 2012-07-26 2015-03-18 Merck Sharp & Dohme Inhibidores del canal de potasio medular externo renal
EP2925322B1 (en) 2012-11-29 2018-10-24 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
US9573961B2 (en) 2012-12-19 2017-02-21 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
WO2014126944A2 (en) 2013-02-18 2014-08-21 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2968288B1 (en) 2013-03-15 2018-07-04 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP3027625B1 (en) 2013-07-31 2018-05-30 Merck Sharp & Dohme Corp. Spiro-fused derivatives of piperidine useful for the treatment of inter alia hypertension and acute or chronic heart failure
RU2744460C2 (ru) 2014-04-15 2021-03-09 Вертекс Фармасьютикалз Инкорпорейтед Фармацевтические композиции для лечения заболеваний, опосредованных муковисцидозным трансмембранным регулятором проводимости
WO2016127358A1 (en) 2015-02-12 2016-08-18 Merck Sharp & Dohme Corp. Inhibitors of renal outer medullary potassium channel
US10669528B2 (en) 2015-06-25 2020-06-02 Children's Medical Center Corporation Methods and compositions relating to hematopoietic stem cell expansion, enrichment, and maintenance
WO2017161001A1 (en) 2016-03-15 2017-09-21 Children's Medical Center Corporation Methods and compositions relating to hematopoietic stem cell expansion
CN106674200B (zh) * 2016-12-21 2019-04-12 西安交通大学 一种含有l-脯氨酰胺片段的化合物及其制备方法和应用
CN108997200A (zh) * 2018-07-17 2018-12-14 成都睿智化学研究有限公司 一种5-氨甲基-哌啶-2-酮的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7030141B2 (en) * 2001-11-29 2006-04-18 Christopher Franklin Bigge Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade
PL377633A1 (pl) * 2003-04-03 2006-02-06 Merck Patent Gmbh Związki karbonylowe
DE10329457A1 (de) * 2003-04-03 2005-01-20 Merck Patent Gmbh Ethinylprolinderivate
DE102004045796A1 (de) * 2004-09-22 2006-03-23 Merck Patent Gmbh Arzneimittel enthaltend Carbonylverbindungen sowie deren Verwendung

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