JP2008510707A5 - - Google Patents
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- Publication number
- JP2008510707A5 JP2008510707A5 JP2007527996A JP2007527996A JP2008510707A5 JP 2008510707 A5 JP2008510707 A5 JP 2008510707A5 JP 2007527996 A JP2007527996 A JP 2007527996A JP 2007527996 A JP2007527996 A JP 2007527996A JP 2008510707 A5 JP2008510707 A5 JP 2008510707A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- alkyl
- base
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 0 *c1c(*)c(*)c(C*N*)c(*)c1 Chemical compound *c1c(*)c(*)c(C*N*)c(*)c1 0.000 description 6
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US60312404P | 2004-08-19 | 2004-08-19 | |
| PCT/US2005/029338 WO2006023611A1 (en) | 2004-08-19 | 2005-08-18 | Process for the synthesis c-2, c-3 substituted n-alkylated indoles useful as cpla2 inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008510707A JP2008510707A (ja) | 2008-04-10 |
| JP2008510707A5 true JP2008510707A5 (https=) | 2008-09-25 |
Family
ID=35219553
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007527996A Ceased JP2008510707A (ja) | 2004-08-19 | 2005-08-18 | ｃＰＬＡ２阻害剤として有用なＣ−２，Ｃ−３置換Ｎ−アルキル化インドールを合成する方法 |
Country Status (24)
| Country | Link |
|---|---|
| US (3) | US7582772B2 (https=) |
| EP (1) | EP1778629B1 (https=) |
| JP (1) | JP2008510707A (https=) |
| KR (1) | KR20070043036A (https=) |
| CN (2) | CN101006048B (https=) |
| AR (1) | AR053410A1 (https=) |
| AT (1) | ATE517084T1 (https=) |
| AU (1) | AU2005277392A1 (https=) |
| BR (1) | BRPI0514431A (https=) |
| CA (1) | CA2576008A1 (https=) |
| CR (1) | CR8936A (https=) |
| EC (1) | ECSP077244A (https=) |
| GT (1) | GT200500224A (https=) |
| HN (1) | HN2005000474A (https=) |
| IL (1) | IL181364A0 (https=) |
| MX (1) | MX2007002042A (https=) |
| NO (1) | NO20071253L (https=) |
| PE (1) | PE20060628A1 (https=) |
| RU (1) | RU2401829C2 (https=) |
| SG (1) | SG155214A1 (https=) |
| SV (1) | SV2006002200A (https=) |
| TW (1) | TW200609214A (https=) |
| UA (1) | UA85428C2 (https=) |
| WO (1) | WO2006023611A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7605156B2 (en) | 2001-12-03 | 2009-10-20 | Wyeth | Methods for the use of inhibitors of cytosolic phospholipase A2 |
| US7713964B2 (en) * | 2001-12-03 | 2010-05-11 | Wyeth Llc | Methods for treating asthmatic conditions |
| US7342119B2 (en) * | 2003-09-30 | 2008-03-11 | Wyeth Holdings Corporation | Process for the synthesis of a CPLA2 inhibitor |
| HN2004000536A (es) | 2003-12-16 | 2009-02-18 | Wyeth Corp | Un procediemiento de sintesis para la alquilacion reductiva de la posicon c-3 de indoles |
| GT200600228A (es) * | 2005-05-27 | 2006-12-26 | Inhibidores de la fosfolipasa a2 citosolica | |
| BRPI0718042A2 (pt) * | 2006-10-31 | 2013-11-12 | Wyeth Corp | Formulações semissólidas de inibidores de enzima fosfolipase |
| EP2104498A2 (en) * | 2006-10-31 | 2009-09-30 | Wyeth | Liquid formulations of phospholipase enzyme inhibitors |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH02115157A (ja) * | 1988-10-24 | 1990-04-27 | Hokko Chem Ind Co Ltd | スルホニルグリシン誘導体および除草剤 |
| ATE440824T1 (de) * | 1999-12-09 | 2009-09-15 | Bayer Cropscience Ag | Nitro-sulfobenzamide |
| US7101875B2 (en) * | 2001-12-03 | 2006-09-05 | Wyeth | Methods for treating arthritic disorders |
| US7713964B2 (en) * | 2001-12-03 | 2010-05-11 | Wyeth Llc | Methods for treating asthmatic conditions |
| US6797708B2 (en) * | 2001-12-03 | 2004-09-28 | Wyeth | Inhibitors of cytosolic phospholipase A2 |
| US7605156B2 (en) | 2001-12-03 | 2009-10-20 | Wyeth | Methods for the use of inhibitors of cytosolic phospholipase A2 |
| US6984735B2 (en) * | 2001-12-03 | 2006-01-10 | Wyeth | Process for making an aldehyde |
| JP4657605B2 (ja) * | 2001-12-03 | 2011-03-23 | ワイス・エルエルシー | 細胞質内ホスホリパーゼａ２の阻害剤 |
| US6635771B2 (en) * | 2001-12-03 | 2003-10-21 | Wyeth | N-benzhydryl indole compounds |
| TW200510305A (en) * | 2003-07-25 | 2005-03-16 | Wyeth Corp | Process for the preparation of CPLA2 inhibitors |
| WO2005012235A1 (en) | 2003-07-29 | 2005-02-10 | Ciba Specialty Chemicals Holding Inc. | 3-aryl-2-cyano-3-hydroxy-acrylic acid derivatives |
| US7582771B2 (en) * | 2003-09-03 | 2009-09-01 | Wyeth | Process for the synthesis of cPLA2 inhibitors |
| US7342119B2 (en) * | 2003-09-30 | 2008-03-11 | Wyeth Holdings Corporation | Process for the synthesis of a CPLA2 inhibitor |
| HN2004000536A (es) * | 2003-12-16 | 2009-02-18 | Wyeth Corp | Un procediemiento de sintesis para la alquilacion reductiva de la posicon c-3 de indoles |
-
2005
- 2005-08-16 AR ARP050103452A patent/AR053410A1/es unknown
- 2005-08-18 KR KR1020077005610A patent/KR20070043036A/ko not_active Ceased
- 2005-08-18 TW TW094128146A patent/TW200609214A/zh unknown
- 2005-08-18 BR BRPI0514431-0A patent/BRPI0514431A/pt not_active IP Right Cessation
- 2005-08-18 GT GT200500224A patent/GT200500224A/es unknown
- 2005-08-18 AU AU2005277392A patent/AU2005277392A1/en not_active Abandoned
- 2005-08-18 EP EP05788529A patent/EP1778629B1/en not_active Expired - Lifetime
- 2005-08-18 CN CN2005800280209A patent/CN101006048B/zh not_active Expired - Fee Related
- 2005-08-18 US US11/207,072 patent/US7582772B2/en not_active Expired - Fee Related
- 2005-08-18 SG SG200905383-6A patent/SG155214A1/en unknown
- 2005-08-18 SV SV2005002200A patent/SV2006002200A/es unknown
- 2005-08-18 JP JP2007527996A patent/JP2008510707A/ja not_active Ceased
- 2005-08-18 CN CN201010200760A patent/CN101830837A/zh active Pending
- 2005-08-18 MX MX2007002042A patent/MX2007002042A/es not_active Application Discontinuation
- 2005-08-18 PE PE2005000959A patent/PE20060628A1/es not_active Application Discontinuation
- 2005-08-18 UA UAA200701724A patent/UA85428C2/ru unknown
- 2005-08-18 WO PCT/US2005/029338 patent/WO2006023611A1/en not_active Ceased
- 2005-08-18 CA CA002576008A patent/CA2576008A1/en not_active Abandoned
- 2005-08-18 AT AT05788529T patent/ATE517084T1/de not_active IP Right Cessation
- 2005-08-18 RU RU2007105231/04A patent/RU2401829C2/ru not_active IP Right Cessation
- 2005-08-24 HN HN2005000474A patent/HN2005000474A/es unknown
-
2007
- 2007-02-13 EC EC2007007244A patent/ECSP077244A/es unknown
- 2007-02-15 IL IL181364A patent/IL181364A0/en unknown
- 2007-02-19 CR CR8936A patent/CR8936A/es not_active Application Discontinuation
- 2007-03-07 NO NO20071253A patent/NO20071253L/no not_active Application Discontinuation
-
2009
- 2009-08-18 US US12/542,914 patent/US7842837B2/en not_active Expired - Fee Related
-
2010
- 2010-11-11 US US12/943,958 patent/US8034960B2/en not_active Expired - Fee Related
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