JP2008500284A5 - - Google Patents

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Publication number
JP2008500284A5
JP2008500284A5 JP2007513296A JP2007513296A JP2008500284A5 JP 2008500284 A5 JP2008500284 A5 JP 2008500284A5 JP 2007513296 A JP2007513296 A JP 2007513296A JP 2007513296 A JP2007513296 A JP 2007513296A JP 2008500284 A5 JP2008500284 A5 JP 2008500284A5
Authority
JP
Japan
Prior art keywords
pyridin
urea
tert
phenyl
butylphenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007513296A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008500284A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/016422 external-priority patent/WO2005113511A1/en
Publication of JP2008500284A publication Critical patent/JP2008500284A/ja
Publication of JP2008500284A5 publication Critical patent/JP2008500284A5/ja
Pending legal-status Critical Current

Links

JP2007513296A 2004-05-12 2005-05-11 血栓症の治療に有用なｐ２ｙ１レセプターのウレアアンタゴニスト Pending JP2008500284A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US57028804P 2004-05-12 2004-05-12
US66581705P 2005-03-28 2005-03-28
PCT/US2005/016422 WO2005113511A1 (en) 2004-05-12 2005-05-11 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
US11/126,915 US7388021B2 (en) 2004-05-12 2005-05-11 Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions

Publications (2)

Publication Number Publication Date
JP2008500284A JP2008500284A (ja) 2008-01-10
JP2008500284A5 true JP2008500284A5 (enExample) 2008-02-21

Family

ID=35456856

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007513296A Pending JP2008500284A (ja) 2004-05-12 2005-05-11 血栓症の治療に有用なｐ２ｙ１レセプターのウレアアンタゴニスト

Country Status (11)

Country Link
US (2) US7388021B2 (enExample)
EP (1) EP1751113B1 (enExample)
JP (1) JP2008500284A (enExample)
KR (1) KR20070032648A (enExample)
AT (1) ATE460402T1 (enExample)
AU (1) AU2005245389A1 (enExample)
DE (1) DE602005019874D1 (enExample)
ES (1) ES2340179T3 (enExample)
MX (1) MXPA06013022A (enExample)
NO (1) NO20065534L (enExample)
WO (1) WO2005113511A1 (enExample)

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EP2528604B1 (en) 2010-01-29 2017-11-22 The Regents of the University of California Acyl piperidine inhibitors of soluble epoxide hydrolase
US8912184B1 (en) 2010-03-01 2014-12-16 Alzheimer's Institute Of America, Inc. Therapeutic and diagnostic methods
BR112012021806A2 (pt) * 2010-03-01 2015-09-08 Myrexis Inc compostos e seus usos terapêusticos.
FR2965262A1 (fr) * 2010-09-24 2012-03-30 Sanofi Aventis Derives de nicotinamide, leur preparation et leur application en therapeutique
EP2739144A4 (en) * 2011-06-20 2015-04-01 Alzheimer S Inst Of America Inc COMPOUNDS AND ITS THERAPEUTIC USE
US9428504B2 (en) * 2012-08-01 2016-08-30 Bristol-Myers Squibb Company 7-hydroxy-spiropipiperidine indolinyl antagonists of P2Y1 receptor
WO2014022343A1 (en) * 2012-08-01 2014-02-06 Bristol-Myers Squibb Company 7-hydroxy-indolinyl antagonists of p2y1 receptor
BR112015022462A8 (pt) * 2013-03-15 2019-11-26 Bristol Myers Squibb Co inibidores de ido, composição farmacêutica, método de inibição de atividade de indolamina 2,3-dioxigenase e uso dos referidos inibidores
GB201705863D0 (en) 2017-04-11 2017-05-24 Univ London Pyridinium salts and uses thereof
US11529819B2 (en) 2017-06-08 2022-12-20 Nippon Soda Co., Ltd. Recording material and compound
WO2019113288A1 (en) 2017-12-07 2019-06-13 Pitco Frialator, Inc. Fluid sensor and control system
DE102018113646B4 (de) 2018-06-07 2021-06-24 Helmholtz-Zentrum Dresden - Rossendorf E.V. 2-Phenoxypyridin-3-amin-Derivate und deren Verwendung
WO2021222637A1 (en) * 2020-04-30 2021-11-04 United States Government As Represented By The Department Of Veterans Affairs Krüppel-like factor 15 (klf15) small molecule agonists in kidney disease
EP4094762A1 (en) * 2021-05-25 2022-11-30 UCL Business Ltd Treatment of neurological indications
EP4095134A1 (en) 2021-05-25 2022-11-30 UCL Business Ltd Polycyclic compounds for the treatment of neurological indications

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US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
MX2007008434A (es) 2005-01-19 2007-07-25 Squibb Bristol Myers Co Derivados de 2-fenoxi-n-(1,3,4-tiadizol-2il)piridin-3-amina y compuestos relacionados como inhibidores del receptor p2y1 para el tratamiento de trastornos tromboembolicos.
WO2007002584A1 (en) 2005-06-27 2007-01-04 Bristol-Myers Squibb Company Linear urea mimics antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
WO2007002634A1 (en) 2005-06-27 2007-01-04 Bristol-Myers Squibb Company Carbocycle and heterocycle antagonists of p2y1 receptor useful in the treatment of thrombotic conditions

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