JP2007529495A5 - - Google Patents
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- Publication number
- JP2007529495A5 JP2007529495A5 JP2007503427A JP2007503427A JP2007529495A5 JP 2007529495 A5 JP2007529495 A5 JP 2007529495A5 JP 2007503427 A JP2007503427 A JP 2007503427A JP 2007503427 A JP2007503427 A JP 2007503427A JP 2007529495 A5 JP2007529495 A5 JP 2007529495A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- benzyl
- piperazin
- phenyl
- hydroxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55380804P | 2004-03-17 | 2004-03-17 | |
| US60/553,808 | 2004-03-17 | ||
| PCT/IB2005/000583 WO2005090300A1 (en) | 2004-03-17 | 2005-03-07 | Novel benzyl(idene)-lactam derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007529495A JP2007529495A (ja) | 2007-10-25 |
| JP2007529495A5 true JP2007529495A5 (https=) | 2008-04-24 |
| JP4880583B2 JP4880583B2 (ja) | 2012-02-22 |
Family
ID=34960867
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007503427A Expired - Fee Related JP4880583B2 (ja) | 2004-03-17 | 2005-03-07 | 新規なベンジル（ベンジリデン）−ラクタム誘導体 |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US7479559B2 (https=) |
| EP (1) | EP1727794B1 (https=) |
| JP (1) | JP4880583B2 (https=) |
| KR (1) | KR20060124770A (https=) |
| CN (1) | CN1934081A (https=) |
| AP (1) | AP2006003726A0 (https=) |
| AR (1) | AR050403A1 (https=) |
| AT (1) | ATE533745T1 (https=) |
| AU (1) | AU2005223481A1 (https=) |
| BR (1) | BRPI0508825A (https=) |
| CA (1) | CA2559530C (https=) |
| CR (1) | CR8618A (https=) |
| DO (1) | DOP2005000035A (https=) |
| EA (1) | EA200601461A1 (https=) |
| EC (1) | ECSP066853A (https=) |
| ES (1) | ES2374629T3 (https=) |
| GT (1) | GT200500051A (https=) |
| IL (1) | IL178105A0 (https=) |
| MA (1) | MA28474B1 (https=) |
| NL (1) | NL1028558C2 (https=) |
| NO (1) | NO20063602L (https=) |
| PA (1) | PA8626501A1 (https=) |
| PE (1) | PE20051153A1 (https=) |
| SV (1) | SV2005002051A (https=) |
| TN (1) | TNSN06287A1 (https=) |
| TW (1) | TW200604165A (https=) |
| UY (1) | UY28811A1 (https=) |
| WO (1) | WO2005090300A1 (https=) |
| ZA (1) | ZA200607133B (https=) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2371927T3 (es) * | 2005-01-13 | 2012-01-11 | Ge Healthcare Limited | Compuestos de bencil-lactama marcados con 11c y su uso como agentes de obtención de imágenes. |
| WO2006136945A1 (en) * | 2005-06-17 | 2006-12-28 | Pfizer Products Inc. | METABOLITES OF 1_ [_6- (1-ETHYL-l-HYDROXY-PROPYL) -PYRIDIN-3-YL] -3- [2- (4-METHYL-PIPERAZIN-I-YL) -BE NZYL] -PYRR0LIDIN-2-0NE AS SERATONIN RECEPTOR ANTAGONISTS |
| WO2007026219A2 (en) * | 2005-08-31 | 2007-03-08 | Pfizer Products Inc. | Combinations of a 5-ht1b antagonist with a noradrenalin re-uptake inhibitor or a serotonin noradrenalin reutake inhibitor for treating cns conditions |
| WO2008068614A2 (en) * | 2006-12-06 | 2008-06-12 | Pfizer Products Inc. | Stereoselective synthesis of 1-[6-ethyl-1,2-dihydroxy-propyl)-pyridin-3-yl]-3-[2-(4-methyl-piperazin-1-yl)-benzyl]-pyrrolidin-2-one |
| FR2948660B1 (fr) * | 2009-07-30 | 2011-08-19 | Oroxcell | Derives de 2-amino-2-phenyl-alkanol, leur preparation et les compositions pharmaceutiques qui les contiennent |
| EP2338873A1 (en) | 2009-12-22 | 2011-06-29 | Gmeiner, Peter | New aminotetraline derivatives |
| AU2010336027A1 (en) * | 2009-12-23 | 2012-07-19 | Auckland Uniservices Limited | Compounds, preparations and uses thereof |
| WO2014028829A1 (en) | 2012-08-16 | 2014-02-20 | The Scripps Research Institute | Novel kappa opioid ligands |
| US20140206667A1 (en) | 2012-11-14 | 2014-07-24 | Michela Gallagher | Methods and compositions for treating schizophrenia |
| KR101861942B1 (ko) * | 2014-01-20 | 2018-06-29 | 에프. 호프만-라 로슈 아게 | 신경 발생을 자극할 수 있는 n-페닐-락탐 유도체 및 이의 신경 장애 치료에서의 용도 |
| TW201706265A (zh) | 2015-03-09 | 2017-02-16 | 必治妥美雅史谷比公司 | 做為Ｒｈｏ激酶（ＲＯＣＫ）抑制劑之內醯胺 |
| WO2020183011A1 (en) | 2019-03-14 | 2020-09-17 | Institut Curie | Htr1d inhibitors and uses thereof in the treatment of cancer |
| CN119219603A (zh) * | 2023-06-28 | 2024-12-31 | 科辉智药(深圳)新药研究中心有限公司 | Sarm1酶活性抑制剂及其用途 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS58189163A (ja) * | 1982-04-02 | 1983-11-04 | Takeda Chem Ind Ltd | 縮合ピロリノン誘導体 |
| IL106142A (en) | 1992-06-29 | 1997-03-18 | Merck & Co Inc | Morpholine and thiomorpholine tachykinin receptor antagonists, their preparation and pharmaceutical compositions containing them |
| DK0689536T3 (da) | 1993-03-16 | 2001-07-30 | Pfizer | Naphthalenderivater |
| JP3786983B2 (ja) * | 1994-01-27 | 2006-06-21 | シエーリング アクチエンゲゼルシャフト | ピロリジノン誘導体 |
| GB9410512D0 (en) | 1994-05-25 | 1994-07-13 | Smithkline Beecham Plc | Novel treatment |
| FI965238L (fi) | 1994-06-29 | 1996-12-27 | Pfizer | Aryyli- ja heteroaryylialkoksinaftaleenijohdannaiset |
| EA001485B1 (ru) * | 1996-03-29 | 2001-04-23 | Пфайзер Инк. | Производные бензил(иден)-лактамов, их получение и применение в качестве селективных (ант)агонистов рецепторов 5-htи/или 5-ht |
| US6423708B1 (en) * | 1996-09-30 | 2002-07-23 | Pfizer Inc | Aralkyl and aralkylidene heterocyclic lactams and imides |
| UA56185C2 (uk) * | 1996-09-30 | 2003-05-15 | Пфайзер Інк. | Аралкіл- та аралкіліденгетероциклічні лактами та іміди, фармацевтична композиція та спосіб лікування |
| DE10002509A1 (de) | 2000-01-21 | 2001-07-26 | Gruenenthal Gmbh | Substituierte Glutarimide |
| US20020049211A1 (en) * | 2000-09-06 | 2002-04-25 | Sobolov-Jaynes Susan Beth | Combination treatment for depression and anxiety |
| TWI263640B (en) * | 2001-12-19 | 2006-10-11 | Bristol Myers Squibb Co | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
-
2005
- 2005-03-07 KR KR1020067019078A patent/KR20060124770A/ko not_active Ceased
- 2005-03-07 JP JP2007503427A patent/JP4880583B2/ja not_active Expired - Fee Related
- 2005-03-07 CN CNA2005800085634A patent/CN1934081A/zh active Pending
- 2005-03-07 WO PCT/IB2005/000583 patent/WO2005090300A1/en not_active Ceased
- 2005-03-07 EA EA200601461A patent/EA200601461A1/ru unknown
- 2005-03-07 AP AP2006003726A patent/AP2006003726A0/xx unknown
- 2005-03-07 AU AU2005223481A patent/AU2005223481A1/en not_active Abandoned
- 2005-03-07 ES ES05708687T patent/ES2374629T3/es not_active Expired - Lifetime
- 2005-03-07 BR BRPI0508825-9A patent/BRPI0508825A/pt not_active IP Right Cessation
- 2005-03-07 CA CA2559530A patent/CA2559530C/en not_active Expired - Fee Related
- 2005-03-07 EP EP05708687A patent/EP1727794B1/en not_active Expired - Lifetime
- 2005-03-07 AT AT05708687T patent/ATE533745T1/de active
- 2005-03-10 DO DO2005000035A patent/DOP2005000035A/es unknown
- 2005-03-15 PE PE2005000296A patent/PE20051153A1/es not_active Application Discontinuation
- 2005-03-15 TW TW094107893A patent/TW200604165A/zh unknown
- 2005-03-15 GT GT200500051A patent/GT200500051A/es unknown
- 2005-03-15 UY UY28811A patent/UY28811A1/es not_active Application Discontinuation
- 2005-03-16 NL NL1028558A patent/NL1028558C2/nl not_active IP Right Cessation
- 2005-03-16 AR ARP050101025A patent/AR050403A1/es unknown
- 2005-03-16 SV SV2005002051A patent/SV2005002051A/es not_active Application Discontinuation
- 2005-03-17 PA PA20058626501A patent/PA8626501A1/es unknown
- 2005-03-17 US US11/083,188 patent/US7479559B2/en not_active Expired - Fee Related
-
2006
- 2006-08-09 NO NO20063602A patent/NO20063602L/no not_active Application Discontinuation
- 2006-08-25 ZA ZA200607133A patent/ZA200607133B/en unknown
- 2006-09-13 CR CR8618A patent/CR8618A/es not_active Application Discontinuation
- 2006-09-14 IL IL178105A patent/IL178105A0/en unknown
- 2006-09-15 MA MA29327A patent/MA28474B1/fr unknown
- 2006-09-15 TN TNP2006000287A patent/TNSN06287A1/fr unknown
- 2006-09-15 EC EC2006006853A patent/ECSP066853A/es unknown
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