JP2007526264A5 - - Google Patents
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- Publication number
- JP2007526264A5 JP2007526264A5 JP2007501151A JP2007501151A JP2007526264A5 JP 2007526264 A5 JP2007526264 A5 JP 2007526264A5 JP 2007501151 A JP2007501151 A JP 2007501151A JP 2007501151 A JP2007501151 A JP 2007501151A JP 2007526264 A5 JP2007526264 A5 JP 2007526264A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- amino
- salt
- tert
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- BPNISPBQIJAMSV-CKIAUBSUSA-N C/C=C(\c1ccc(C#Cc2ccccc2F)[o]1)/N(CC1)CCC1c1cccc(CN)c1 Chemical compound C/C=C(\c1ccc(C#Cc2ccccc2F)[o]1)/N(CC1)CCC1c1cccc(CN)c1 BPNISPBQIJAMSV-CKIAUBSUSA-N 0.000 description 1
- 0 CC1(*)C=C(CN2S(C)(C)CC[Si]2(C)C)C=C(C2(CCN(Cc3ccccc3)CC2)O)C=C1 Chemical compound CC1(*)C=C(CN2S(C)(C)CC[Si]2(C)C)C=C(C2(CCN(Cc3ccccc3)CC2)O)C=C1 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04004799.5 | 2004-03-02 | ||
| EP04004799A EP1571150A1 (en) | 2004-03-02 | 2004-03-02 | Process for the preparation of tryptase inhibitors |
| US58574504P | 2004-07-06 | 2004-07-06 | |
| US60/585,745 | 2004-07-06 | ||
| PCT/EP2005/001676 WO2005095385A1 (en) | 2004-03-02 | 2005-02-18 | Process for the preparation of tryptase inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007526264A JP2007526264A (ja) | 2007-09-13 |
| JP2007526264A5 true JP2007526264A5 (enExample) | 2008-03-27 |
| JP4851440B2 JP4851440B2 (ja) | 2012-01-11 |
Family
ID=34745976
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007501151A Expired - Fee Related JP4851440B2 (ja) | 2004-03-02 | 2005-02-18 | トリプターゼ阻害剤の製造方法 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20130225825A1 (enExample) |
| EP (2) | EP1571150A1 (enExample) |
| JP (1) | JP4851440B2 (enExample) |
| CN (2) | CN1950362B (enExample) |
| AT (1) | ATE447567T1 (enExample) |
| AU (1) | AU2005229319B2 (enExample) |
| BR (1) | BRPI0508430A (enExample) |
| CA (1) | CA2557391C (enExample) |
| DK (1) | DK1723140T3 (enExample) |
| ES (1) | ES2334245T3 (enExample) |
| NZ (1) | NZ549224A (enExample) |
| PL (1) | PL1723140T3 (enExample) |
| PT (1) | PT1723140E (enExample) |
| RS (1) | RS51144B (enExample) |
| RU (1) | RU2378271C2 (enExample) |
| SI (1) | SI1723140T1 (enExample) |
| TN (1) | TNSN06260A1 (enExample) |
| UA (1) | UA85701C2 (enExample) |
| WO (1) | WO2005095385A1 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200840566A (en) * | 2006-12-22 | 2008-10-16 | Esteve Labor Dr | Heterocyclyl-substituted-ethylamino-phenyl derivatives, their preparation and use as medicaments |
| EP2224803B1 (en) * | 2007-11-21 | 2014-04-02 | Janssen Pharmaceutica N.V. | Spiropiperidines for use as tryptase inhibitors |
| CN103508936A (zh) * | 2008-08-22 | 2014-01-15 | 赛诺菲-安万特 | 用于制备吲哚苄胺化合物的中间体 |
| WO2011037947A1 (en) * | 2009-09-24 | 2011-03-31 | Sanofi-Aventis U.S. Llc | Synthesis of (4-fluoro-3-piperidin-4-yl-benzyl)-carbamic acid tert-butyl ester and intermediates thereof |
| JP2013515723A (ja) * | 2009-12-23 | 2013-05-09 | サノフイ | 炎症性腸疾患の処置 |
| US20140113934A1 (en) | 2011-06-20 | 2014-04-24 | E I Du Pont De Nemours And Company | Heterocyclic compounds for treating helminth infections |
| JP2015502936A (ja) | 2011-11-28 | 2015-01-29 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニーＥ．Ｉ．Ｄｕ Ｐｏｎｔ Ｄｅ Ｎｅｍｏｕｒｓ Ａｎｄ Ｃｏｍｐａｎｙ | スルホンアミド駆虫薬 |
| WO2014099837A1 (en) | 2012-12-18 | 2014-06-26 | E. I. Du Pont De Nemours And Company | Sulfonamide anthelmintics |
| CN111793101B (zh) | 2020-07-17 | 2022-09-30 | 四川大学 | C-核苷化合物的合成方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0401166B1 (de) * | 1989-06-01 | 1995-02-22 | Ciba-Geigy Ag | Neue, stickstoffhaltige Titanocene und deren Verwendung |
| US5252753A (en) * | 1991-11-01 | 1993-10-12 | Ortho Pharmaceutical Corporation | Process for the preparation of certain substituted biphenyl tetrazoles and compounds thereof |
| IL122072A (en) * | 1996-11-14 | 2001-03-19 | Akzo Nobel Nv | Piperidine derivatives their preparation and pharmaceutical compositions containing them |
| WO1999018053A1 (en) * | 1997-10-02 | 1999-04-15 | The University Of Western Ontario | Preparation of radiolabelled haloaromatics via polymer-bound intermediates |
| US20020045613A1 (en) * | 2000-04-27 | 2002-04-18 | Heinz Pauls | 1-aroyl-piperidinyl benzamidines |
| DZ3347A1 (fr) * | 2000-05-22 | 2001-11-29 | Aventis Pharma Inc | Dérivés d'arylméthylamine pour leur utilisation comme inhibiteurs de la tryptase |
| JP4846238B2 (ja) * | 2002-10-18 | 2011-12-28 | マクマスター ユニバーシティー | 放射線標識した化合物の精製方法 |
| GB0308613D0 (en) * | 2002-12-26 | 2003-05-21 | Aventis Pharma Inc | 4-(3-Aminomethylphenyl) piperidin-1-yl- 5-(2-fluorophenylethynyl) furan-2-yl- methanone as an inhibitor of mast cell tryptase |
-
2004
- 2004-03-02 EP EP04004799A patent/EP1571150A1/en not_active Withdrawn
-
2005
- 2005-02-18 BR BRPI0508430-0A patent/BRPI0508430A/pt not_active IP Right Cessation
- 2005-02-18 JP JP2007501151A patent/JP4851440B2/ja not_active Expired - Fee Related
- 2005-02-18 EP EP05779890A patent/EP1723140B1/en not_active Expired - Lifetime
- 2005-02-18 UA UAA200610386A patent/UA85701C2/ru unknown
- 2005-02-18 RS RSP-2009/0532A patent/RS51144B/sr unknown
- 2005-02-18 AT AT05779890T patent/ATE447567T1/de active
- 2005-02-18 ES ES05779890T patent/ES2334245T3/es not_active Expired - Lifetime
- 2005-02-18 DK DK05779890.2T patent/DK1723140T3/da active
- 2005-02-18 NZ NZ549224A patent/NZ549224A/en not_active IP Right Cessation
- 2005-02-18 PT PT05779890T patent/PT1723140E/pt unknown
- 2005-02-18 RU RU2006134623/04A patent/RU2378271C2/ru not_active IP Right Cessation
- 2005-02-18 CN CN2005800140491A patent/CN1950362B/zh not_active Expired - Fee Related
- 2005-02-18 CN CN2008101787837A patent/CN101429194B/zh not_active Expired - Fee Related
- 2005-02-18 SI SI200530896T patent/SI1723140T1/sl unknown
- 2005-02-18 PL PL05779890T patent/PL1723140T3/pl unknown
- 2005-02-18 CA CA2557391A patent/CA2557391C/en not_active Expired - Fee Related
- 2005-02-18 AU AU2005229319A patent/AU2005229319B2/en not_active Ceased
- 2005-02-18 WO PCT/EP2005/001676 patent/WO2005095385A1/en not_active Ceased
-
2006
- 2006-08-15 TN TNP2006000260A patent/TNSN06260A1/en unknown
-
2013
- 2013-04-11 US US13/861,066 patent/US20130225825A1/en not_active Abandoned
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