JP2007511519A - 液状投薬形態物におけるトピラメートの制御放出 - Google Patents

液状投薬形態物におけるトピラメートの制御放出 Download PDF

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Publication number
JP2007511519A
JP2007511519A JP2006539847A JP2006539847A JP2007511519A JP 2007511519 A JP2007511519 A JP 2007511519A JP 2006539847 A JP2006539847 A JP 2006539847A JP 2006539847 A JP2006539847 A JP 2006539847A JP 2007511519 A JP2007511519 A JP 2007511519A
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Japan
Prior art keywords
dosage form
topiramate
layer
drug
liquid
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JP2006539847A
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English (en)
Japanese (ja)
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JP2007511519A5 (cg-RX-API-DMAC7.html
Inventor
リー，シヤオリング
ラム，アンドリユー
ドング，リアング
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アルザ・コーポレーシヨン
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Publication of JP2007511519A publication Critical patent/JP2007511519A/ja
Publication of JP2007511519A5 publication Critical patent/JP2007511519A5/ja
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2006539847A 2003-11-14 2004-11-12 液状投薬形態物におけるトピラメートの制御放出 Pending JP2007511519A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51995803P 2003-11-14 2003-11-14
PCT/US2004/037616 WO2005048981A1 (en) 2003-11-14 2004-11-12 Controlled release of topirimate in liquid dosage forms

Publications (2)

Publication Number Publication Date
JP2007511519A true JP2007511519A (ja) 2007-05-10
JP2007511519A5 JP2007511519A5 (cg-RX-API-DMAC7.html) 2007-12-27

Family

ID=34619401

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006539847A Pending JP2007511519A (ja) 2003-11-14 2004-11-12 液状投薬形態物におけるトピラメートの制御放出

Country Status (13)

Country Link
US (1) US20050129765A1 (cg-RX-API-DMAC7.html)
EP (1) EP1684713A1 (cg-RX-API-DMAC7.html)
JP (1) JP2007511519A (cg-RX-API-DMAC7.html)
KR (1) KR20060120193A (cg-RX-API-DMAC7.html)
CN (1) CN1905857A (cg-RX-API-DMAC7.html)
AU (1) AU2004291081A1 (cg-RX-API-DMAC7.html)
CA (1) CA2545834A1 (cg-RX-API-DMAC7.html)
IL (1) IL175605A0 (cg-RX-API-DMAC7.html)
MX (1) MXPA06005462A (cg-RX-API-DMAC7.html)
NO (1) NO20062739L (cg-RX-API-DMAC7.html)
TW (1) TW200528144A (cg-RX-API-DMAC7.html)
WO (1) WO2005048981A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200604882B (cg-RX-API-DMAC7.html)

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US20050232995A1 (en) 2002-07-29 2005-10-20 Yam Nyomi V Methods and dosage forms for controlled delivery of paliperidone and risperidone
MXPA06002067A (es) * 2003-08-22 2006-08-11 Johnson & Johnson Suministro gradual de topiramato durante periodo prolongado.
WO2005065648A2 (en) * 2003-12-29 2005-07-21 Alza Corporation, Inc., Novel drug compositions and dosage forms of topiramate
AU2004312082A1 (en) * 2003-12-29 2005-07-21 Alza Corporation, Inc. Novel drug compositions and dosage forms
MX2007014713A (es) * 2005-05-25 2008-02-14 Janssen Pharmaceutica Nv Formulacion pediatrica de topiramato.
WO2008027557A2 (en) * 2006-08-31 2008-03-06 Spherics, Inc. Topiramate compositions and methods of enhancing its bioavailability
EP2394643B1 (en) 2006-11-17 2015-09-02 Supernus Pharmaceuticals, Inc. Sustained-release formulations of topiramate
EP2363113B1 (en) * 2006-12-04 2017-08-02 Supernus Pharmaceuticals, Inc. Enhanced immediate release formulations of topiramate
EP2219624A2 (en) * 2007-11-08 2010-08-25 Glaxo Group Limited Pharmaceutical formulations
US20120145572A1 (en) * 2009-04-20 2012-06-14 Ecole Polytechnique Federale De Lausanne (Epfl) Containers assembled in fluid and corresponding production
CN102579367B (zh) * 2012-03-23 2014-03-12 中国人民解放军军事医学科学院毒物药物研究所 托吡酯缓释药物组合物、其制备方法及用途
CN103316026B (zh) 2012-03-23 2016-05-11 中国人民解放军军事医学科学院毒物药物研究所 含芬特明和托吡酯的联合产品及其制备方法
EP2829270B1 (en) 2012-03-23 2020-11-11 Institute of Pharmacology and Toxicology Academy of Military Medical Sciences P.L.A. China Joint product containing synephrine and topiramate
US8652527B1 (en) 2013-03-13 2014-02-18 Upsher-Smith Laboratories, Inc Extended-release topiramate capsules
US9101545B2 (en) 2013-03-15 2015-08-11 Upsher-Smith Laboratories, Inc. Extended-release topiramate capsules
CN108379588B (zh) * 2018-03-05 2024-07-02 合肥合源药业有限公司 托吡酯组合物
US20210169844A1 (en) 2019-12-10 2021-06-10 Tulex Pharmaceuticals Inc. Compositions and methods for treating epilepsy, seizures and other conditions
US12290504B2 (en) 2023-04-11 2025-05-06 Tap Pharmaceuticals Ag Aqueous formulations of topiramate

Citations (2)

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JP2002532406A (ja) * 1998-12-17 2002-10-02 アルザ・コーポレーション 複合コーティングによる液体充填ゼラチンカプセルの放出制御システムへの変換
US6559293B1 (en) * 2002-02-15 2003-05-06 Transform Pharmaceuticals, Inc. Topiramate sodium trihydrate

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JP2002532406A (ja) * 1998-12-17 2002-10-02 アルザ・コーポレーション 複合コーティングによる液体充填ゼラチンカプセルの放出制御システムへの変換
US6559293B1 (en) * 2002-02-15 2003-05-06 Transform Pharmaceuticals, Inc. Topiramate sodium trihydrate

Also Published As

Publication number Publication date
IL175605A0 (en) 2006-09-05
US20050129765A1 (en) 2005-06-16
TW200528144A (en) 2005-09-01
ZA200604882B (en) 2007-11-28
AU2004291081A1 (en) 2005-06-02
CN1905857A (zh) 2007-01-31
WO2005048981A1 (en) 2005-06-02
CA2545834A1 (en) 2005-06-02
NO20062739L (no) 2006-08-14
MXPA06005462A (es) 2006-12-15
EP1684713A1 (en) 2006-08-02
KR20060120193A (ko) 2006-11-24

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