JP2007500716A5 - - Google Patents

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Publication number
JP2007500716A5
JP2007500716A5 JP2006522073A JP2006522073A JP2007500716A5 JP 2007500716 A5 JP2007500716 A5 JP 2007500716A5 JP 2006522073 A JP2006522073 A JP 2006522073A JP 2006522073 A JP2006522073 A JP 2006522073A JP 2007500716 A5 JP2007500716 A5 JP 2007500716A5
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JP
Japan
Prior art keywords
alkyl
group
hydrogen
cycloalkyl
independently selected
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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JP2006522073A
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English (en)
Japanese (ja)
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JP4884219B2 (ja
JP2007500716A (ja
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Priority claimed from PCT/US2004/024542 external-priority patent/WO2005011654A2/en
Publication of JP2007500716A publication Critical patent/JP2007500716A/ja
Publication of JP2007500716A5 publication Critical patent/JP2007500716A5/ja
Application granted granted Critical
Publication of JP4884219B2 publication Critical patent/JP4884219B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006522073A 2003-07-29 2004-07-29 ピリジル誘導体および治療剤としてのその用途 Expired - Fee Related JP4884219B2 (ja)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
US49114003P 2003-07-29 2003-07-29
US60/491,140 2003-07-29
US49132203P 2003-07-30 2003-07-30
US49108003P 2003-07-30 2003-07-30
US49111603P 2003-07-30 2003-07-30
US49114103P 2003-07-30 2003-07-30
US60/491,141 2003-07-30
US60/491,322 2003-07-30
US60/491,116 2003-07-30
US60/491,080 2003-07-30
PCT/US2004/024542 WO2005011654A2 (en) 2003-07-29 2004-07-29 Pyridyl derivatives and their use as therapeutic agents

Publications (3)

Publication Number Publication Date
JP2007500716A JP2007500716A (ja) 2007-01-18
JP2007500716A5 true JP2007500716A5 (https=) 2007-09-13
JP4884219B2 JP4884219B2 (ja) 2012-02-29

Family

ID=34120125

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006522073A Expired - Fee Related JP4884219B2 (ja) 2003-07-29 2004-07-29 ピリジル誘導体および治療剤としてのその用途

Country Status (17)

Country Link
US (3) US7763618B2 (https=)
EP (1) EP1651605B1 (https=)
JP (1) JP4884219B2 (https=)
KR (1) KR20060036105A (https=)
AT (1) ATE556056T1 (https=)
AU (1) AU2004261250B2 (https=)
BR (1) BRPI0413059A (https=)
CA (1) CA2533898A1 (https=)
EC (1) ECSP066314A (https=)
ES (1) ES2386354T3 (https=)
IL (1) IL173397A0 (https=)
MA (1) MA28012A1 (https=)
MX (1) MXPA06001202A (https=)
NO (1) NO20060973L (https=)
SG (1) SG145695A1 (https=)
TN (1) TNSN06035A1 (https=)
WO (1) WO2005011654A2 (https=)

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WO2008062276A2 (en) * 2006-11-20 2008-05-29 Glenmark Pharmaceuticals S.A. Acetylene derivatives as stearoyl coa desaturase inhibitors
US7638541B2 (en) 2006-12-28 2009-12-29 Metabolex Inc. 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine
WO2008091863A1 (en) 2007-01-23 2008-07-31 Kalypsys, Inc. Sulfonyl-substituted bicyclic compounds as ppar modulators for the treatment of non-alcoholic steatohepatitis
US8575167B2 (en) 2007-02-06 2013-11-05 Takeda Pharmaceutical Company Limited Spiro compounds having stearoyl-CoA desaturase action
CA2685266C (en) 2007-04-27 2014-01-28 Purdue Pharma L.P. Trpv1 antagonists and uses thereof for the treatment of prevention of pain, ui and ulcer, ibd, or ibs in an animal
WO2008157844A1 (en) 2007-06-21 2008-12-24 Forest Laboratories Holdings Limited Novel piperazine derivatives as inhibitors of stearoyl-coa desaturase
AU2008279447A1 (en) 2007-07-19 2009-01-29 Metabolex, Inc. N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders
BRPI0815048B8 (pt) 2007-08-08 2021-05-25 Graceway Pharmaceuticals Llc derivados de fenóxi-pirrolidinas, seus usos e composições farmacêuticas
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