JP2006528215A5 - - Google Patents
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- Publication number
- JP2006528215A5 JP2006528215A5 JP2006529752A JP2006529752A JP2006528215A5 JP 2006528215 A5 JP2006528215 A5 JP 2006528215A5 JP 2006529752 A JP2006529752 A JP 2006529752A JP 2006529752 A JP2006529752 A JP 2006529752A JP 2006528215 A5 JP2006528215 A5 JP 2006528215A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- reacted
- give
- hcl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 41
- 150000003839 salts Chemical class 0.000 claims description 3
- XJUZRXYOEPSWMB-UHFFFAOYSA-N Chloromethyl methyl ether Chemical compound COCCl XJUZRXYOEPSWMB-UHFFFAOYSA-N 0.000 claims description 2
- 239000002253 acid Substances 0.000 claims description 2
- 238000004519 manufacturing process Methods 0.000 claims description 2
- 238000007363 ring formation reaction Methods 0.000 claims description 2
- 0 C*(C=C1)C=Nc2c1nc(-c([s]c1c(*)cc3)nc1c3OC)[n]2COC Chemical compound C*(C=C1)C=Nc2c1nc(-c([s]c1c(*)cc3)nc1c3OC)[n]2COC 0.000 description 4
- 238000000034 method Methods 0.000 description 2
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP03009842 | 2003-05-13 | ||
| PCT/EP2004/004843 WO2004101558A1 (en) | 2003-05-13 | 2004-05-06 | 2-imidazo-benzothiazoles as adenosine receptor ligands |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006528215A JP2006528215A (ja) | 2006-12-14 |
| JP2006528215A5 true JP2006528215A5 (https=) | 2009-11-26 |
| JP4408291B2 JP4408291B2 (ja) | 2010-02-03 |
Family
ID=33395778
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006529752A Expired - Fee Related JP4408291B2 (ja) | 2003-05-13 | 2004-05-06 | アデノシン受容体リガンドとしての２−イミダゾ−ベンゾチアゾール |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7122545B2 (https=) |
| EP (1) | EP1636217B1 (https=) |
| JP (1) | JP4408291B2 (https=) |
| KR (1) | KR100710453B1 (https=) |
| CN (1) | CN100372844C (https=) |
| AT (1) | ATE407133T1 (https=) |
| AU (1) | AU2004238508B2 (https=) |
| BR (1) | BRPI0410315A (https=) |
| CA (1) | CA2523959A1 (https=) |
| DE (1) | DE602004016328D1 (https=) |
| ES (1) | ES2313001T3 (https=) |
| MX (1) | MXPA05012120A (https=) |
| PL (1) | PL1636217T3 (https=) |
| RU (1) | RU2340612C2 (https=) |
| WO (1) | WO2004101558A1 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1910385B1 (en) * | 2005-08-04 | 2013-07-24 | Sirtris Pharmaceuticals, Inc. | Benzothiazoles and thiazolopyridines as sirtuin modulators |
| TW200736252A (en) | 2006-01-27 | 2007-10-01 | Astrazeneca Ab | Novel heteroaryl substituted benzothiazoles |
| TW200813035A (en) | 2006-06-19 | 2008-03-16 | Astrazeneca Ab | Novel heteroaryl substituted benzoxazoles |
| TW200901998A (en) | 2007-03-06 | 2009-01-16 | Astrazeneca Ab | Novel 2-heteroaryl substituted benzothiophenes and benzofuranes |
| WO2010115736A2 (en) * | 2009-04-02 | 2010-10-14 | Merck Serono S.A. | Dihydroorotate dehydrogenase inhibitors |
| EP2414340A1 (en) * | 2009-04-03 | 2012-02-08 | Dainippon Sumitomo Pharma Co., Ltd. | Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof |
| US8575336B2 (en) | 2011-07-27 | 2013-11-05 | Pfizer Limited | Indazoles |
| WO2016164565A1 (en) * | 2015-04-08 | 2016-10-13 | University Of Delaware | Trans-cycloheptenes and hetero-trans-cycloheptenes for bioorthogonal coupling |
| WO2018193090A2 (en) * | 2017-04-21 | 2018-10-25 | Amneal Pharmaceuticals Company Gmbh | Process for preparation of eliglustat hemitartrate and intermediates thereof |
| AU2018320673B2 (en) | 2017-08-21 | 2023-03-30 | Merck Patent Gmbh | Benzimidazole derivatives as adenosine receptor antagonists |
| WO2025160629A1 (en) * | 2024-01-31 | 2025-08-07 | Certa Therapeutics Pty Ltd | Proton sensing gpcr modulators |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI91859C (fi) * | 1987-06-17 | 1994-08-25 | Eisai Co Ltd | Analogiamenetelmä antiallergisena aineena aktiivisen bentsotiatsolijohdannaisen valmistamiseksi |
| IL90337A0 (en) * | 1988-05-24 | 1989-12-15 | Pfizer | Aromatic and heterocyclic carboxamide derivatives as antineoplastic agents |
| IT1260444B (it) * | 1992-01-24 | 1996-04-09 | Mario Brufani | Derivati della 8-(1-amminocicloalchil)1,3-dialchilxantina, procedimenbto di preparazione e loro composizioni farmaceutiche antidepressive, nootropiche e psicostimolanti |
| US6037473A (en) * | 1997-11-13 | 2000-03-14 | Haarmann & Reimer Gmbh | Use of substituted benzazoles as UV absorbers, new benzazoles and processes for their preparation |
| US6841549B1 (en) * | 1999-07-02 | 2005-01-11 | Eisai Co., Ltd. | Condensed imidazole compounds and a therapeutic agent for diabetes mellitus |
| AU8181701A (en) * | 2000-06-21 | 2002-01-02 | Hoffmann La Roche | Benzothiazole derivatives |
| PL1628662T3 (pl) * | 2003-05-21 | 2007-07-31 | Hoffmann La Roche | Pochodne benzotiazolu i ich zastosowanie w leczeniu chorób związanych z receptorem adenozynowym A2A |
-
2004
- 2004-05-06 AU AU2004238508A patent/AU2004238508B2/en not_active Ceased
- 2004-05-06 PL PL04731369T patent/PL1636217T3/pl unknown
- 2004-05-06 JP JP2006529752A patent/JP4408291B2/ja not_active Expired - Fee Related
- 2004-05-06 CN CNB2004800117819A patent/CN100372844C/zh not_active Expired - Fee Related
- 2004-05-06 WO PCT/EP2004/004843 patent/WO2004101558A1/en not_active Ceased
- 2004-05-06 DE DE602004016328T patent/DE602004016328D1/de not_active Expired - Lifetime
- 2004-05-06 EP EP04731369A patent/EP1636217B1/en not_active Expired - Lifetime
- 2004-05-06 CA CA002523959A patent/CA2523959A1/en not_active Abandoned
- 2004-05-06 AT AT04731369T patent/ATE407133T1/de not_active IP Right Cessation
- 2004-05-06 RU RU2005138546/04A patent/RU2340612C2/ru not_active IP Right Cessation
- 2004-05-06 BR BRPI0410315-7A patent/BRPI0410315A/pt not_active IP Right Cessation
- 2004-05-06 MX MXPA05012120A patent/MXPA05012120A/es active IP Right Grant
- 2004-05-06 KR KR1020057021535A patent/KR100710453B1/ko not_active Expired - Fee Related
- 2004-05-06 ES ES04731369T patent/ES2313001T3/es not_active Expired - Lifetime
- 2004-05-11 US US10/843,241 patent/US7122545B2/en not_active Expired - Fee Related
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