JP2011506323A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2011506323A5 JP2011506323A5 JP2010536949A JP2010536949A JP2011506323A5 JP 2011506323 A5 JP2011506323 A5 JP 2011506323A5 JP 2010536949 A JP2010536949 A JP 2010536949A JP 2010536949 A JP2010536949 A JP 2010536949A JP 2011506323 A5 JP2011506323 A5 JP 2011506323A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrogen
- group
- formula
- alkyl
- oxygen protecting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1241107P | 2007-12-07 | 2007-12-07 | |
| US1240907P | 2007-12-07 | 2007-12-07 | |
| US1240807P | 2007-12-07 | 2007-12-07 | |
| US61/012,409 | 2007-12-07 | ||
| US61/012,408 | 2007-12-07 | ||
| US61/012,411 | 2007-12-07 | ||
| US8004808P | 2008-07-11 | 2008-07-11 | |
| US61/080,048 | 2008-07-11 | ||
| PCT/US2008/013498 WO2009075818A1 (en) | 2007-12-07 | 2008-12-08 | Intermediates and methods for making zearalenone macrolide analogs |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014042331A Division JP2014141498A (ja) | 2007-12-07 | 2014-03-05 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011506323A JP2011506323A (ja) | 2011-03-03 |
| JP2011506323A5 true JP2011506323A5 (https=) | 2012-02-02 |
| JP5496908B2 JP5496908B2 (ja) | 2014-05-21 |
Family
ID=40445478
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010536950A Active JP5492786B2 (ja) | 2007-12-07 | 2008-12-08 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
| JP2010536949A Active JP5496908B2 (ja) | 2007-12-07 | 2008-12-08 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
| JP2014042331A Withdrawn JP2014141498A (ja) | 2007-12-07 | 2014-03-05 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010536950A Active JP5492786B2 (ja) | 2007-12-07 | 2008-12-08 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014042331A Withdrawn JP2014141498A (ja) | 2007-12-07 | 2014-03-05 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (3) | US8350059B2 (https=) |
| EP (2) | EP2231635B1 (https=) |
| JP (3) | JP5492786B2 (https=) |
| CN (2) | CN101889006B (https=) |
| BR (2) | BRPI0820958B1 (https=) |
| CA (2) | CA2708141C (https=) |
| IL (2) | IL205954A (https=) |
| MX (2) | MX2010005999A (https=) |
| RU (2) | RU2478630C2 (https=) |
| WO (2) | WO2009075823A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1653059A (zh) | 2002-03-08 | 2005-08-10 | 卫材株式会社 | 用作医药品的大环化合物 |
| KR101667960B1 (ko) | 2007-07-25 | 2016-10-20 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 암 치료에서 이용하기 위한 멀티키나아제 억제제 |
| RU2478630C2 (ru) * | 2007-12-07 | 2013-04-10 | ЭЙСАН Ар ЭНД Ди МЕНЕДЖМЕНТ КО., ЛТД. | Промежуточные соединения и способы получения зеараленоновых макролидных аналогов |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL69666A (en) * | 1982-09-13 | 1987-10-20 | Lilly Co Eli | 20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use |
| GB9225396D0 (en) | 1992-12-04 | 1993-01-27 | Sandoz Ltd | Improvements in or relating to organic compounds |
| US5795910A (en) | 1994-10-28 | 1998-08-18 | Cor Therapeutics, Inc. | Method and compositions for inhibiting protein kinases |
| SK286592B6 (sk) * | 1997-07-08 | 2009-01-07 | Bristol-Myers Squibb Company | Derivát epotilónu, farmaceutický prostriedok s jeho obsahom a jeho použitie |
| JP2004292314A (ja) | 2000-12-14 | 2004-10-21 | Chugai Pharmaceut Co Ltd | ケラチノサイト増殖抑制剤 |
| JP2004292315A (ja) | 2000-12-14 | 2004-10-21 | Chugai Pharmaceut Co Ltd | Ｔａｋ１阻害剤 |
| CN1653059A (zh) * | 2002-03-08 | 2005-08-10 | 卫材株式会社 | 用作医药品的大环化合物 |
| US7915306B2 (en) * | 2002-03-08 | 2011-03-29 | Eisai Co., Ltd. | Macrocyclic compounds useful as pharmaceuticals |
| JP5465006B2 (ja) | 2006-08-11 | 2014-04-09 | ユニベルシテ・ドウ・ストラスブール | キナーゼおよびｈｓｐ９０の阻害剤として有用な大環状化合物 |
| WO2008149244A2 (en) * | 2007-06-05 | 2008-12-11 | Nicolas Winssinger | Compositions and methods comprising analogues of radicicol a |
| TW200924749A (en) * | 2007-07-25 | 2009-06-16 | Eisai R & Amp D Man Co Ltd | Zearalenone macrolide derivatives and uses of the same |
| KR101667960B1 (ko) * | 2007-07-25 | 2016-10-20 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 암 치료에서 이용하기 위한 멀티키나아제 억제제 |
| RU2478630C2 (ru) | 2007-12-07 | 2013-04-10 | ЭЙСАН Ар ЭНД Ди МЕНЕДЖМЕНТ КО., ЛТД. | Промежуточные соединения и способы получения зеараленоновых макролидных аналогов |
-
2008
- 2008-12-08 RU RU2010128103/04A patent/RU2478630C2/ru active
- 2008-12-08 MX MX2010005999A patent/MX2010005999A/es active IP Right Grant
- 2008-12-08 WO PCT/US2008/013512 patent/WO2009075823A1/en not_active Ceased
- 2008-12-08 US US12/746,672 patent/US8350059B2/en active Active
- 2008-12-08 BR BRPI0820958-8A patent/BRPI0820958B1/pt active IP Right Grant
- 2008-12-08 CA CA2708141A patent/CA2708141C/en active Active
- 2008-12-08 RU RU2010128096/04A patent/RU2497803C2/ru active
- 2008-12-08 EP EP08860534.0A patent/EP2231635B1/en active Active
- 2008-12-08 MX MX2010006091A patent/MX2010006091A/es active IP Right Grant
- 2008-12-08 JP JP2010536950A patent/JP5492786B2/ja active Active
- 2008-12-08 CN CN2008801195442A patent/CN101889006B/zh active Active
- 2008-12-08 US US12/746,675 patent/US8507696B2/en active Active
- 2008-12-08 JP JP2010536949A patent/JP5496908B2/ja active Active
- 2008-12-08 CN CN200880119543.8A patent/CN101889005B/zh active Active
- 2008-12-08 WO PCT/US2008/013498 patent/WO2009075818A1/en not_active Ceased
- 2008-12-08 BR BRPI0820953-7A patent/BRPI0820953B1/pt active IP Right Grant
- 2008-12-08 CA CA2708143A patent/CA2708143C/en active Active
- 2008-12-08 EP EP08860344.4A patent/EP2231634B1/en active Active
-
2010
- 2010-05-25 IL IL205954A patent/IL205954A/en active IP Right Grant
- 2010-05-26 IL IL205983A patent/IL205983A/en active IP Right Grant
-
2013
- 2013-01-03 US US13/733,562 patent/US20130211103A1/en not_active Abandoned
-
2014
- 2014-03-05 JP JP2014042331A patent/JP2014141498A/ja not_active Withdrawn
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2009533369A5 (https=) | ||
| RU2009105669A (ru) | Способ получения 3-замещенных 2-амино-5-галогенбензамидов | |
| JP2012515142A5 (https=) | ||
| JP2010510976A5 (https=) | ||
| JP6307087B2 (ja) | ベンズアミド化合物の合成に有用な化合物 | |
| JP2018058894A (ja) | （２ｓ，５ｒ）−６−ベンジルオキシ−７−オキソ−１，６−ジアザ−ビシクロ［３．２．１］オクタン−２−カルボン酸のナトリウム塩 | |
| EA038078B1 (ru) | Промежуточные соединения, используемые для синтеза селективного ингибитора протеинкиназы, и способы их получения | |
| RU2013112946A (ru) | Способ получения промежуточных соединений для получения ингибиторов nep | |
| JP4268871B2 (ja) | ピリミジノン化合物及びその薬剤として許容される塩の製造方法 | |
| RU2009111276A (ru) | Способ получения 1-(3, 4-дихлорбензил)-5-октилбигуанида или его соли | |
| JP2011506323A5 (https=) | ||
| TNSN08142A1 (en) | Synthesis of renin inhibitors involving a cycloaddition reaction | |
| CN1869036A (zh) | 7－取代－3－氯吡咯并[3,4－b]吡啶化合物 | |
| EP2958893B1 (en) | Asymmetric synthesis of a substituted pyrrolidine-2-carboxamide | |
| KR101430116B1 (ko) | 스트레커 반응용 촉매를 사용하는 키랄성 α-아미노나이트릴의 제조방법 | |
| CN113754605B (zh) | 一种含氮配体及其制备方法和应用 | |
| KR20090027192A (ko) | (+) 및 (-)-1-(3,4-디클로로페닐)-3-아자비시클로[3.1.0]헥산의 합성 방법 | |
| CA2647590A1 (en) | Process for production of ethylenediamine derivatives having halogenated carbamate group and acyl group, and intermediates for production of the derivatives | |
| RU2010147864A (ru) | Способы получения замещенных гетероциклов -149 | |
| JP4790901B2 (ja) | ４−アミノ−５−シアノイミダゾール誘導体及びその中間体の製造方法 | |
| RU2010128103A (ru) | Промежуточные соединения и способы получения зеараленовых макролидных аналогов | |
| JP4032861B2 (ja) | β−オキソニトリル誘導体又はそのアルカリ金属塩の製法 | |
| KR101453413B1 (ko) | 알파-카르볼린 유도체의 제조방법 | |
| JP4899385B2 (ja) | ３−アミノメチルオキセタン化合物の製法 | |
| JP2016538251A (ja) | ３−アルキルチオ−２−ブロモピリジンの製造方法 |