JP2006521393A5 - - Google Patents
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- Publication number
- JP2006521393A5 JP2006521393A5 JP2006509302A JP2006509302A JP2006521393A5 JP 2006521393 A5 JP2006521393 A5 JP 2006521393A5 JP 2006509302 A JP2006509302 A JP 2006509302A JP 2006509302 A JP2006509302 A JP 2006509302A JP 2006521393 A5 JP2006521393 A5 JP 2006521393A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- carbon moiety
- formula
- substituted carbon
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims description 20
- 238000000034 method Methods 0.000 claims description 18
- 229910052794 bromium Inorganic materials 0.000 claims description 12
- 150000001875 compounds Chemical class 0.000 claims description 12
- 229910052801 chlorine Inorganic materials 0.000 claims description 10
- 229910052740 iodine Inorganic materials 0.000 claims description 7
- 229910052731 fluorine Inorganic materials 0.000 claims description 6
- -1 2-substituted-5-oxo-3-pyrazolidinecarboxylate compound Chemical class 0.000 claims description 5
- 229910052736 halogen Inorganic materials 0.000 claims description 5
- 150000002367 halogens Chemical class 0.000 claims description 5
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 5
- 229910052799 carbon Inorganic materials 0.000 claims description 4
- 239000002904 solvent Substances 0.000 claims description 4
- 229910052727 yttrium Inorganic materials 0.000 claims description 4
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 3
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 3
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 3
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 3
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 claims description 3
- 125000006650 (C2-C4) alkynyl group Chemical group 0.000 claims description 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 3
- 125000004663 dialkyl amino group Chemical group 0.000 claims description 3
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims description 3
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 3
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 3
- 239000002253 acid Substances 0.000 claims description 2
- 125000000217 alkyl group Chemical group 0.000 claims description 2
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims description 2
- 150000001721 carbon Chemical group 0.000 claims description 2
- OAKJQQAXSVQMHS-UHFFFAOYSA-N hydrazine Substances NN OAKJQQAXSVQMHS-UHFFFAOYSA-N 0.000 claims description 2
- 150000002429 hydrazines Chemical class 0.000 claims description 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 2
- 239000002516 radical scavenger Substances 0.000 claims description 2
- 125000003107 substituted aryl group Chemical group 0.000 claims description 2
- 150000003443 succinic acid derivatives Chemical class 0.000 claims description 2
- WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 description 3
- YMWUJEATGCHHMB-UHFFFAOYSA-N Dichloromethane Chemical compound ClCCl YMWUJEATGCHHMB-UHFFFAOYSA-N 0.000 description 3
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 description 3
- HQQTZCPKNZVLFF-UHFFFAOYSA-N 4h-1,2-benzoxazin-3-one Chemical class C1=CC=C2ONC(=O)CC2=C1 HQQTZCPKNZVLFF-UHFFFAOYSA-N 0.000 description 2
- 0 C*c1cc(*)cc(*)c1NC(c1cc(*)n[n]1C1=CC(C)(*)C=CC=*1)=O Chemical compound C*c1cc(*)cc(*)c1NC(c1cc(*)n[n]1C1=CC(C)(*)C=CC=*1)=O 0.000 description 2
- HEDRZPFGACZZDS-UHFFFAOYSA-N Chloroform Chemical compound ClC(Cl)Cl HEDRZPFGACZZDS-UHFFFAOYSA-N 0.000 description 2
- WYURNTSHIVDZCO-UHFFFAOYSA-N Tetrahydrofuran Chemical compound C1CCOC1 WYURNTSHIVDZCO-UHFFFAOYSA-N 0.000 description 2
- PXBFMLJZNCDSMP-UHFFFAOYSA-N 2-Aminobenzamide Chemical class NC(=O)C1=CC=CC=C1N PXBFMLJZNCDSMP-UHFFFAOYSA-N 0.000 description 1
- 150000001412 amines Chemical class 0.000 description 1
- 125000000623 heterocyclic group Chemical group 0.000 description 1
- 238000010992 reflux Methods 0.000 description 1
- 239000000126 substance Substances 0.000 description 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 description 1
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US45756103P | 2003-03-26 | 2003-03-26 | |
| US60/457,561 | 2003-03-26 | ||
| PCT/US2004/009188 WO2004087689A1 (en) | 2003-03-26 | 2004-03-25 | Preparation and use of 2-substituted-5-oxo-3- pyrazolidinecarboxylates |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006521393A JP2006521393A (ja) | 2006-09-21 |
| JP2006521393A5 true JP2006521393A5 (https=) | 2007-04-26 |
| JP4750019B2 JP4750019B2 (ja) | 2011-08-17 |
Family
ID=33131691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006509302A Expired - Fee Related JP4750019B2 (ja) | 2003-03-26 | 2004-03-25 | ２−置換−５−オキソ−３−ピラゾリジンカルボキシレートの製造および使用 |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US7442799B2 (https=) |
| EP (1) | EP1606276B1 (https=) |
| JP (1) | JP4750019B2 (https=) |
| KR (1) | KR101208748B1 (https=) |
| CN (1) | CN100522958C (https=) |
| AT (1) | ATE340791T1 (https=) |
| AU (1) | AU2004225981A1 (https=) |
| BR (1) | BRPI0409049A (https=) |
| DE (1) | DE602004002579T2 (https=) |
| DK (1) | DK1606276T3 (https=) |
| ES (1) | ES2274477T3 (https=) |
| IL (1) | IL169998A (https=) |
| PL (1) | PL1606276T3 (https=) |
| TW (1) | TWI367882B (https=) |
| WO (1) | WO2004087689A1 (https=) |
| ZA (1) | ZA200506096B (https=) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2424840T3 (es) | 2003-01-28 | 2013-10-09 | E.I. Du Pont De Nemours And Company | Insecticidas tipo ciano antranilamida |
| EP1631564A1 (en) | 2003-06-12 | 2006-03-08 | E.I. Dupont De Nemours And Company | Method for preparing fused oxazinones |
| AU2005306363B2 (en) * | 2004-11-18 | 2012-08-09 | E. I. Du Pont De Nemours And Company | Anthranilamide insecticides |
| AU2006283181A1 (en) * | 2005-08-24 | 2007-03-01 | E. I. Du Pont De Nemours And Company | Anthranilamides for controlling invertebrate pests |
| TWI415827B (zh) | 2006-12-21 | 2013-11-21 | Du Pont | 製備２-胺基-５-氰基苯甲酸衍生物之方法 |
| JP5495618B2 (ja) * | 2009-05-21 | 2014-05-21 | 国立大学法人 名古屋工業大学 | 光学活性トリフルオロメチル基含有化合物、その製造方法並びにそれを用いたトリフルオロメチル基含有光学活性アミン類の製造方法 |
| US8871939B2 (en) | 2011-01-28 | 2014-10-28 | E I Du Pont De Nemours And Company | Method for preparing 2-aminobenzamide derivatives |
| CA2894399A1 (en) | 2012-12-06 | 2014-06-12 | Quanticel Pharmaceuticals, Inc. | Histone demethylase inhibitors |
| CN106928183B (zh) * | 2015-12-29 | 2019-09-24 | 沈阳中化农药化工研发有限公司 | 吡啶基吡唑烷酮羧酸类化合物的制备方法 |
| CN106831705B (zh) * | 2016-12-28 | 2021-02-19 | 江苏扬农化工集团有限公司 | 一种吡啶基吡唑烷酮羧酸酯类化合物的合成方法 |
| CN109053726A (zh) * | 2018-09-14 | 2018-12-21 | 烟台万润药业有限公司 | 一种唑吡坦酸的制备方法 |
| AU2020334337A1 (en) * | 2019-08-21 | 2022-03-17 | Gharda Chemicals Limited | Process for synthesis of pyrazolidinone compounds |
| CN110483480A (zh) * | 2019-09-11 | 2019-11-22 | 江苏优普生物化学科技股份有限公司 | 2-(3-氯吡啶-2-基)-5-羟基-3-吡唑烷甲酸乙酯的合成方法 |
| CN111440144A (zh) * | 2020-03-06 | 2020-07-24 | 山东华科化工有限公司 | 一种微通道工业化生产溴代吡唑烷酸的方法 |
| CN111620850B (zh) * | 2020-05-27 | 2021-06-29 | 江苏七洲绿色化工股份有限公司 | 一种1-(3-氯吡啶-2-基)-3-溴-1h-吡唑-5-甲酸酯的制备方法 |
| US11529599B1 (en) | 2021-12-13 | 2022-12-20 | Cana Technology, Inc. | Electromechanical valve sequencing for fluid mixture dispensing devices |
| TW202342443A (zh) | 2022-01-31 | 2023-11-01 | 美商富曼西公司 | 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法 |
| TW202409000A (zh) | 2022-08-29 | 2024-03-01 | 美商富曼西公司 | 用於製備３－鹵代－４，５－二氫－１ｈ－吡唑之高效新方法 |
| WO2025188963A1 (en) | 2024-03-06 | 2025-09-12 | Fmc Corporation | Metal catalyzed synthesis of 2-aminobenzamide derivatives |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL121416C (https=) | 1961-05-31 | |||
| JPH01305071A (ja) | 1988-06-03 | 1989-12-08 | Nippon Oil Co Ltd | オキサゾロン誘導体の製造方法 |
| US5962523A (en) | 1996-10-25 | 1999-10-05 | Discovery Laboratories, Inc. | Methods of using butyric acid derivatives to protect against hair loss |
| DK1187805T3 (da) | 1999-05-18 | 2007-04-16 | Sigma Tau Ind Farmaceuti | Fremgangsmåde til fremstilling af R-(-)-carnitin ud fra S-(-)-chlorravsyre eller ud fra et derivat deraf |
| US7038057B2 (en) * | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| TWI356822B (en) * | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| TWI343376B (en) * | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
-
2004
- 2004-03-09 TW TW093106257A patent/TWI367882B/zh not_active IP Right Cessation
- 2004-03-25 ES ES04758355T patent/ES2274477T3/es not_active Expired - Lifetime
- 2004-03-25 WO PCT/US2004/009188 patent/WO2004087689A1/en not_active Ceased
- 2004-03-25 DE DE602004002579T patent/DE602004002579T2/de not_active Expired - Lifetime
- 2004-03-25 DK DK04758355T patent/DK1606276T3/da active
- 2004-03-25 ZA ZA200506096A patent/ZA200506096B/en unknown
- 2004-03-25 JP JP2006509302A patent/JP4750019B2/ja not_active Expired - Fee Related
- 2004-03-25 EP EP04758355A patent/EP1606276B1/en not_active Expired - Lifetime
- 2004-03-25 AU AU2004225981A patent/AU2004225981A1/en not_active Abandoned
- 2004-03-25 CN CNB2004800081395A patent/CN100522958C/zh not_active Expired - Lifetime
- 2004-03-25 US US10/546,165 patent/US7442799B2/en not_active Expired - Lifetime
- 2004-03-25 AT AT04758355T patent/ATE340791T1/de active
- 2004-03-25 PL PL04758355T patent/PL1606276T3/pl unknown
- 2004-03-25 BR BRPI0409049-7A patent/BRPI0409049A/pt active Search and Examination
-
2005
- 2005-07-31 IL IL169998A patent/IL169998A/en not_active IP Right Cessation
- 2005-09-23 KR KR1020057017883A patent/KR101208748B1/ko not_active Expired - Fee Related
-
2008
- 2008-09-19 US US12/234,063 patent/US7834186B2/en not_active Expired - Lifetime
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