TWI367882B - Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates - Google Patents
Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylatesInfo
- Publication number
- TWI367882B TWI367882B TW093106257A TW93106257A TWI367882B TW I367882 B TWI367882 B TW I367882B TW 093106257 A TW093106257 A TW 093106257A TW 93106257 A TW93106257 A TW 93106257A TW I367882 B TWI367882 B TW I367882B
- Authority
- TW
- Taiwan
- Prior art keywords
- formula
- disclosed
- substituted
- disclosure
- compound
- Prior art date
Links
- -1 2-substituted-5-oxo-3-pyrazolidinecarboxylates Chemical class 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- OAKJQQAXSVQMHS-UHFFFAOYSA-N hydrazine Substances NN OAKJQQAXSVQMHS-UHFFFAOYSA-N 0.000 abstract 1
- 150000002429 hydrazines Chemical class 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 239000002516 radical scavenger Substances 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 150000003443 succinic acid derivatives Chemical class 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
- C09B—ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
- C09B67/00—Influencing the physical, e.g. the dyeing or printing properties of dyestuffs without chemical reactions, e.g. by treating with solvents grinding or grinding assistants, coating of pigments or dyes; Process features in the making of dyestuff preparations; Dyestuff preparations of a special physical nature, e.g. tablets, films
- C09B67/006—Preparation of organic pigments
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Agronomy & Crop Science (AREA)
- Medicinal Chemistry (AREA)
- Plant Pathology (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US45756103P | 2003-03-26 | 2003-03-26 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TW200504050A TW200504050A (en) | 2005-02-01 |
| TWI367882B true TWI367882B (en) | 2012-07-11 |
Family
ID=33131691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW093106257A TWI367882B (en) | 2003-03-26 | 2004-03-09 | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US7442799B2 (https=) |
| EP (1) | EP1606276B1 (https=) |
| JP (1) | JP4750019B2 (https=) |
| KR (1) | KR101208748B1 (https=) |
| CN (1) | CN100522958C (https=) |
| AT (1) | ATE340791T1 (https=) |
| AU (1) | AU2004225981A1 (https=) |
| BR (1) | BRPI0409049A (https=) |
| DE (1) | DE602004002579T2 (https=) |
| DK (1) | DK1606276T3 (https=) |
| ES (1) | ES2274477T3 (https=) |
| IL (1) | IL169998A (https=) |
| PL (1) | PL1606276T3 (https=) |
| TW (1) | TWI367882B (https=) |
| WO (1) | WO2004087689A1 (https=) |
| ZA (1) | ZA200506096B (https=) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1599463T1 (sl) | 2003-01-28 | 2013-10-30 | E.I. Du Pont De Nemours And Company | Ciano antranilamidni insekticidi |
| KR20060008336A (ko) | 2003-06-12 | 2006-01-26 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 융합된 옥사지논 제조 방법 |
| ES2413442T3 (es) * | 2004-11-18 | 2013-07-16 | E. I. Du Pont De Nemours And Company | Insecticidas de antranilamida |
| AU2006283181A1 (en) * | 2005-08-24 | 2007-03-01 | E. I. Du Pont De Nemours And Company | Anthranilamides for controlling invertebrate pests |
| TWI415827B (zh) | 2006-12-21 | 2013-11-21 | Du Pont | 製備２-胺基-５-氰基苯甲酸衍生物之方法 |
| JP5495618B2 (ja) * | 2009-05-21 | 2014-05-21 | 国立大学法人 名古屋工業大学 | 光学活性トリフルオロメチル基含有化合物、その製造方法並びにそれを用いたトリフルオロメチル基含有光学活性アミン類の製造方法 |
| KR20140006007A (ko) | 2011-01-28 | 2014-01-15 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 2-아미노벤즈아미드 유도체의 제조 방법 |
| EP2928471B1 (en) | 2012-12-06 | 2020-10-14 | Celgene Quanticel Research, Inc. | Histone demethylase inhibitors |
| CN106928183B (zh) * | 2015-12-29 | 2019-09-24 | 沈阳中化农药化工研发有限公司 | 吡啶基吡唑烷酮羧酸类化合物的制备方法 |
| CN106831705B (zh) * | 2016-12-28 | 2021-02-19 | 江苏扬农化工集团有限公司 | 一种吡啶基吡唑烷酮羧酸酯类化合物的合成方法 |
| CN109053726A (zh) * | 2018-09-14 | 2018-12-21 | 烟台万润药业有限公司 | 一种唑吡坦酸的制备方法 |
| BR112022003171A2 (pt) * | 2019-08-21 | 2022-05-17 | Gharda Chemicals Ltd | Processo para a síntese de compostos de pirazolidinona |
| CN110483480A (zh) * | 2019-09-11 | 2019-11-22 | 江苏优普生物化学科技股份有限公司 | 2-(3-氯吡啶-2-基)-5-羟基-3-吡唑烷甲酸乙酯的合成方法 |
| CN111440144A (zh) * | 2020-03-06 | 2020-07-24 | 山东华科化工有限公司 | 一种微通道工业化生产溴代吡唑烷酸的方法 |
| CN111620850B (zh) * | 2020-05-27 | 2021-06-29 | 江苏七洲绿色化工股份有限公司 | 一种1-(3-氯吡啶-2-基)-3-溴-1h-吡唑-5-甲酸酯的制备方法 |
| US11529599B1 (en) | 2021-12-13 | 2022-12-20 | Cana Technology, Inc. | Electromechanical valve sequencing for fluid mixture dispensing devices |
| TW202342443A (zh) | 2022-01-31 | 2023-11-01 | 美商富曼西公司 | 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法 |
| TW202409000A (zh) | 2022-08-29 | 2024-03-01 | 美商富曼西公司 | 用於製備３－鹵代－４，５－二氫－１ｈ－吡唑之高效新方法 |
| WO2025188963A1 (en) | 2024-03-06 | 2025-09-12 | Fmc Corporation | Metal catalyzed synthesis of 2-aminobenzamide derivatives |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL279140A (https=) * | 1961-05-31 | |||
| JPH01305071A (ja) | 1988-06-03 | 1989-12-08 | Nippon Oil Co Ltd | オキサゾロン誘導体の製造方法 |
| US5962523A (en) | 1996-10-25 | 1999-10-05 | Discovery Laboratories, Inc. | Methods of using butyric acid derivatives to protect against hair loss |
| JP4584464B2 (ja) | 1999-05-18 | 2010-11-24 | シグマ−タウ・インドゥストリエ・ファルマチェウチケ・リウニテ・ソシエタ・ペル・アチオニ | Ｓ−（−）−クロロコハク酸またはその誘導体からｒ−（−）−カルニチンを調製するための方法 |
| AR036872A1 (es) * | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| TWI327566B (en) * | 2001-08-13 | 2010-07-21 | Du Pont | Novel substituted ihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use |
| DE60236600D1 (de) * | 2001-08-13 | 2010-07-15 | Du Pont | Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung |
| TWI343376B (en) * | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
-
2004
- 2004-03-09 TW TW093106257A patent/TWI367882B/zh not_active IP Right Cessation
- 2004-03-25 DK DK04758355T patent/DK1606276T3/da active
- 2004-03-25 JP JP2006509302A patent/JP4750019B2/ja not_active Expired - Fee Related
- 2004-03-25 DE DE602004002579T patent/DE602004002579T2/de not_active Expired - Lifetime
- 2004-03-25 ZA ZA200506096A patent/ZA200506096B/en unknown
- 2004-03-25 BR BRPI0409049-7A patent/BRPI0409049A/pt active Search and Examination
- 2004-03-25 WO PCT/US2004/009188 patent/WO2004087689A1/en not_active Ceased
- 2004-03-25 US US10/546,165 patent/US7442799B2/en not_active Expired - Lifetime
- 2004-03-25 CN CNB2004800081395A patent/CN100522958C/zh not_active Expired - Lifetime
- 2004-03-25 EP EP04758355A patent/EP1606276B1/en not_active Expired - Lifetime
- 2004-03-25 AU AU2004225981A patent/AU2004225981A1/en not_active Abandoned
- 2004-03-25 ES ES04758355T patent/ES2274477T3/es not_active Expired - Lifetime
- 2004-03-25 PL PL04758355T patent/PL1606276T3/pl unknown
- 2004-03-25 AT AT04758355T patent/ATE340791T1/de active
-
2005
- 2005-07-31 IL IL169998A patent/IL169998A/en not_active IP Right Cessation
- 2005-09-23 KR KR1020057017883A patent/KR101208748B1/ko not_active Expired - Fee Related
-
2008
- 2008-09-19 US US12/234,063 patent/US7834186B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| US20090036686A1 (en) | 2009-02-05 |
| PL1606276T3 (pl) | 2007-01-31 |
| CN100522958C (zh) | 2009-08-05 |
| AU2004225981A1 (en) | 2004-10-14 |
| EP1606276A1 (en) | 2005-12-21 |
| KR20050114693A (ko) | 2005-12-06 |
| TW200504050A (en) | 2005-02-01 |
| ATE340791T1 (de) | 2006-10-15 |
| US20070021468A1 (en) | 2007-01-25 |
| US7834186B2 (en) | 2010-11-16 |
| BRPI0409049A (pt) | 2006-03-28 |
| JP2006521393A (ja) | 2006-09-21 |
| ES2274477T3 (es) | 2007-05-16 |
| CN1764658A (zh) | 2006-04-26 |
| IL169998A (en) | 2011-07-31 |
| JP4750019B2 (ja) | 2011-08-17 |
| EP1606276B1 (en) | 2006-09-27 |
| ZA200506096B (en) | 2006-10-25 |
| KR101208748B1 (ko) | 2012-12-05 |
| WO2004087689A1 (en) | 2004-10-14 |
| US7442799B2 (en) | 2008-10-28 |
| DE602004002579D1 (de) | 2006-11-09 |
| DK1606276T3 (da) | 2007-02-05 |
| DE602004002579T2 (de) | 2007-06-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Annulment or lapse of patent due to non-payment of fees |