JP2006511506A5 - - Google Patents

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Publication number
JP2006511506A5
JP2006511506A5 JP2004554902A JP2004554902A JP2006511506A5 JP 2006511506 A5 JP2006511506 A5 JP 2006511506A5 JP 2004554902 A JP2004554902 A JP 2004554902A JP 2004554902 A JP2004554902 A JP 2004554902A JP 2006511506 A5 JP2006511506 A5 JP 2006511506A5
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JP
Japan
Prior art keywords
hydrogen
derivatives
yloxy
dimethylamine
symbols
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004554902A
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English (en)
Japanese (ja)
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JP4782425B2 (ja
JP2006511506A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/IN2003/000370 external-priority patent/WO2004048328A2/en
Publication of JP2006511506A publication Critical patent/JP2006511506A/ja
Publication of JP2006511506A5 publication Critical patent/JP2006511506A5/ja
Application granted granted Critical
Publication of JP4782425B2 publication Critical patent/JP4782425B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2004554902A 2002-11-28 2003-11-25 N−アリールスルホニル−3−アミノアルコキシインドール Expired - Fee Related JP4782425B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN883MA2002 2002-11-28
IN883/MAS/2002 2002-11-28
PCT/IN2003/000370 WO2004048328A2 (en) 2002-11-28 2003-11-25 N-arylsulfonyl-3-aminoalkoxyindoles

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011043072A Division JP2011116769A (ja) 2002-11-28 2011-02-28 N−アリールスルホニル−3−アミノアルコキシインドール

Publications (3)

Publication Number Publication Date
JP2006511506A JP2006511506A (ja) 2006-04-06
JP2006511506A5 true JP2006511506A5 (https=) 2007-01-18
JP4782425B2 JP4782425B2 (ja) 2011-09-28

Family

ID=34362365

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2004554902A Expired - Fee Related JP4782425B2 (ja) 2002-11-28 2003-11-25 N−アリールスルホニル−3−アミノアルコキシインドール
JP2011043072A Pending JP2011116769A (ja) 2002-11-28 2011-02-28 N−アリールスルホニル−3−アミノアルコキシインドール

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2011043072A Pending JP2011116769A (ja) 2002-11-28 2011-02-28 N−アリールスルホニル−3−アミノアルコキシインドール

Country Status (18)

Country Link
US (2) US7507835B2 (https=)
EP (1) EP1567492B1 (https=)
JP (2) JP4782425B2 (https=)
KR (1) KR100776118B1 (https=)
CN (2) CN1720227A (https=)
AU (1) AU2003285759B2 (https=)
BR (1) BRPI0315958B8 (https=)
CA (1) CA2507505C (https=)
CY (1) CY1114241T1 (https=)
EA (1) EA009193B1 (https=)
ES (1) ES2425143T3 (https=)
MX (1) MXPA05005700A (https=)
NO (1) NO331805B1 (https=)
NZ (1) NZ540842A (https=)
PT (1) PT1567492E (https=)
SI (1) SI1567492T1 (https=)
WO (1) WO2004048328A2 (https=)
ZA (1) ZA200504044B (https=)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA05005700A (es) * 2002-11-28 2005-08-16 Suven Life Sciences Ltd N-arilsulfonil-3-aminoalcoxiindoles.
EA009367B1 (ru) * 2002-12-18 2007-12-28 Сувен Лайф Сайенсиз Лимитед ПРОИЗВОДНЫЕ 5-ТИА-5-ДИОКСО-4b-АЗАИНДЕНО[2,1-a]ИНДЕНА, ОБЛАДАЮЩИЕ АФФИННОСТЬЮ К РЕЦЕПТОРУ СЕРОТОНИНА
AU2004312229B2 (en) 2004-01-02 2010-05-20 Suven Life Sciences Limited Novel Indeno[2,1a]indenes and isoindolo[2,1-a]indoles
BRPI0520579B8 (pt) 2005-08-12 2021-05-25 Suven Life Sciences Ltd composto, processo para a preparação de um composto e composição farmacêutica
KR101250820B1 (ko) 2005-08-16 2013-04-04 수벤 라이프 사이언시스 리미티드 개선된 로사르탄 제조 방법
KR100724095B1 (ko) * 2005-10-21 2007-06-04 한국표준과학연구원 정밀 전류, 전압 및 전력 측정장치
MX2009006077A (es) 2007-01-08 2009-06-17 Suven Life Sciences Ltd Compuestos de 5-(heterociclil)alquil-n-(arilsulfonil)indol y su uso como ligandos de la 5-hidroxitriptamina6.
EP1947085A1 (en) * 2007-01-19 2008-07-23 Laboratorios del Dr. Esteve S.A. Substituted indole sulfonamide compounds, their preparation and use as medicaments
EA016594B1 (ru) 2007-05-03 2012-06-29 Сувен Лайф Сайенсиз Лимитед Производные 1-(аминоалкоксиарилсульфонил)индола в качестве 5-нтлигандов
US7964627B2 (en) 2007-10-26 2011-06-21 Suven Life Sciences Limited Amino arylsulfonamide compounds and their use as 5-HT6 ligands
AR072297A1 (es) * 2008-06-27 2010-08-18 Novartis Ag Derivados de indol-2-il-piridin-3-ilo, composicion farmaceutica que los comprende y su uso en medicamentos para el tratamiento de enfermedades mediadas por la sintasa aldosterona.
EP2149573A1 (en) * 2008-08-01 2010-02-03 Laboratorios Del. Dr. Esteve, S.A. Substituted indole sulfonamide compounds their preparation and use as medicaments
US8318725B2 (en) 2008-09-17 2012-11-27 Suven Life Sciences Limited Aryl indolyl sulfonamide compounds and their use as 5-HT6 ligands
CA2737282C (en) 2008-09-17 2014-03-25 Suven Life Sciences Limited Aryl sulfonamide amine compounds and their use as 5-ht6 ligands
JP5628937B2 (ja) 2010-01-05 2014-11-19 スベン ライフ サイエンシズ リミティド 5−ht6受容体リガンドとしてのスルホン化合物
EP2932922B1 (en) * 2012-12-13 2018-09-05 Olympus Corporation Treatment device
DE102013013602A1 (de) * 2013-08-19 2015-02-19 Trützschler GmbH + Co KG Textilmaschinenfabrik Vorrichtung an einer Karde oder Krempel für Baumwolle, Chemiefasern u. dgl. mit einer drehbaren Abstreifwalze
EP3083588B1 (en) 2013-12-20 2020-12-09 Sunshine Lake Pharma Co., Ltd. Aromatic heterocyclic compounds and their application in pharmaceuticals

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE111890C (https=)
US723550A (en) * 1902-09-15 1903-03-24 Eagle Lock Co Padlock.
CH481104A (de) * 1967-01-25 1969-11-15 Geigy Ag J R Verfahren zur Herstellung von neuen Indolderivaten
US3860608A (en) * 1969-05-27 1975-01-14 Novo Terapeutisk Labor As 3-aminoalkyloxyindoles
US3860609A (en) * 1969-05-27 1975-01-14 Novo Terapeutisk Labor As 3-aminoalkyloxyindoles
GB1306230A (https=) * 1969-05-27 1973-02-07
ZA795239B (en) 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds
ZA815541B (en) * 1980-08-12 1983-03-30 Glaxo Group Ltd Heterocyclic compounds
JPS57200362A (en) 1981-06-05 1982-12-08 Mitsui Toatsu Chem Inc Preparation of indoxyl
GB8600397D0 (en) 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
GB8719167D0 (en) 1987-08-13 1987-09-23 Glaxo Group Ltd Chemical compounds
JPH01139564A (ja) * 1987-08-31 1989-06-01 Terumo Corp N−置換インドールエステル化合物、その製造法ならびに該化合物を用いた試験組成物および試験具
GB8724912D0 (en) 1987-10-23 1987-11-25 Wellcome Found Indole derivatives
GB8819024D0 (en) 1988-08-10 1988-09-14 Glaxo Group Ltd Chemical compounds
IL96891A0 (en) 1990-01-17 1992-03-29 Merck Sharp & Dohme Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them
CA2042295A1 (fr) 1990-05-15 1991-11-16 Jacques Chauveau Derives de mediateurs endogenes, leurs sels, procede de preparation, applications, et compositions les renfermant
PT97888B (pt) 1990-06-07 1998-12-31 Zeneca Ltd Processo para a preparacao de compostos heterociclicos derivados de indol e de composicoes farmaceuticas que os contem
CZ283018B6 (cs) 1991-02-01 1997-12-17 Merck Sharp And Dohme Limited Deriváty imidazolu, triazolu a tetrazolu a farmaceutické přípravky na jejich bázi
GB9113802D0 (en) 1991-06-26 1991-08-14 Smithkline Beecham Plc Medicaments
GB9210400D0 (en) 1992-05-15 1992-07-01 Merck Sharp & Dohme Therapeutic agents
KR940007001A (ko) 1992-09-16 1994-04-26 최승주 새로운 n-신나모일-2-메틸-5-메톡시-3-인돌 아세트산 에스테르, 그 제조방법 및 이를 함유하는 약학적 제제
IL130169A (en) 1999-05-27 2006-08-20 Neurim Pharma 1991 Indole derivatives, and pharmaceutical preparations, skin protection preparations, and cosmetics containing them
FR2799757B1 (fr) 1999-10-15 2001-12-14 Adir Nouveaux derives polycycliques azaindoliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2821843B1 (fr) * 2001-03-12 2003-05-09 Servier Lab Nouveaux derives d'isoindoloindolones, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
DK1523486T3 (da) * 2002-06-21 2008-03-03 Suven Life Sciences Ltd Tetracykliske arylsulfonylindoler med serotoninreceptor-affinitet
ATE373425T1 (de) * 2002-07-22 2007-10-15 Basf Ag Synergistiche herbizide zusammensetzungen
MXPA05005700A (es) * 2002-11-28 2005-08-16 Suven Life Sciences Ltd N-arilsulfonil-3-aminoalcoxiindoles.

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