JP2005530847A5 - - Google Patents
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- Publication number
- JP2005530847A5 JP2005530847A5 JP2004516609A JP2004516609A JP2005530847A5 JP 2005530847 A5 JP2005530847 A5 JP 2005530847A5 JP 2004516609 A JP2004516609 A JP 2004516609A JP 2004516609 A JP2004516609 A JP 2004516609A JP 2005530847 A5 JP2005530847 A5 JP 2005530847A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- isothiazolecarboxamide
- dichloro
- process according
- aminocarbonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 238000000034 method Methods 0.000 claims 7
- ZMXDDKWLCZADIW-UHFFFAOYSA-N N,N-Dimethylformamide Chemical compound CN(C)C=O ZMXDDKWLCZADIW-UHFFFAOYSA-N 0.000 claims 6
- PXBFMLJZNCDSMP-UHFFFAOYSA-N 2-Aminobenzamide Chemical compound NC(=O)C1=CC=CC=C1N PXBFMLJZNCDSMP-UHFFFAOYSA-N 0.000 claims 2
- 239000012024 dehydrating agents Substances 0.000 claims 2
- 239000003085 diluting agent Substances 0.000 claims 2
- VSCBEYLFHZIKQA-UHFFFAOYSA-N n-(2-carbamoylphenyl)-3,4-dichloro-1,2-thiazole-5-carboxamide Chemical compound NC(=O)C1=CC=CC=C1NC(=O)C1=C(Cl)C(Cl)=NS1 VSCBEYLFHZIKQA-UHFFFAOYSA-N 0.000 claims 2
- XHXFXVLFKHQFAL-UHFFFAOYSA-N phosphoryl trichloride Chemical compound ClP(Cl)(Cl)=O XHXFXVLFKHQFAL-UHFFFAOYSA-N 0.000 claims 2
- FYSNRJHAOHDILO-UHFFFAOYSA-N thionyl chloride Chemical compound ClS(Cl)=O FYSNRJHAOHDILO-UHFFFAOYSA-N 0.000 claims 2
- MSSXWKAJMRSAGF-UHFFFAOYSA-N 3,4-dichloro-1,2-thiazole-5-carbonyl chloride Chemical compound ClC(=O)C=1SN=C(Cl)C=1Cl MSSXWKAJMRSAGF-UHFFFAOYSA-N 0.000 claims 1
- YGYAWVDWMABLBF-UHFFFAOYSA-N Phosgene Chemical compound ClC(Cl)=O YGYAWVDWMABLBF-UHFFFAOYSA-N 0.000 claims 1
- 239000002253 acid Substances 0.000 claims 1
- 238000006243 chemical reaction Methods 0.000 claims 1
- QQVDYSUDFZZPSU-UHFFFAOYSA-M chloromethylidene(dimethyl)azanium;chloride Chemical compound [Cl-].C[N+](C)=CCl QQVDYSUDFZZPSU-UHFFFAOYSA-M 0.000 claims 1
- WLPCAERCXQSYLQ-UHFFFAOYSA-N isotianil Chemical compound ClC1=NSC(C(=O)NC=2C(=CC=CC=2)C#N)=C1Cl WLPCAERCXQSYLQ-UHFFFAOYSA-N 0.000 claims 1
- 239000000203 mixture Substances 0.000 claims 1
- 238000005580 one pot reaction Methods 0.000 claims 1
- 239000002904 solvent Substances 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10228732A DE10228732A1 (de) | 2002-06-27 | 2002-06-27 | Verfahren zur Herstellung von 3,4-Dichlor-N-(2-cyano-phenyl)-5-isothiazolcarboxamid |
| PCT/EP2003/006360 WO2004002968A1 (de) | 2002-06-27 | 2003-06-17 | Verfahren zur herstellung von 3,4-dichlor-n-(2-cyano-phenyl)-5-isothiazolcarboxamid |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005530847A JP2005530847A (ja) | 2005-10-13 |
| JP2005530847A5 true JP2005530847A5 (enExample) | 2006-08-10 |
| JP4551762B2 JP4551762B2 (ja) | 2010-09-29 |
Family
ID=29723489
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004516609A Expired - Lifetime JP4551762B2 (ja) | 2002-06-27 | 2003-06-17 | ３，４−ジクロロ−ｎ−（２−シアノフェニル）−５−イソチアゾールカルボキサミドの製造方法 |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1519926B1 (enExample) |
| JP (1) | JP4551762B2 (enExample) |
| KR (1) | KR101069222B1 (enExample) |
| CN (1) | CN1325483C (enExample) |
| AT (1) | ATE308530T1 (enExample) |
| AU (1) | AU2003238510A1 (enExample) |
| DE (2) | DE10228732A1 (enExample) |
| TW (1) | TWI266766B (enExample) |
| WO (1) | WO2004002968A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102005035617A1 (de) | 2005-07-29 | 2007-02-15 | Bayer Cropscience Ag | Verfahren zur Herstellung von 3,4-Dichlor-N-(2-cyano-phenyl)-5-isothiazolcarboxamid |
| CN103483287B (zh) * | 2013-10-12 | 2015-07-08 | 南开大学 | 一类含3,4-二氯异噻唑的双酰胺类化合物及其制备方法和用途 |
| IL271148B (en) * | 2017-06-14 | 2022-08-01 | Bayer Ag | Process for preparing 3,4-dichloro-n-(2-cyanophenyl)-5-isothiazolecarboxamide |
| TW201943708A (zh) * | 2018-04-06 | 2019-11-16 | 德商拜耳廠股份有限公司 | 製備３，４－二氯－ｎ－（２－氰苯基）－５－異噻唑羧醯胺之方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2115625B2 (de) * | 1971-03-31 | 1978-07-06 | Basf Ag, 6700 Ludwigshafen | Verfahren zur Herstellung von N-o-Cyanophenyl-N', N'-disubstituierten Formamidinen und deren Salzen |
| DE2115624A1 (de) * | 1971-03-31 | 1972-10-12 | Badische Anilin & Soda Fabrik AG, 6700 Ludwigshafen | Verfahren zur Herstellung von o Amino benzonitrilen |
| DE19750012A1 (de) * | 1997-11-12 | 1999-05-20 | Bayer Ag | Isothiazolcarbonsäureamide |
-
2002
- 2002-06-27 DE DE10228732A patent/DE10228732A1/de not_active Withdrawn
-
2003
- 2003-06-17 AT AT03732578T patent/ATE308530T1/de not_active IP Right Cessation
- 2003-06-17 WO PCT/EP2003/006360 patent/WO2004002968A1/de not_active Ceased
- 2003-06-17 JP JP2004516609A patent/JP4551762B2/ja not_active Expired - Lifetime
- 2003-06-17 CN CNB038203294A patent/CN1325483C/zh not_active Expired - Lifetime
- 2003-06-17 KR KR1020047021038A patent/KR101069222B1/ko not_active Expired - Lifetime
- 2003-06-17 DE DE50301572T patent/DE50301572D1/de not_active Expired - Lifetime
- 2003-06-17 AU AU2003238510A patent/AU2003238510A1/en not_active Abandoned
- 2003-06-17 EP EP03732578A patent/EP1519926B1/de not_active Expired - Lifetime
- 2003-06-26 TW TW092117350A patent/TWI266766B/zh not_active IP Right Cessation
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