JP2005512985A5 - - Google Patents
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- Publication number
- JP2005512985A5 JP2005512985A5 JP2003540160A JP2003540160A JP2005512985A5 JP 2005512985 A5 JP2005512985 A5 JP 2005512985A5 JP 2003540160 A JP2003540160 A JP 2003540160A JP 2003540160 A JP2003540160 A JP 2003540160A JP 2005512985 A5 JP2005512985 A5 JP 2005512985A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- halogen
- optionally substituted
- phenyl
- carbon atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 229910052736 halogen Inorganic materials 0.000 claims 15
- 150000002367 halogens Chemical class 0.000 claims 15
- -1 cyano, carboxyl Chemical group 0.000 claims 11
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 10
- 125000004432 carbon atom Chemical group C* 0.000 claims 9
- 125000000217 alkyl group Chemical group 0.000 claims 8
- 150000001875 compounds Chemical class 0.000 claims 7
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 3
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims 2
- 125000003282 alkyl amino group Chemical group 0.000 claims 2
- 239000003085 diluting agent Substances 0.000 claims 2
- 229910052739 hydrogen Inorganic materials 0.000 claims 2
- 239000001257 hydrogen Substances 0.000 claims 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims 2
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims 1
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims 1
- FHFIXRRHKSMREA-UHFFFAOYSA-N 2-(thiophen-2-ylmethylsulfinyl)-5-(trifluoromethyl)pyrimidine Chemical compound N1=CC(C(F)(F)F)=CN=C1S(=O)CC1=CC=CS1 FHFIXRRHKSMREA-UHFFFAOYSA-N 0.000 claims 1
- DACORWPQRQVHBR-UHFFFAOYSA-N 2-(thiophen-2-ylmethylsulfonyl)-5-(trifluoromethyl)pyrimidine Chemical compound N1=CC(C(F)(F)F)=CN=C1S(=O)(=O)CC1=CC=CS1 DACORWPQRQVHBR-UHFFFAOYSA-N 0.000 claims 1
- IVTRMSHONMYNDK-UHFFFAOYSA-N 2-benzylsulfanyl-4-chloro-5-methylpyrimidine Chemical compound N1=C(Cl)C(C)=CN=C1SCC1=CC=CC=C1 IVTRMSHONMYNDK-UHFFFAOYSA-N 0.000 claims 1
- BDOPQKITZWRPQM-UHFFFAOYSA-N 2-benzylsulfonyl-5-(trifluoromethyl)pyrimidine Chemical compound N1=CC(C(F)(F)F)=CN=C1S(=O)(=O)CC1=CC=CC=C1 BDOPQKITZWRPQM-UHFFFAOYSA-N 0.000 claims 1
- WOOGFIPTSBYUFR-UHFFFAOYSA-N 4,6-dichloro-5-methyl-2-(naphthalen-2-ylmethylsulfanyl)pyrimidine Chemical compound N1=C(Cl)C(C)=C(Cl)N=C1SCC1=CC=C(C=CC=C2)C2=C1 WOOGFIPTSBYUFR-UHFFFAOYSA-N 0.000 claims 1
- NWKNAOQJLIJBGN-UHFFFAOYSA-N 4-chloro-2-[(2,4-dichlorophenyl)methylsulfanyl]-5-methylpyrimidine Chemical compound N1=C(Cl)C(C)=CN=C1SCC1=CC=C(Cl)C=C1Cl NWKNAOQJLIJBGN-UHFFFAOYSA-N 0.000 claims 1
- DHHHQULBJQNTGM-UHFFFAOYSA-N 4-chloro-2-[(4-chlorophenyl)methylsulfanyl]-5-methylpyrimidine Chemical compound N1=C(Cl)C(C)=CN=C1SCC1=CC=C(Cl)C=C1 DHHHQULBJQNTGM-UHFFFAOYSA-N 0.000 claims 1
- DWWFADHDYAGCQG-UHFFFAOYSA-N 4-chloro-2-[chloro(phenyl)methyl]sulfanyl-5-methylpyrimidine Chemical compound N1=C(Cl)C(C)=CN=C1SC(Cl)C1=CC=CC=C1 DWWFADHDYAGCQG-UHFFFAOYSA-N 0.000 claims 1
- XVYALGAWXBETTK-UHFFFAOYSA-N 5-methyl-2-[(1-methyl-5-nitroimidazol-2-yl)methylsulfanyl]pyrimidine Chemical compound N1=CC(C)=CN=C1SCC1=NC=C([N+]([O-])=O)N1C XVYALGAWXBETTK-UHFFFAOYSA-N 0.000 claims 1
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical class O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims 1
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims 1
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 claims 1
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims 1
- 125000004414 alkyl thio group Chemical group 0.000 claims 1
- 125000001769 aryl amino group Chemical group 0.000 claims 1
- 125000003236 benzoyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C(*)=O 0.000 claims 1
- 239000003054 catalyst Substances 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000004663 dialkyl amino group Chemical group 0.000 claims 1
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims 1
- 125000004472 dialkylaminosulfonyl group Chemical group 0.000 claims 1
- 239000000945 filler Substances 0.000 claims 1
- 125000002541 furyl group Chemical group 0.000 claims 1
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 claims 1
- 230000002363 herbicidal effect Effects 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 125000001624 naphthyl group Chemical group 0.000 claims 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 1
- 125000002971 oxazolyl group Chemical group 0.000 claims 1
- 239000007800 oxidant agent Substances 0.000 claims 1
- 230000001590 oxidative effect Effects 0.000 claims 1
- 125000000951 phenoxy group Chemical group [H]C1=C([H])C([H])=C(O*)C([H])=C1[H] 0.000 claims 1
- 125000003170 phenylsulfonyl group Chemical group C1(=CC=CC=C1)S(=O)(=O)* 0.000 claims 1
- 125000004076 pyridyl group Chemical group 0.000 claims 1
- 125000000714 pyrimidinyl group Chemical group 0.000 claims 1
- 125000001424 substituent group Chemical group 0.000 claims 1
- 239000004094 surface-active agent Substances 0.000 claims 1
- 125000000335 thiazolyl group Chemical group 0.000 claims 1
- 125000001544 thienyl group Chemical group 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10154075A DE10154075A1 (de) | 2001-11-02 | 2001-11-02 | Substituierte Pyrimidine |
| PCT/EP2002/011744 WO2003037878A1 (de) | 2001-11-02 | 2002-10-21 | Substituierte pyrimidine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005512985A JP2005512985A (ja) | 2005-05-12 |
| JP2005512985A5 true JP2005512985A5 (https=) | 2006-01-05 |
Family
ID=7704536
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003540160A Pending JP2005512985A (ja) | 2001-11-02 | 2002-10-21 | 置換ピリミジン化合物 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20050065166A1 (https=) |
| EP (1) | EP1444208A1 (https=) |
| JP (1) | JP2005512985A (https=) |
| AR (1) | AR037130A1 (https=) |
| DE (1) | DE10154075A1 (https=) |
| WO (1) | WO2003037878A1 (https=) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2477046C2 (ru) * | 2006-11-22 | 2013-03-10 | Сумитомо Кемикал Компани, Лимитед | Агент для ингибирования сигнальной функции цитокинина |
| US8097712B2 (en) | 2007-11-07 | 2012-01-17 | Beelogics Inc. | Compositions for conferring tolerance to viral disease in social insects, and the use thereof |
| US8962584B2 (en) | 2009-10-14 | 2015-02-24 | Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd. | Compositions for controlling Varroa mites in bees |
| ES2641642T3 (es) | 2010-03-08 | 2017-11-10 | Monsanto Technology Llc | Moléculas de polinucleótido para regulación génica en plantas |
| MX342856B (es) | 2011-09-13 | 2016-10-13 | Monsanto Technology Llc | Metodos y composiciones para el control de malezas. |
| AU2012308753B2 (en) | 2011-09-13 | 2018-05-17 | Monsanto Technology Llc | Methods and compositions for weed control |
| CN103974967A (zh) | 2011-09-13 | 2014-08-06 | 孟山都技术公司 | 用于杂草控制的方法和组合物 |
| US10806146B2 (en) | 2011-09-13 | 2020-10-20 | Monsanto Technology Llc | Methods and compositions for weed control |
| US10829828B2 (en) | 2011-09-13 | 2020-11-10 | Monsanto Technology Llc | Methods and compositions for weed control |
| BR112014005958A2 (pt) | 2011-09-13 | 2020-10-13 | Monsanto Technology Llc | métodos e composições químicas agrícolas para controle de planta, método de redução de expressão de um gene accase em uma planta, cassete de expressão microbiana, método para fazer um polinucleotídeo, método de identificação de polinucleotídeos úteis na modulação de expressão do gene accase e composição herbicida |
| US10760086B2 (en) | 2011-09-13 | 2020-09-01 | Monsanto Technology Llc | Methods and compositions for weed control |
| UA116089C2 (uk) | 2011-09-13 | 2018-02-12 | Монсанто Текнолоджи Ллс | Спосіб та композиція для боротьби з бур'янами (варіанти) |
| EP3434779A1 (en) | 2011-09-13 | 2019-01-30 | Monsanto Technology LLC | Methods and compositions for weed control |
| US10240161B2 (en) | 2012-05-24 | 2019-03-26 | A.B. Seeds Ltd. | Compositions and methods for silencing gene expression |
| US10683505B2 (en) | 2013-01-01 | 2020-06-16 | Monsanto Technology Llc | Methods of introducing dsRNA to plant seeds for modulating gene expression |
| WO2014106837A2 (en) | 2013-01-01 | 2014-07-10 | A. B. Seeds Ltd. | ISOLATED dsRNA MOLECULES AND METHODS OF USING SAME FOR SILENCING TARGET MOLECULES OF INTEREST |
| EP2971185A4 (en) | 2013-03-13 | 2017-03-08 | Monsanto Technology LLC | Methods and compositions for weed control |
| BR112015022797A2 (pt) | 2013-03-13 | 2017-11-07 | Monsanto Technology Llc | método para controle de ervas daninhas, composição herbicida, cassete de expressão microbiano e método de produção de polinucleotídeo |
| US10568328B2 (en) | 2013-03-15 | 2020-02-25 | Monsanto Technology Llc | Methods and compositions for weed control |
| RU2703498C2 (ru) | 2013-07-19 | 2019-10-17 | Монсанто Текнолоджи Ллс | Композиции и способы борьбы с leptinotarsa |
| US9850496B2 (en) | 2013-07-19 | 2017-12-26 | Monsanto Technology Llc | Compositions and methods for controlling Leptinotarsa |
| HUE070313T2 (hu) | 2013-11-04 | 2025-05-28 | Greenlight Biosciences Inc | Ízeltlábú paraziták és kártevõfertõzöttség szabályozására szolgáló készítmények és eljárások |
| UA119253C2 (uk) | 2013-12-10 | 2019-05-27 | Біолоджикс, Інк. | Спосіб боротьби із вірусом у кліща varroa та у бджіл |
| AU2015206585A1 (en) | 2014-01-15 | 2016-07-21 | Monsanto Technology Llc | Methods and compositions for weed control using EPSPS polynucleotides |
| WO2015125858A1 (ja) * | 2014-02-24 | 2015-08-27 | 日本曹達株式会社 | ヘテロアリール化合物およびその用途 |
| BR112016022711A2 (pt) | 2014-04-01 | 2017-10-31 | Monsanto Technology Llc | composições e métodos para controle de pragas de inseto |
| US10988764B2 (en) | 2014-06-23 | 2021-04-27 | Monsanto Technology Llc | Compositions and methods for regulating gene expression via RNA interference |
| EP3161138A4 (en) | 2014-06-25 | 2017-12-06 | Monsanto Technology LLC | Methods and compositions for delivering nucleic acids to plant cells and regulating gene expression |
| RU2021123470A (ru) | 2014-07-29 | 2021-09-06 | Монсанто Текнолоджи Ллс | Композиции и способы борьбы с насекомыми-вредителями |
| BR112017003295A2 (pt) | 2014-09-19 | 2018-01-23 | Isagro Spa | 1,3,4-tiadiazóis com uma atividade herbicida, suas composições agronômicas e uso relativo |
| JP6942632B2 (ja) | 2015-01-22 | 2021-09-29 | モンサント テクノロジー エルエルシー | Leptinotarsa防除用組成物及びその方法 |
| US10883103B2 (en) | 2015-06-02 | 2021-01-05 | Monsanto Technology Llc | Compositions and methods for delivery of a polynucleotide into a plant |
| EP3302030A4 (en) | 2015-06-03 | 2019-04-24 | Monsanto Technology LLC | METHOD AND COMPOSITIONS FOR INTRODUCING NUCLEIC ACIDS IN PLANTS |
| IT201800009385A1 (it) | 2018-10-11 | 2020-04-11 | Isagro Spa | Derivati caffeinici ad attività nematocida, loro composizioni agronomiche e relativo uso |
| IT201900001339A1 (it) | 2019-01-30 | 2020-07-30 | Isagro Spa | Derivati teofillinici ad attività nematocida, loro composizioni agronomiche e relativo uso |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4057634A (en) * | 1974-01-24 | 1977-11-08 | Hoechst Aktiengesellschaft | Antiprotozoal(1-alkyl-5-nitro-imidazolyl-2-alkyl)-pyridazines |
| DE2403340A1 (de) * | 1974-01-24 | 1975-07-31 | Hoechst Ag | (1-alkyl-5-nitro-imidazolyl-2-alkyl)- heteroaryl-verbindungen und verfahren zu ihrer herstellung |
| ATE16799T1 (de) * | 1980-01-10 | 1985-12-15 | Nyegaard & Co As | Pyrimidin-2-sulfide und ihre s-oxide zur verwendung in der medizin, die verbindungen enthaltende pharmazeutische zusammensetzungen, verfahren zu ihrer herstellung und die verbindungen an sich, sofern sie neu sind. |
| GB2135992B (en) * | 1983-01-11 | 1986-09-24 | Nyegaard & Co As | Substituted pyrimidines and processes for their preparation |
| GB8712396D0 (en) * | 1987-05-27 | 1987-07-01 | May & Baker Ltd | Composition of matter |
| JPH0559015A (ja) * | 1991-06-26 | 1993-03-09 | Otsuka Chem Co Ltd | ピリミジン誘導体及び該誘導体を有効成分とする除草剤 |
| KR100354309B1 (ko) * | 1993-11-12 | 2003-01-06 | 파마시아 앤드 업존 캄파니 | 피리미딘-티오알킬및알킬에테르화합물 |
-
2001
- 2001-11-02 DE DE10154075A patent/DE10154075A1/de not_active Withdrawn
-
2002
- 2002-10-21 JP JP2003540160A patent/JP2005512985A/ja active Pending
- 2002-10-21 US US10/493,781 patent/US20050065166A1/en not_active Abandoned
- 2002-10-21 WO PCT/EP2002/011744 patent/WO2003037878A1/de not_active Ceased
- 2002-10-21 EP EP02777320A patent/EP1444208A1/de not_active Withdrawn
- 2002-10-29 AR ARP020104107A patent/AR037130A1/es unknown
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