AR037130A1 - Pirimidinas substituidas - Google Patents
Pirimidinas substituidasInfo
- Publication number
- AR037130A1 AR037130A1 ARP020104107A ARP020104107A AR037130A1 AR 037130 A1 AR037130 A1 AR 037130A1 AR P020104107 A ARP020104107 A AR P020104107A AR P020104107 A ARP020104107 A AR P020104107A AR 037130 A1 AR037130 A1 AR 037130A1
- Authority
- AR
- Argentina
- Prior art keywords
- halogen
- alkyl
- substituted
- appropriate
- alkoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/38—One sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Pirimidinas substituidas de la fórmula general (1) a su uso como agentes para el tratamiento de las plantas, especialmente como herbicidas y a procedimientos para su preparación. Reivindicación 1: Compuesto de la fórmula general (1) en la que; n significa los números 0, 1 ó 2; A significa alcanodiilo de cadena lineal o de cadena ramificada C1-6; R1 significa, hidrógeno, halógeno, alquilo C1-6 substituido, en caso dado, por halógeno o por alcoxi C1-4, o significa fenilo substituido, en caso dado, por halógeno o por alquilo C1-4; R2 significa alquilo C1-6 sustituido, en caso dado, por halógeno o por alcoxi C1-4, significa cicloalquilo C3-8 sustituido, en caso dado, por halógeno o por alquilo C1-4, o significa fenil-alquilo C1-4 substituido , en caso dado, por halógeno o por alquilo C1-4, o junto con R1 o junto con R3 significa, respectivamente, alcanodiilo C3-5 substituido, en caso dado, por alquilo C1-4 o un benzo-agrupamiento substituido, en caso dado, por halógeno o por alquilo C1-4; R3 significa hidrógeno, halógeno, alquilo C1-6 substituido, en caso dado, por halógeno o por alcoxi C1-4, o fenilo substituido, en caso dado, por halógeno o por alquilo C1-4; y Z significa fenilo, naftilo, piridinilo, pirimidinilo, furilo, tienilo, oxazolilo o tiazolilo, substituidos respectivamente, en caso dado, eligiéndose respectivamente los posibles sustituyentes preferentemente entre la siguiente enumeración: nitro, ciano, carboxilo, carbamoílo, tiocarbomoílo, halógeno; alquilo, alcoxi, alcoxicarbonilo, alquiltio, alquilsulfinilo, alquilsulfonilo, alquilamino, alquilaminocarbonilo o alquilcarbonilamino con, respectivamente C1-6 en los grupos alquilo, substituidos respectivamente, en caso dado, por ciano, carboxilo, carbamoílo, tiocarbamoílo, halógeno, alcoxi C1-4, alquiltio C1-4, alquilsulfinilo C1-4 o alquilsulfonilo C1-4; alquilendioxi C1-2, dialquilamino, dialquilaminocarbonilo o dialquilaminosulfonilo con, respectivamente C1-4 en los grupos alquilo, substituidos respectivamente, en caso dado, por halógeno; fenilo, fenoxi, feniltio, fenilsulfinilo, fenilsulfonilo, fenilamino, fenilcarbonilamino, fenil-alquilo C1-4, fenil-alcoxi C1-4, fenoxi-alquilo C1-4, fenil-alquiltio C1-4, fenil-alquilsulfinilo C1-4, fenil-alquilsulfonilo C1-4, fenil-alquilamino C1-4, sustituidos respectivamente, en cada dado, nitro, ciano, carboxilo, carbamoilo, tiocarbamoilo, halógeno alquilo C1-4, halógenoalquilo C1-4, alcoxi C1-4, por halógenoalcoxi C1-4, alquiltio C1-4, halógenoalquiltio C1-4, alquilsulfinilo C1-4, halógenoalquilsulfinilo C1-4, alquilsulfonilo C1-4 o halógenoalquilsulfonilo C1-4; quedando excluidos los compuestos conocidos con anterioridad 2-benciltio-4-cloro-5metil-pirimidina, 4-cloro-2-(2,4-diclorobenciltio)-5-metilpirimidina, 4-cloro-2-(cloro-benciltio)-5-metilpirimidina y 4-cloro-2-(4-cloro-benciltio)-5-metilpirimidina (véase la publicación J. Org. Chem. 27 (1962), 181-185), el compuesto 4,6-dicloro-5metil-2-(naftalen-2-ilmetiltio)pirimidina, el compuesto 5-metil-2-[(1-metil-5-nitro-1H-imidazol-2-il)metiltio]-pirimidina, así como los compuestos 2-(tien-2-ilmetilsulfonil)-5-triflúormetilpirimidina, 2-fenilmetiltio-5-triflúormetilpirimidina, 2-(tien-2-ilmetiltio)-5-triflúormetilpirimidina, 2-fenilmetilsulfonil-5-triflúormetilpirimidina y 2-(tien-2-ilmetilsulfinil)-5-triflúormetilpirimidina.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10154075A DE10154075A1 (de) | 2001-11-02 | 2001-11-02 | Substituierte Pyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR037130A1 true AR037130A1 (es) | 2004-10-20 |
Family
ID=7704536
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP020104107A AR037130A1 (es) | 2001-11-02 | 2002-10-29 | Pirimidinas substituidas |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20050065166A1 (es) |
| EP (1) | EP1444208A1 (es) |
| JP (1) | JP2005512985A (es) |
| AR (1) | AR037130A1 (es) |
| DE (1) | DE10154075A1 (es) |
| WO (1) | WO2003037878A1 (es) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20140054433A (ko) | 2006-11-22 | 2014-05-08 | 스미또모 가가꾸 가부시끼가이샤 | 사이토카이닌 신호전달을 저해할 수 있는 물질 |
| US8097712B2 (en) | 2007-11-07 | 2012-01-17 | Beelogics Inc. | Compositions for conferring tolerance to viral disease in social insects, and the use thereof |
| US8962584B2 (en) | 2009-10-14 | 2015-02-24 | Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd. | Compositions for controlling Varroa mites in bees |
| PE20130649A1 (es) | 2010-03-08 | 2013-07-13 | Monsanto Technology Llc | Moleculas polinucleotidicas para regulacion genetica en plantas |
| MX348495B (es) | 2011-09-13 | 2017-06-14 | Monsanto Technology Llc | Metodos y composiciones para el control de malezas. |
| BR112014005795A2 (pt) | 2011-09-13 | 2020-12-08 | Monsanto Technology Llc | métodos de controle de plantas, de redução da expressão de um gene de hppd de uma planta, de preparação de um nucleotídeo, e de identificação de polinucleotídeos úteis na modulação da expressão do gene de hppd no tratamento externo de uma planta, composições e cassete de expressão microbiana |
| US10806146B2 (en) | 2011-09-13 | 2020-10-20 | Monsanto Technology Llc | Methods and compositions for weed control |
| US10829828B2 (en) | 2011-09-13 | 2020-11-10 | Monsanto Technology Llc | Methods and compositions for weed control |
| WO2013040033A1 (en) | 2011-09-13 | 2013-03-21 | Monsanto Technology Llc | Methods and compositions for weed control |
| CA2848695A1 (en) | 2011-09-13 | 2013-03-21 | Monsanto Technology Llc | Methods and composition for weed control comprising inhibiting ppg oxidase |
| CN107739737A (zh) | 2011-09-13 | 2018-02-27 | 孟山都技术公司 | 用于杂草控制的方法和组合物 |
| US10760086B2 (en) | 2011-09-13 | 2020-09-01 | Monsanto Technology Llc | Methods and compositions for weed control |
| WO2013040057A1 (en) | 2011-09-13 | 2013-03-21 | Monsanto Technology Llc | Methods and compositions for weed control |
| CA2873828A1 (en) | 2012-05-24 | 2013-11-28 | A.B. Seeds Ltd. | Naked dsrna for silencing target molecules in plant seeds |
| EA032406B1 (ru) | 2013-01-01 | 2019-05-31 | Эй.Би. СИДЗ ЛТД. | СПОСОБЫ ВВЕДЕНИЯ дсРНК В СЕМЕНА РАСТЕНИЙ ДЛЯ МОДУЛЯЦИИ ЭКСПРЕССИИ ГЕНОВ |
| US10683505B2 (en) | 2013-01-01 | 2020-06-16 | Monsanto Technology Llc | Methods of introducing dsRNA to plant seeds for modulating gene expression |
| AR095232A1 (es) | 2013-03-13 | 2015-09-30 | Monsanto Technology Llc | Métodos y composiciones para el control de malezas |
| UY35385A (es) | 2013-03-13 | 2014-09-30 | Monsanto Technology Llc | ?métodos y composiciones para el control de malezas?. |
| US10568328B2 (en) | 2013-03-15 | 2020-02-25 | Monsanto Technology Llc | Methods and compositions for weed control |
| US9850496B2 (en) | 2013-07-19 | 2017-12-26 | Monsanto Technology Llc | Compositions and methods for controlling Leptinotarsa |
| BR112016000555B1 (pt) | 2013-07-19 | 2022-12-27 | Monsanto Technology Llc | Método para controlar uma infestação da espécie de leptinotarsa em uma planta, composição inseticida e construção de dna recombinante |
| AR098295A1 (es) | 2013-11-04 | 2016-05-26 | Monsanto Technology Llc | Composiciones y métodos para controlar infestaciones de plagas y parásitos de los artrópodos |
| UA119253C2 (uk) | 2013-12-10 | 2019-05-27 | Біолоджикс, Інк. | Спосіб боротьби із вірусом у кліща varroa та у бджіл |
| MX368629B (es) | 2014-01-15 | 2019-10-08 | Monsanto Technology Llc | Metodos y composiciones para el control de malezas utilizando polinucleotidos de 5-enolpiruvilshikimato-3-fosfato sintasa (epsps). |
| WO2015125858A1 (ja) * | 2014-02-24 | 2015-08-27 | 日本曹達株式会社 | ヘテロアリール化合物およびその用途 |
| BR112016022711A2 (pt) | 2014-04-01 | 2017-10-31 | Monsanto Technology Llc | composições e métodos para controle de pragas de inseto |
| AU2015280252A1 (en) | 2014-06-23 | 2017-01-12 | Monsanto Technology Llc | Compositions and methods for regulating gene expression via RNA interference |
| WO2015200539A1 (en) | 2014-06-25 | 2015-12-30 | Monsanto Technology Llc | Methods and compositions for delivering nucleic acids to plant cells and regulating gene expression |
| US10378012B2 (en) | 2014-07-29 | 2019-08-13 | Monsanto Technology Llc | Compositions and methods for controlling insect pests |
| EP3194393B1 (en) | 2014-09-19 | 2020-03-11 | ISAGRO S.p.A. | 1,3,4-thiadiazoles having a herbicidal activity, their agronomical compositions and relative use |
| PL3256589T3 (pl) | 2015-01-22 | 2022-02-21 | Monsanto Technology Llc | Kompozycje i sposoby kontrolowania leptinotarsa |
| US10883103B2 (en) | 2015-06-02 | 2021-01-05 | Monsanto Technology Llc | Compositions and methods for delivery of a polynucleotide into a plant |
| CN108024517A (zh) | 2015-06-03 | 2018-05-11 | 孟山都技术公司 | 用于将核酸引入到植物中的方法和组合物 |
| IT201800009385A1 (it) | 2018-10-11 | 2020-04-11 | Isagro Spa | Derivati caffeinici ad attività nematocida, loro composizioni agronomiche e relativo uso |
| IT201900001339A1 (it) | 2019-01-30 | 2020-07-30 | Isagro Spa | Derivati teofillinici ad attività nematocida, loro composizioni agronomiche e relativo uso |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4057634A (en) * | 1974-01-24 | 1977-11-08 | Hoechst Aktiengesellschaft | Antiprotozoal(1-alkyl-5-nitro-imidazolyl-2-alkyl)-pyridazines |
| DE2403340A1 (de) * | 1974-01-24 | 1975-07-31 | Hoechst Ag | (1-alkyl-5-nitro-imidazolyl-2-alkyl)- heteroaryl-verbindungen und verfahren zu ihrer herstellung |
| ATE16799T1 (de) * | 1980-01-10 | 1985-12-15 | Nyegaard & Co As | Pyrimidin-2-sulfide und ihre s-oxide zur verwendung in der medizin, die verbindungen enthaltende pharmazeutische zusammensetzungen, verfahren zu ihrer herstellung und die verbindungen an sich, sofern sie neu sind. |
| GB2135992B (en) * | 1983-01-11 | 1986-09-24 | Nyegaard & Co As | Substituted pyrimidines and processes for their preparation |
| GB8712396D0 (en) * | 1987-05-27 | 1987-07-01 | May & Baker Ltd | Composition of matter |
| JPH0559015A (ja) * | 1991-06-26 | 1993-03-09 | Otsuka Chem Co Ltd | ピリミジン誘導体及び該誘導体を有効成分とする除草剤 |
| WO1995013267A1 (en) * | 1993-11-12 | 1995-05-18 | The Upjohn Company | Pyrimidine-thioalkyl and alkylether compounds |
-
2001
- 2001-11-02 DE DE10154075A patent/DE10154075A1/de not_active Withdrawn
-
2002
- 2002-10-21 WO PCT/EP2002/011744 patent/WO2003037878A1/de active Application Filing
- 2002-10-21 JP JP2003540160A patent/JP2005512985A/ja active Pending
- 2002-10-21 EP EP02777320A patent/EP1444208A1/de not_active Withdrawn
- 2002-10-21 US US10/493,781 patent/US20050065166A1/en not_active Abandoned
- 2002-10-29 AR ARP020104107A patent/AR037130A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003037878A1 (de) | 2003-05-08 |
| DE10154075A1 (de) | 2003-05-15 |
| JP2005512985A (ja) | 2005-05-12 |
| US20050065166A1 (en) | 2005-03-24 |
| EP1444208A1 (de) | 2004-08-11 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR037130A1 (es) | Pirimidinas substituidas | |
| DK1864975T3 (da) | Nikotinamid-derivater anvendelige som P38-inhibitorer | |
| AR055613A1 (es) | Formas cristalinas delta y epsilon de mesilato de imatinib | |
| ECSP066643A (es) | PIRIDO [2,3-d] PIRIMIDINA-2,4-DIAMINAS COMO INHIBIDORES DE PDE 2 | |
| CY1106801T1 (el) | Νεες ετεροκυκλικες ενωσεις, η παρασκευη τους και η χρηση τους ως φαρμακα, ιδιαιτερα ως αντιβακτηριακα | |
| BR0311195A (pt) | Processo de preparação de rosuvastatina | |
| ECSP056072A (es) | Pirimidinonas sustituidas | |
| NO20081003L (no) | 2-Aminopyrimidinderivater som modulatorer av histamin-H4-reseptoraktivitet | |
| ATE516291T1 (de) | Thenopyrimidin-verbindungen mit fungizider aktivität | |
| CY1105553T1 (el) | Υποκαταστατα 2-πυριμιδινυλιο-6,7,8,9-τετραϋδροπυριμιδο[1,2-α]πυριμιδιν-4-ονιο και 7-πυριμιδινυλιο-2,3-διυδροιμιδαζο[1,2-α]πυριμιδιν-5(1η)ονιο για νευροεκφυλιστικες διαταραχες | |
| ATE517896T1 (de) | P38-kinase-inhibitoren | |
| ECSP088821A (es) | Derivados de tioxantina y su uso como inhibidores de la mpo | |
| DK1817300T3 (da) | Forstærkere af glutamat-receptorer | |
| BR0312695A (pt) | Derivados de 1h-pirrolidina-2,4-diona espirocìclicos substituìdos por cis-alcóxi | |
| ATE400570T1 (de) | 2,4,6-trisubstituierte pyrimidine als inhibitoren von phosphatidylinosit-(pi-)3-kinase und deren verwendung bei der behandlung von krebs | |
| ATE413392T1 (de) | Kondensierte heteroyralderivate und deren verwendung als p38-kinase-inhibitoren | |
| AR029838A1 (es) | Heterociclos benzonitrogenados sustituidos | |
| UY27338A1 (es) | Nuevos derivados de ácido sulfónico | |
| ECSP044999A (es) | Agentes antidiabeticos | |
| BRPI0412834A (pt) | derivados de nicotinamida usados como inibidores da pde4 | |
| BRPI0821114A2 (pt) | Composto, uso de um composto e método para tratar qualquer mamífero afetado por câncer | |
| EA200802248A1 (ru) | Способы применения соединений 4-амино-5-хлортиено[2,3-d]-пиримидина в качестве инсектицидов | |
| AR055564A1 (es) | Derivados de quinazolina | |
| AR026337A1 (es) | Benzoil-ciclohexanodionas y benzoil-pirazoles, procedimiento para su preparacion y su utilizacion como herbicidas y reguladores del crecimiento de lasplantas | |
| UY29707A1 (es) | Compuestos de 7-amino-6-heteroaril-1,2,4-triazolo(1,5-a)pirimidina y su empleo para combatir hongos daninos |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |