JP2005508953A5 - - Google Patents

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Publication number
JP2005508953A5
JP2005508953A5 JP2003534421A JP2003534421A JP2005508953A5 JP 2005508953 A5 JP2005508953 A5 JP 2005508953A5 JP 2003534421 A JP2003534421 A JP 2003534421A JP 2003534421 A JP2003534421 A JP 2003534421A JP 2005508953 A5 JP2005508953 A5 JP 2005508953A5
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JP
Japan
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hydrogen
compound
alkyl
compound according
ring
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JP2003534421A
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Japanese (ja)
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JP2005508953A (ja
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Priority claimed from PCT/US2002/032354 external-priority patent/WO2003031438A1/en
Publication of JP2005508953A publication Critical patent/JP2005508953A/ja
Publication of JP2005508953A5 publication Critical patent/JP2005508953A5/ja
Withdrawn legal-status Critical Current

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JP2003534421A 2001-10-10 2002-10-10 キナーゼ阻害剤としての３−［４−（置換ヘテロサイクリル）−ピロール−２−イルメチリデン］−２−インドリノン誘導体 Withdrawn JP2005508953A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32822601P 2001-10-10 2001-10-10
PCT/US2002/032354 WO2003031438A1 (en) 2001-10-10 2002-10-10 3-[4-(substituted heterocyclyl)-pyrrol-2-ylmethylidene]-2-indolinone derivatives as kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2005508953A JP2005508953A (ja) 2005-04-07
JP2005508953A5 true JP2005508953A5 (enExample) 2006-01-05

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003534421A Withdrawn JP2005508953A (ja) 2001-10-10 2002-10-10 キナーゼ阻害剤としての３−［４−（置換ヘテロサイクリル）−ピロール−２−イルメチリデン］−２−インドリノン誘導体

Country Status (7)

Country Link
US (1) US6642232B2 (enExample)
EP (1) EP1434774A1 (enExample)
JP (1) JP2005508953A (enExample)
BR (1) BR0213185A (enExample)
CA (1) CA2462950A1 (enExample)
MX (1) MXPA04003385A (enExample)
WO (1) WO2003031438A1 (enExample)

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WO2010011834A2 (en) 2008-07-24 2010-01-28 Teva Pharmaceutical Industries Ltd. Sunitinib and salts thereof and their polymorphs
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EP2694058B1 (en) 2011-04-08 2015-11-04 Beta Pharma, Inc. New indolinone protein kinase inhibitors
JP6039683B2 (ja) 2011-11-23 2016-12-07 ポートラ ファーマシューティカルズ， インコーポレイテッド ピラジンキナーゼ阻害剤
CN104829596B (zh) * 2014-02-10 2017-02-01 石家庄以岭药业股份有限公司 吡咯取代吲哚酮类衍生物、其制备方法、包含该衍生物的组合物、及其用途
KR102289684B1 (ko) * 2016-09-29 2021-08-12 이쿼녹스 사이언시스, 엘엘씨 키나아제 억제제 화합물의 다결정형(polymorphic form), 이를 함유한 약물 조성물 및 그의 제조방법과 응용

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