JP2005507932A - 肥満の処置のためのフェニル置換５−員窒素含有複素環 - Google Patents

肥満の処置のためのフェニル置換５−員窒素含有複素環 Download PDF

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JP2005507932A
JP2005507932A JP2003539676A JP2003539676A JP2005507932A JP 2005507932 A JP2005507932 A JP 2005507932A JP 2003539676 A JP2003539676 A JP 2003539676A JP 2003539676 A JP2003539676 A JP 2003539676A JP 2005507932 A JP2005507932 A JP 2005507932A
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コイシユ，フイリツプ・デイ・ジー
オコナー，ステイーブン・ジエイ
ウイケンス，フイリツプ
ツアング，チエンツイー
ツアング，ハイ−ジユン
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バイエル・フアーマシユーチカルズ・コーポレーシヨン
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    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/18—One oxygen or sulfur atom
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    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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JP2003539676A 2001-10-12 2002-10-15 肥満の処置のためのフェニル置換５−員窒素含有複素環 Withdrawn JP2005507932A (ja)

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Application Number Priority Date Filing Date Title
US32923601P 2001-10-12 2001-10-12
PCT/US2002/032895 WO2003037332A1 (en) 2001-10-12 2002-10-15 Phenyl substituted 5-membered nitrogen containing heterocycles for the treatment of obesity

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JP2005507932A true JP2005507932A (ja) 2005-03-24
JP2005507932A5 JP2005507932A5 (https=) 2006-01-05

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US (1) US20050014805A1 (https=)
EP (1) EP1435951B1 (https=)
JP (1) JP2005507932A (https=)
CA (1) CA2463441A1 (https=)
DE (1) DE60208815T2 (https=)
ES (1) ES2256560T3 (https=)
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Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007052843A1 (ja) * 2005-11-04 2007-05-10 Takeda Pharmaceutical Company Limited 複素環アミド化合物およびその用途
JP2016512209A (ja) * 2013-03-13 2016-04-25 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ベンゾオキサゼピン化合物の作製方法
JP2018500286A (ja) * 2014-10-30 2018-01-11 ヤンセン ファーマシューティカ エヌ．ベー． ＲＯＲγｔのモジュレーターとしてのアミド置換チアゾール
JP2019506415A (ja) * 2016-02-11 2019-03-07 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 有害生物防除剤としての置換２−（ヘタ）アリール−イミダゾリル−カルボキサミド類
US10975068B2 (en) 2016-04-27 2021-04-13 Janssen Pharmaceutica Nv 6-aminopyridin-3-yl thiazoles as modulators of RORγT
US10975037B2 (en) 2018-06-18 2021-04-13 Janssen Pharmaceutica Nv Phenyl substituted pyrazoles as modulators of RORγt
US10975057B2 (en) 2018-06-18 2021-04-13 Janssen Pharmaceutica Nv 6-aminopyridin-3-yl pyrazoles as modulators of RORgT
US11034658B2 (en) 2018-06-18 2021-06-15 Janssen Pharmaceutica Nv Pyridinyl pyrazoles as modulators of RORγT
US11345666B2 (en) 2018-06-18 2022-05-31 Janssen Pharmaceutica Nv Phenyl and pyridinyl substituted imidazoles as modulators of RORγT

Families Citing this family (48)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003007887A2 (en) 2001-07-20 2003-01-30 Merck & Co., Inc. Substituted imidazoles as cannabinoid receptor modulators
NZ534757A (en) 2002-03-12 2006-07-28 Merck & Co Inc Substituted amides
WO2004058727A1 (en) * 2002-12-20 2004-07-15 Bayer Pharmaceuticals Corporation Substituted 3,5-dihydro-4h-imidazol-4-ones for the treatment of obesity
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JP2006518738A (ja) * 2003-02-12 2006-08-17 トランス　テック　ファーマ，インコーポレイテッド 治療薬としての置換アゾール誘導体
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