JP2005506977A5 - - Google Patents
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- Publication number
- JP2005506977A5 JP2005506977A5 JP2003523216A JP2003523216A JP2005506977A5 JP 2005506977 A5 JP2005506977 A5 JP 2005506977A5 JP 2003523216 A JP2003523216 A JP 2003523216A JP 2003523216 A JP2003523216 A JP 2003523216A JP 2005506977 A5 JP2005506977 A5 JP 2005506977A5
- Authority
- JP
- Japan
- Prior art keywords
- amino acid
- acid halide
- halide according
- unsubstituted
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- -1 amino acid halide Chemical class 0.000 claims 16
- 229910052739 hydrogen Inorganic materials 0.000 claims 8
- 239000001257 hydrogen Substances 0.000 claims 8
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 5
- 125000000217 alkyl group Chemical group 0.000 claims 5
- 150000002431 hydrogen Chemical class 0.000 claims 3
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 claims 3
- 229910052757 nitrogen Inorganic materials 0.000 claims 3
- 125000006239 protecting group Chemical group 0.000 claims 3
- 125000006374 C2-C10 alkenyl group Chemical group 0.000 claims 2
- 125000005865 C2-C10alkynyl group Chemical group 0.000 claims 2
- YLQBMQCUIZJEEH-UHFFFAOYSA-N Furan Chemical compound C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 claims 2
- KAESVJOAVNADME-UHFFFAOYSA-N Pyrrole Chemical compound C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 claims 2
- YTPLMLYBLZKORZ-UHFFFAOYSA-N Thiophene Chemical compound C=1C=CSC=1 YTPLMLYBLZKORZ-UHFFFAOYSA-N 0.000 claims 2
- 125000001072 heteroaryl group Chemical group 0.000 claims 2
- NSPMIYGKQJPBQR-UHFFFAOYSA-N 4H-1,2,4-triazole Chemical compound C=1N=CNN=1 NSPMIYGKQJPBQR-UHFFFAOYSA-N 0.000 claims 1
- KXDHJXZQYSOELW-UHFFFAOYSA-N Carbamic acid Chemical group NC(O)=O KXDHJXZQYSOELW-UHFFFAOYSA-N 0.000 claims 1
- ZCQWOFVYLHDMMC-UHFFFAOYSA-N Oxazole Chemical compound C1=COC=N1 ZCQWOFVYLHDMMC-UHFFFAOYSA-N 0.000 claims 1
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical compound C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 claims 1
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000006242 amine protecting group Chemical group 0.000 claims 1
- 125000001475 halogen functional group Chemical group 0.000 claims 1
- 125000004356 hydroxy functional group Chemical group O* 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 229910052717 sulfur Inorganic materials 0.000 claims 1
- 229930192474 thiophene Natural products 0.000 claims 1
- 0 CN(*)C1C=C(*)N(*)*1 Chemical compound CN(*)C1C=C(*)N(*)*1 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US31615101P | 2001-08-30 | 2001-08-30 | |
| US10/061,617 US6677487B2 (en) | 2001-08-30 | 2002-02-01 | α-haloenamine reagents |
| PCT/US2002/027953 WO2003018552A2 (en) | 2001-08-30 | 2002-08-30 | Aromatic and heteroaromatic acid halides for synthesizing polyamides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005506977A JP2005506977A (ja) | 2005-03-10 |
| JP2005506977A5 true JP2005506977A5 (https=) | 2006-01-05 |
Family
ID=26741280
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003524956A Pending JP2005501898A (ja) | 2001-08-30 | 2002-08-13 | α−ハロエナミン試剤 |
| JP2003523216A Withdrawn JP2005506977A (ja) | 2001-08-30 | 2002-08-30 | ポリアミド合成用の芳香族及びヘテロ芳香族酸ハロゲン化物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003524956A Pending JP2005501898A (ja) | 2001-08-30 | 2002-08-13 | α−ハロエナミン試剤 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US6677487B2 (https=) |
| EP (2) | EP1421056A1 (https=) |
| JP (2) | JP2005501898A (https=) |
| KR (2) | KR20040029461A (https=) |
| CN (2) | CN1561326A (https=) |
| AU (2) | AU2002323122B2 (https=) |
| BR (2) | BR0212553A (https=) |
| CA (2) | CA2458859A1 (https=) |
| IL (2) | IL160609A0 (https=) |
| MX (2) | MXPA04001957A (https=) |
| PL (2) | PL368829A1 (https=) |
| RS (2) | RS26104A (https=) |
| RU (2) | RU2004109226A (https=) |
| WO (2) | WO2003020684A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6677487B2 (en) * | 2001-08-30 | 2004-01-13 | Pharmacia Corporation | α-haloenamine reagents |
| CN102399241A (zh) * | 2010-09-09 | 2012-04-04 | 信诺美（北京）化工科技有限公司 | 一种芳香基磷酸二酯的合成方法 |
| WO2015125721A1 (ja) * | 2014-02-18 | 2015-08-27 | 日産化学工業株式会社 | 電荷輸送性ワニス |
| US20190084928A1 (en) * | 2016-04-01 | 2019-03-21 | National University Corporation Chiba University | Method for producing nitrogen-containing aromatic amide, method for producing pyrrole-imidazole polyamide, and compound |
| CN113979962A (zh) | 2017-03-31 | 2022-01-28 | 先正达参股股份有限公司 | 杀真菌组合物 |
| CN113754553B (zh) * | 2021-10-18 | 2022-12-13 | 江苏快达农化股份有限公司 | 一种连续法合成水杨酰胺的方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2638356A1 (de) | 1976-08-26 | 1978-03-02 | Bayer Ag | Verfahren zur herstellung vinylsubstituierter cyclopropancarbonsaeureester |
| DE2715336A1 (de) | 1977-04-06 | 1978-10-19 | Bayer Ag | Verfahren zur herstellung viergliedriger cyclischer ketone |
| US4794109A (en) | 1982-11-16 | 1988-12-27 | Ciba-Geigy Corporation | 6-hydroxy-lower alkylpenem compounds, pharmaceutical preparations that contain these compounds, and the use of the latter |
| FI873183A7 (fi) | 1986-07-23 | 1988-01-24 | Ciba Geigy Ag | Kompleksit optisesti aktiivisten sokeriligandien kanssa, menetelmä niiden valmistamiseksi ja niiden käyttö. |
| US5218097A (en) | 1988-12-07 | 1993-06-08 | Ciba-Geigy Corporation | Process for the preparation of protected mono-sugar and oligo-sugar halides |
| CH681623A5 (en) * | 1990-11-05 | 1993-04-30 | Ciba Geigy Ag | Prodn. of alpha-halo:enamine halogenating agents - comprises two stage halogenation of di:substd. acetamide in presence of carboxamide or lactam catalyst and addn. of amine |
| US5459131A (en) | 1991-03-15 | 1995-10-17 | American Cyanamid Company | Renin inhibitors |
| US5643878A (en) | 1991-09-12 | 1997-07-01 | Ciba-Geigy Corporation | 5-amino-4-hydroxyhexanoic acid derivatives |
| US5273991A (en) | 1992-07-29 | 1993-12-28 | Research Corporation Technologies, Inc. | Imidazole-containing compositions and methods of use thereof analogs of distamycin |
| US5441876A (en) | 1993-07-30 | 1995-08-15 | The United States Of America As Represented By The Secretary Of The Navy | Process for the preparation of headgroup-modified phospholipids using phosphatidylhydroxyalkanols as intermediates |
| US5514643A (en) | 1993-08-16 | 1996-05-07 | Lucky Ltd. | 2-aminothiazolecarboxamide derivatives, processes for preparing the same and use thereof for controlling phytopathogenic organisms |
| WO1996033972A1 (en) * | 1995-04-28 | 1996-10-31 | Glaxo Group Limited | Methods for synthesizing diverse collections of pyridines, pyrimidines, 1,4-dihydro derivatives thereof, and piperidine derivatives |
| GB2310207A (en) | 1996-02-15 | 1997-08-20 | Pharmacia Spa | Antiviral ureido derivatives of substituted heterocyclic compounds |
| US6090947A (en) | 1996-02-26 | 2000-07-18 | California Institute Of Technology | Method for the synthesis of pyrrole and imidazole carboxamides on a solid support |
| MY129541A (en) | 1996-06-25 | 2007-04-30 | Novartis Ag | Substituded 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators |
| DE19805431A1 (de) | 1998-02-11 | 1999-08-12 | Merck Patent Gmbh | Heteroaromatische Oligoamide als Affinitätsliganden |
| EP1169038B9 (en) | 1999-04-15 | 2013-07-10 | Bristol-Myers Squibb Company | Cyclic protein tyrosine kinase inhibitors |
| US6677487B2 (en) * | 2001-08-30 | 2004-01-13 | Pharmacia Corporation | α-haloenamine reagents |
-
2002
- 2002-02-01 US US10/061,617 patent/US6677487B2/en not_active Expired - Fee Related
- 2002-08-13 IL IL16060902A patent/IL160609A0/xx unknown
- 2002-08-13 PL PL02368829A patent/PL368829A1/xx not_active Application Discontinuation
- 2002-08-13 RU RU2004109226/04A patent/RU2004109226A/ru not_active Application Discontinuation
- 2002-08-13 KR KR10-2004-7003127A patent/KR20040029461A/ko not_active Ceased
- 2002-08-13 JP JP2003524956A patent/JP2005501898A/ja active Pending
- 2002-08-13 CN CNA028190084A patent/CN1561326A/zh active Pending
- 2002-08-13 EP EP02757083A patent/EP1421056A1/en not_active Withdrawn
- 2002-08-13 RS YU26104A patent/RS26104A/sr unknown
- 2002-08-13 AU AU2002323122A patent/AU2002323122B2/en not_active Expired - Fee Related
- 2002-08-13 BR BR0212553-6A patent/BR0212553A/pt not_active IP Right Cessation
- 2002-08-13 MX MXPA04001957A patent/MXPA04001957A/es not_active Application Discontinuation
- 2002-08-13 CA CA002458859A patent/CA2458859A1/en not_active Abandoned
- 2002-08-13 WO PCT/US2002/025609 patent/WO2003020684A1/en not_active Ceased
- 2002-08-30 PL PL02368830A patent/PL368830A1/xx not_active Application Discontinuation
- 2002-08-30 IL IL16059602A patent/IL160596A0/xx unknown
- 2002-08-30 MX MXPA04001958A patent/MXPA04001958A/es unknown
- 2002-08-30 AU AU2002332809A patent/AU2002332809B2/en not_active Expired - Fee Related
- 2002-08-30 CA CA002458616A patent/CA2458616A1/en not_active Abandoned
- 2002-08-30 JP JP2003523216A patent/JP2005506977A/ja not_active Withdrawn
- 2002-08-30 RS YUP-260/04A patent/RS26004A/sr unknown
- 2002-08-30 CN CNA028192117A patent/CN1561333A/zh active Pending
- 2002-08-30 KR KR10-2004-7003109A patent/KR20040029460A/ko not_active Ceased
- 2002-08-30 EP EP02796456A patent/EP1430028A2/en not_active Withdrawn
- 2002-08-30 BR BR0212393-2A patent/BR0212393A/pt not_active IP Right Cessation
- 2002-08-30 WO PCT/US2002/027953 patent/WO2003018552A2/en not_active Ceased
- 2002-08-30 RU RU2004109225/04A patent/RU2004109225A/ru not_active Application Discontinuation
-
2003
- 2003-09-17 US US10/664,123 patent/US6924396B2/en not_active Expired - Fee Related
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