JP2005503327A5 - - Google Patents

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Publication number
JP2005503327A5
JP2005503327A5 JP2002564480A JP2002564480A JP2005503327A5 JP 2005503327 A5 JP2005503327 A5 JP 2005503327A5 JP 2002564480 A JP2002564480 A JP 2002564480A JP 2002564480 A JP2002564480 A JP 2002564480A JP 2005503327 A5 JP2005503327 A5 JP 2005503327A5
Authority
JP
Japan
Prior art keywords
methoxy
isophthalamide
benzyl
ylmethyl
benzodioxol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002564480A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005503327A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2002/000344 external-priority patent/WO2002064547A2/en
Publication of JP2005503327A publication Critical patent/JP2005503327A/ja
Publication of JP2005503327A5 publication Critical patent/JP2005503327A5/ja
Pending legal-status Critical Current

Links

JP2002564480A 2001-02-14 2002-02-04 マトリックスメタロプロテイナーゼ阻害剤としてのイソフタル酸誘導体 Pending JP2005503327A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26873601P 2001-02-14 2001-02-14
PCT/IB2002/000344 WO2002064547A2 (en) 2001-02-14 2002-02-04 Isophthalic acid derivatives as matrix metalloproteinase inhibitors

Publications (2)

Publication Number Publication Date
JP2005503327A JP2005503327A (ja) 2005-02-03
JP2005503327A5 true JP2005503327A5 (enExample) 2008-05-29

Family

ID=23024241

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002564480A Pending JP2005503327A (ja) 2001-02-14 2002-02-04 マトリックスメタロプロテイナーゼ阻害剤としてのイソフタル酸誘導体

Country Status (13)

Country Link
US (2) US6995151B2 (enExample)
EP (1) EP1362028A2 (enExample)
JP (1) JP2005503327A (enExample)
AR (1) AR032679A1 (enExample)
BR (1) BR0207201A (enExample)
CA (1) CA2435376A1 (enExample)
DO (1) DOP2002000333A (enExample)
MX (1) MXPA03006598A (enExample)
PA (1) PA8539801A1 (enExample)
PE (1) PE20020859A1 (enExample)
TN (1) TNSN02008A1 (enExample)
UY (1) UY27169A1 (enExample)
WO (1) WO2002064547A2 (enExample)

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DOP2002000333A (es) * 2001-02-14 2002-09-30 Warner Lambert Co Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
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US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
MXPA04002537A (es) 2001-10-12 2004-05-31 Warner Lambert Co Alquinos como inhibidores de metaloproteinasa de matriz.
US6962922B2 (en) 2001-10-12 2005-11-08 Warner-Lambert Company Llc Alkynylated quinazoline compounds
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US6747147B2 (en) 2002-03-08 2004-06-08 Warner-Lambert Company Oxo-azabicyclic compounds
US6894057B2 (en) 2002-03-08 2005-05-17 Warner-Lambert Company Oxo-azabicyclic compounds
US20040006077A1 (en) * 2002-06-25 2004-01-08 Bernard Gaudilliere Thiazine and oxazine derivatives as MMP-13 inhibitors
EP1531904A1 (en) * 2002-07-17 2005-05-25 Warner-Lambert Company LLC Combination of an allosteric inhibitor of matrix metalloproteinase-13 with a selective inhibitor of cyclooxygenase-2 that is not celecoxib or valdecoxib
MXPA05000754A (es) * 2002-07-17 2005-04-19 Warner Lambert Co Combinacion de un inhibidor carboxilico alosterico de la metaloproteinasa de matriz-13 con celecoxib o valdecoxib.
BR0312708A (pt) * 2002-07-17 2005-04-26 Warner Lambert Co Combinação de um inibidor alcina alostérico de metaloproteinase-13 de matriz com celecoxib ou valdecoxib
BR0312727A (pt) * 2002-07-17 2005-04-19 Warner Lambert Co Combinação de um inibidor alostérico da metaloproteinase-13 de matriz com celecoxib ou valdecoxib
CA2497658A1 (en) 2002-08-13 2004-02-19 Warner-Lambert Company Llc Chromone derivatives as matrix metalloproteinase inhibitors
MXPA05001603A (es) 2002-08-13 2005-04-25 Warner Lambert Co Derivados monociclicos como inhibidores de metaloproteinasa de matriz.
AU2003249477A1 (en) * 2002-08-13 2004-02-25 Warner-Lambert Company Llc Heterobicylcic metalloproteinase inhibitors
WO2004014375A2 (en) 2002-08-13 2004-02-19 Warner-Lambert Company Llc Fused bicyclic metalloproteinase inhibitors
WO2004014869A2 (en) * 2002-08-13 2004-02-19 Warner-Lambert Company Llc 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
AU2003249535A1 (en) * 2002-08-13 2004-02-25 Warner-Lambert Company Llc 1,6-fused uracil derivatives as matrix metalloproteinase inhibitors
AU2003253186A1 (en) 2002-08-13 2004-02-25 Warner-Lambert Company Llc Fused tetrahydropyridine derivatives as matrix metalloproteinase inhibitors
MXPA05001786A (es) 2002-08-13 2005-04-25 Warner Lambert Co Derivados de azaisoquinolina como inhibidores de la metaloproteinasa de matriz.
MXPA05001784A (es) * 2002-08-13 2005-04-25 Warner Lambert Co Derivados de isoquinolina como inhibidores de metaloproteinasa de matriz.
WO2004014384A2 (en) * 2002-08-13 2004-02-19 Warner-Lambert Company Llc Cyclic compounds containing zinc binding groups as matrix metalloproteinase inhibitors
MXPA05001783A (es) 2002-08-13 2005-04-25 Warner Lambert Co Derivados de pirimidina-2,4-diona como inhibidores de las metaloproteinasas de matriz.
WO2004014378A1 (en) 2002-08-13 2004-02-19 Warner-Lambert Company Llc 3-isoquinolinone derivatives as matrix metalloproteinase inhiitors
WO2004014365A1 (en) * 2002-08-13 2004-02-19 Warner-Lambert Company Llc Phthalimide derivatives as matrix metalloproteinase inhibitors
PA8578101A1 (es) 2002-08-13 2004-05-07 Warner Lambert Co Derivados de heterobiarilo como inhibidores de metaloproteinasa de la matriz
AU2003250470A1 (en) 2002-08-13 2004-02-25 Warner-Lambert Company Llc Pyrimidinone fused bicyclic metalloproteinase inhibitors
EP1394159A1 (fr) * 2002-08-13 2004-03-03 Warner-Lambert Company LLC Nouveaux dérivés de thiophène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
AU2003253165A1 (en) * 2002-08-13 2004-02-25 Warner-Lambert Company Llc Pyrimidine fused bicyclic metalloproteinase inhibitors
US20040142950A1 (en) * 2003-01-17 2004-07-22 Bunker Amy Mae Amide and ester matrix metalloproteinase inhibitors
WO2005046683A1 (en) 2003-10-07 2005-05-26 Renovis, Inc. Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
US20060247231A1 (en) * 2003-12-18 2006-11-02 Warner-Lambert Company Llc Amide and ester matrix metalloproteinase inhibitors
TW200529812A (en) 2003-12-26 2005-09-16 Chugai Pharmaceutical Co Ltd Benzamide derivatives
EP1820795A4 (en) 2004-12-07 2010-10-20 Toyama Chemical Co Ltd NEW ANTHRANILIC ACID DERIVATIVE OR SALT FROM IT
US7576099B2 (en) 2005-02-28 2009-08-18 Renovis, Inc. Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
FI20085415A0 (fi) * 2008-05-06 2008-05-06 Raimo Tuominen Proteiinikinaaseja muuntavia aineita
JP5657201B2 (ja) * 2008-09-30 2015-01-21 サンメディカル株式会社 酵素阻害作用または酵素阻害作用と抗菌作用とを有する歯科用組成物
CN102224151A (zh) 2008-11-20 2011-10-19 万能药生物有限公司 新的抗微生物剂
RU2012102094A (ru) 2009-06-26 2013-08-10 Панацеа Биотек Лтд. Новые азабициклогексаны
CN103012189A (zh) * 2012-12-20 2013-04-03 天津理工大学 具有抗血小板聚集作用的酰胺类化合物及其制备和应用
CN105693518B (zh) * 2014-11-28 2018-12-14 天津耀宇生物技术有限公司 从三棱中提取邻苯二甲酸二丁酯的方法及其应用
CN105884620A (zh) * 2016-04-22 2016-08-24 东南大学 4-羟基-1，3苯二甲酸二酯类衍生物及其制备和应用
CN116769179B (zh) * 2023-06-21 2024-02-06 中国科学院沈阳应用生态研究所 一种含间苯二甲酸的配位聚合物及其制备方法

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DOP2002000332A (es) 2001-02-14 2002-08-30 Warner Lambert Co Inhibidores de piridina de metaloproteinasas de la matriz
DOP2002000333A (es) * 2001-02-14 2002-09-30 Warner Lambert Co Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
JP2004518723A (ja) 2001-02-14 2004-06-24 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー ピリミジンマトリックスメタロプロテイナーゼ阻害剤
DE10160357A1 (de) 2001-12-08 2003-06-18 Aventis Pharma Gmbh Verwendung von Pyridin-2,4-dicarbonsäurediamiden und Pyrimidin-4,6-dicarbonsäurediamiden zur selektiven Inhibierung von Kollagenasen
US6933298B2 (en) * 2001-12-08 2005-08-23 Aventis Pharma Deutschland Gmbh Pyridine-2,4-dicarboxylic acid diamides and pyrimidine-4,6-dicarboxylic acid diamides and the use thereof for selectively inhibiting collagenases

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