JP2004531570A5 - - Google Patents

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Publication number
JP2004531570A5
JP2004531570A5 JP2002592931A JP2002592931A JP2004531570A5 JP 2004531570 A5 JP2004531570 A5 JP 2004531570A5 JP 2002592931 A JP2002592931 A JP 2002592931A JP 2002592931 A JP2002592931 A JP 2002592931A JP 2004531570 A5 JP2004531570 A5 JP 2004531570A5
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JP
Japan
Prior art keywords
alkyl
amino
alkoxy
hydroxy
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002592931A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004531570A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/016529 external-priority patent/WO2002096421A1/en
Publication of JP2004531570A publication Critical patent/JP2004531570A/ja
Publication of JP2004531570A5 publication Critical patent/JP2004531570A5/ja
Pending legal-status Critical Current

Links

JP2002592931A 2001-05-22 2002-05-22 Crf1モジュレーターとしての5−置換−2−アリールピリジン Pending JP2004531570A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29270301P 2001-05-22 2001-05-22
PCT/US2002/016529 WO2002096421A1 (en) 2001-05-22 2002-05-22 5-substituted-2-arylpyridines as crf1 modulators

Publications (2)

Publication Number Publication Date
JP2004531570A JP2004531570A (ja) 2004-10-14
JP2004531570A5 true JP2004531570A5 (https=) 2006-01-05

Family

ID=23125823

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002592931A Pending JP2004531570A (ja) 2001-05-22 2002-05-22 Crf1モジュレーターとしての5−置換−2−アリールピリジン

Country Status (20)

Country Link
US (2) US7223778B2 (https=)
EP (1) EP1392302A1 (https=)
JP (1) JP2004531570A (https=)
KR (1) KR20040015716A (https=)
AP (1) AP2003002920A0 (https=)
BG (1) BG108490A (https=)
BR (1) BR0209920A (https=)
CA (1) CA2448198A1 (https=)
EC (1) ECSP034860A (https=)
HR (1) HRP20031056A2 (https=)
HU (1) HUP0400316A2 (https=)
IL (1) IL158958A0 (https=)
IS (1) IS7046A (https=)
MX (1) MXPA03010692A (https=)
NO (1) NO20035183D0 (https=)
PL (1) PL367153A1 (https=)
RU (1) RU2003134010A (https=)
SK (1) SK15432003A3 (https=)
TN (1) TNSN03119A1 (https=)
WO (1) WO2002096421A1 (https=)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003249369A1 (en) 2002-06-21 2004-01-06 Cellular Genomics, Inc. Certain amino-substituted monocycles as kinase modulators
AU2003291403A1 (en) * 2002-11-08 2004-06-03 Neurogen Corporation 3-substituted-6-aryl pyridined as ligands of c5a receptors
WO2005007627A1 (ja) * 2003-07-18 2005-01-27 Nihon Nohyaku Co., Ltd. フェニルピリジン誘導体、その中間体及びこれを有効成分とする除草剤
US20070099938A1 (en) * 2003-10-24 2007-05-03 Ono Pharmaceutical Co., Ltd. Antistress drug and medical use thereof
RU2423979C2 (ru) * 2005-06-17 2011-07-20 АФТ Фармасьютикалз Лимитед Новая фармацевтическая композиция и ее применение в способе лечения пациентов с гиперемией и отеком слизистой оболочки верхних дыхательных путей
EP1945632B1 (en) 2005-11-08 2013-09-18 Vertex Pharmaceuticals Incorporated Heterocyclic modulators of atp-binding cassette transporters
US8969386B2 (en) 2007-05-09 2015-03-03 Vertex Pharmaceuticals Incorporated Modulators of CFTR
US8048898B2 (en) * 2007-08-01 2011-11-01 Taisho Pharmaceutical Co., Ltd Inhibitor of binding of S1P1
SI2225230T1 (sl) 2007-12-07 2017-03-31 Vertex Pharmaceuticals Incorporated Trdne oblike 3-(6-(1-2,2-difluorobenzo(d)(1,3)dioxol-5-il)ciklopropan- karboksamido)-3-metilpiridin-2-il) benzojske kisline
EP2639224B1 (en) * 2007-12-07 2016-08-24 Vertex Pharmaceuticals Incorporated Process for producing cycloalkylcarboxiamido-pyridine benzoic acids
AU2013205160B2 (en) * 2007-12-07 2016-05-19 Vertex Pharmaceuticals Incorporated Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
NZ720282A (en) 2008-02-28 2017-12-22 Vertex Pharma Heteroaryl derivatives as cftr modulators
HRP20211752T1 (hr) 2010-04-07 2022-02-18 Vertex Pharmaceuticals Incorporated Farmaceutski pripravci 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioksol-5-il)ciklopropankarboksamido)-3-metilpiridin-2-il)benzojeve kiseline i njihova primjena
WO2013112804A1 (en) 2012-01-25 2013-08-01 Vertex Pharmaceuticals Incorporated Formulations of 3-(6-(1-(2.2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid
JP6219922B2 (ja) * 2012-03-30 2017-10-25 ダウ アグロサイエンシィズ エルエルシー 3−置換−6−トリフルオロメチルピリジンを調製する方法およびハロゲン化6−トリクロロメチルピリジンを使用する方法
JP6963896B2 (ja) 2013-11-12 2021-11-10 バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated Cftr媒介性疾患の処置のための医薬組成物を調製する方法
PT3221692T (pt) 2014-11-18 2021-09-10 Vertex Pharma Processo de realização de testagem de alta produtividade por cromatografia líquida de alta eficiência
KR101750453B1 (ko) 2015-09-11 2017-06-23 동아대학교 산학협력단 손잡이 세정이 가능한 샤워헤드용 방향제어밸브
US10399944B2 (en) 2017-08-10 2019-09-03 Janssen Pharmaceutica Nv Pyridin-2-one derivatives of formula (III) useful as EP3 receptor antagonists
US10336701B2 (en) 2017-08-10 2019-07-02 Janssen Pharmaceutica Nv Pyridin-2-one derivatives of formula (II) useful as EP3 receptor antagonists
US10590083B2 (en) 2017-08-10 2020-03-17 Janssen Pharmaceutica Nv Pyridin-2-one derivatives of formula (I) useful as EP3 receptor antagonists

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1147068A (en) 1966-12-02 1969-04-02 Ici Ltd Phenyl-pyridine derivatives
GB9012017D0 (en) * 1990-05-30 1990-07-18 Ici Plc Fungicidal compounds
DE4315867A1 (de) * 1993-05-12 1994-11-17 Hoechst Ag 3-Chlorpyridine, Verfahren zu ihrer Herstellung und ihre Verwendung in Flüssigkristallmischungen
DE4323916A1 (de) 1993-07-16 1995-01-19 Basf Ag Substituierte 2-Phenylpyridine
TW530047B (en) 1994-06-08 2003-05-01 Pfizer Corticotropin releasing factor antagonists
US5849758A (en) * 1995-05-30 1998-12-15 American Cyanamid Company Herbicidal 2, 6-disubstituted pyridines and 2, 4-disubstituted pyrimidines
DE19748439A1 (de) * 1997-11-03 1999-05-06 Hoechst Ag 1,6-Disubstituierte Naphthalinderivate und ihre Verwendung in flüssigkristallinen Mischungen
PL365238A1 (en) 2000-02-16 2004-12-27 Neurogen Corporation Substituted arylpyrazines
EP1233949A2 (en) 2000-03-16 2002-08-28 Neurogen Corporation 5-substituted arylpyrimidines

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