JP2004524315A5 - - Google Patents

Download PDF

Info

Publication number
JP2004524315A5
JP2004524315A5 JP2002567926A JP2002567926A JP2004524315A5 JP 2004524315 A5 JP2004524315 A5 JP 2004524315A5 JP 2002567926 A JP2002567926 A JP 2002567926A JP 2002567926 A JP2002567926 A JP 2002567926A JP 2004524315 A5 JP2004524315 A5 JP 2004524315A5
Authority
JP
Japan
Prior art keywords
alkyl
group
halogenoalkyl
optionally
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002567926A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004524315A (ja
Filing date
Publication date
Priority claimed from DE10108480A external-priority patent/DE10108480A1/de
Application filed filed Critical
Publication of JP2004524315A publication Critical patent/JP2004524315A/ja
Publication of JP2004524315A5 publication Critical patent/JP2004524315A5/ja
Pending legal-status Critical Current

Links

JP2002567926A 2001-02-22 2002-02-11 ピラゾリルピリミジン Pending JP2004524315A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10108480A DE10108480A1 (de) 2001-02-22 2001-02-22 Pyrazolylpyrimidine
PCT/EP2002/001400 WO2002068413A1 (de) 2001-02-22 2002-02-11 Pyrazolylpyrimidine

Publications (2)

Publication Number Publication Date
JP2004524315A JP2004524315A (ja) 2004-08-12
JP2004524315A5 true JP2004524315A5 (enExample) 2005-12-22

Family

ID=7675081

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002567926A Pending JP2004524315A (ja) 2001-02-22 2002-02-11 ピラゾリルピリミジン

Country Status (13)

Country Link
US (1) US7087616B2 (enExample)
EP (1) EP1363905A1 (enExample)
JP (1) JP2004524315A (enExample)
KR (1) KR100854583B1 (enExample)
CN (1) CN1301992C (enExample)
BR (1) BR0207509A (enExample)
DE (1) DE10108480A1 (enExample)
HU (1) HUP0303241A2 (enExample)
IL (1) IL157298A0 (enExample)
MX (1) MXPA03007433A (enExample)
TW (1) TWI236475B (enExample)
WO (1) WO2002068413A1 (enExample)
ZA (1) ZA200306468B (enExample)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI372050B (en) * 2003-07-03 2012-09-11 Astex Therapeutics Ltd (morpholin-4-ylmethyl-1h-benzimidazol-2-yl)-1h-pyrazoles
MX2007008008A (es) 2004-12-30 2007-11-12 Astex Therapeutics Ltd Compuestos de pirazol que modulan la actividad de las cinasas cdk, gsk y aurora.
DE102005058418A1 (de) * 2005-12-07 2007-06-21 Bayer Cropscience Gmbh Verfahren zur Herstellung von Haloalkyl(thio)vinimidiniumsalzen und 4-(Haloalkyl(thio))-pyrazolen und deren Umsetzung zu Pflanzenschutzmitteln
JP5474354B2 (ja) * 2005-12-30 2014-04-16 アステックス、セラピューティックス、リミテッド 医薬化合物
US8435970B2 (en) * 2006-06-29 2013-05-07 Astex Therapeutics Limited Pharmaceutical combinations of 1-cyclopropyl-3-[3-(5-morpholin-4-ylmethyl-1H-benzoimidazol-2-yl)-1H-pyrazol-4-yl]-urea
JP2009542608A (ja) * 2006-06-29 2009-12-03 アステックス・セラピューティクス・リミテッド 医薬組合せ剤
DE102007003036A1 (de) * 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
DE102007044032A1 (de) 2007-09-14 2009-03-19 Bayer Healthcare Ag Substituierte heterocyclische Verbindungen und ihre Verwendung
DE102007048447A1 (de) 2007-10-10 2009-04-16 Bayer Healthcare Ag Substituierte Dihydropyrazolthione und ihre Verwendung
EP2135865A1 (de) * 2008-06-17 2009-12-23 Bayer CropScience AG Substituierte 1-(Diazinyl) pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
US20110190365A1 (en) * 2008-08-14 2011-08-04 Bayer Crop Science Ag Insecticidal 4-phenyl-1H-pyrazoles
DE112010001898T5 (de) * 2009-04-27 2012-08-02 Dow Agrosciences Llc Insektizide Pyridinverbindungen
CN102573478B (zh) * 2009-10-12 2015-12-16 拜尔农作物科学股份公司 作为杀虫剂的1-(吡啶-3-基)-吡唑和1-(嘧啶-5-基)-吡唑
AR078947A1 (es) 2009-11-11 2011-12-14 Bayer Cropscience Ag Compuestos de diazinil-pirazolilo y procesos de preparacion de los mismos
JP2012116796A (ja) * 2010-12-01 2012-06-21 Sumitomo Chemical Co Ltd ヘテロ芳香環化合物およびその有害生物防除用途
CN104302640A (zh) 2012-03-16 2015-01-21 埃克希金医药品有限公司 3,5-二氨基吡唑激酶抑制剂
NZ631142A (en) 2013-09-18 2016-03-31 Axikin Pharmaceuticals Inc Pharmaceutically acceptable salts of 3,5-diaminopyrazole kinase inhibitors
MY195016A (en) 2014-08-04 2023-01-03 Nuevolution As Optionally Fused Heterocyclyl-Substituted Derivatives of Pyrimidine Useful for The Treatment of Inflammatory, Metabolic, Oncologic and Autoimmune Diseases
WO2016057931A1 (en) 2014-10-10 2016-04-14 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration
MY191736A (en) 2014-12-23 2022-07-13 Axikin Pharmaceuticals Inc 3,5-diaminopyrazole kinase inhibitors
AU2020405446A1 (en) 2019-12-20 2022-05-26 Nuevolution A/S Compounds active towards nuclear receptors
BR112022012205A2 (pt) 2019-12-20 2022-09-13 Nuevolution As Compostos ativos para receptores nucleares
JP7713954B2 (ja) 2020-03-31 2025-07-28 ヌエヴォリューション・アクティーゼルスカブ 核内受容体に対して活性な化合物
CA3174252A1 (en) 2020-03-31 2021-10-07 Nuevolution A/S Compounds active towards nuclear receptors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910910A (en) * 1972-03-31 1975-10-07 American Home Prod (2-Pyrimidinylthio) alkanoic acids, esters, amides and hydrazides
US4663327A (en) * 1984-05-23 1987-05-05 Bayer Aktiengesellschaft 1-heteroaryl-4-aryl-pyrazolin-5-ones
EP0702670A1 (de) 1993-06-07 1996-03-27 Bayer Ag Iodpropargylcarbamate und ihre verwendung als biozide im pflanzen- und materialschutz
CN1153779A (zh) * 1995-09-28 1997-07-09 山道士有限公司 2-(4-吡唑基氧基-嘧啶-5-基)乙酸衍生物
AU5412998A (en) * 1996-12-16 1998-07-15 Sumitomo Chemical Company, Limited Pyrazoline compounds and use as plant disease control agent

Similar Documents

Publication Publication Date Title
AU681075B2 (en) Antiproliferative quinazolines
AU2009313134B8 (en) Novel halogen-substituted compounds
ZA200306468B (en) Pyrazolyl pyrimidines.
EP1383187A3 (en) Nonaqueous electrolytic solution and nonaqueous secondary battery using the same
EP2100876A3 (en) Phenol derivatives and their use as Rotamase inhibitors
MY136662A (en) Cyano anthranilamide insecticides
PL1736510T3 (pl) Mieszanka żywiczna na bazie polikwasu mlekowego
EP1693705A3 (en) Resist composition, compound for use in the resist composition and pattern forming method using the resist composition
JP2004524310A5 (enExample)
RU2006138241A (ru) Способ получения 5-гидрокси-4-тиометилпиразольного соединения
AU2017388496A1 (en) Pyrimidine derivative
EP0122580B1 (de) Pyrimidinderivate, deren Herstellung und pharmazeutische Präparate
GB0417910D0 (en) Organic compounds
JP2006526587A5 (enExample)
BRPI0407194A (pt) processo para controlar a inversão de um fluido de perfuração e processo para controlar a umectabilidade de uma crosta de lodo
BRPI0416778A (pt) banho ácido para depositar eletroliticamente um depósito de cobre contendo compostos de fenazìnio monoméricos halogenados ou pseuso-halogenados
CA2418090A1 (en) Hydraulic fracturing fluid containing viscoelastic branched chain surfactant
EP2088142A3 (en) Dihydropyrimidines, process for their preparation and use thereof.
WO1997005116A1 (de) Substituierte aminouracile
Prukała New compounds via Mannich reaction of cytosine, paraformaldehyde and cyclic secondary amines
EP0804424A1 (de) Substituierte pyrimidin(thi)one
EP1921075A3 (en) A process for the preparation of pyridine-methylsulfinyl compounds
RU2003114858A (ru) Замещенные фенилурацилы
WO2016208773A1 (ja) オリゴヌクレオチド誘導体
EP1296957A2 (en) Synthesis of chlorinated pyrimidines