JP2006526587A5 - - Google Patents
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- Publication number
- JP2006526587A5 JP2006526587A5 JP2006508237A JP2006508237A JP2006526587A5 JP 2006526587 A5 JP2006526587 A5 JP 2006526587A5 JP 2006508237 A JP2006508237 A JP 2006508237A JP 2006508237 A JP2006508237 A JP 2006508237A JP 2006526587 A5 JP2006526587 A5 JP 2006526587A5
- Authority
- JP
- Japan
- Prior art keywords
- carbon atoms
- represented
- alkyl
- formula
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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- KLSJWNVTNUYHDU-UHFFFAOYSA-N Amitrole Chemical compound NC1=NC=NN1 KLSJWNVTNUYHDU-UHFFFAOYSA-N 0.000 claims description 2
- 125000004432 carbon atom Chemical group C* 0.000 claims 23
- 229910052736 halogen Inorganic materials 0.000 claims 13
- 150000002367 halogens Chemical group 0.000 claims 13
- 125000000217 alkyl group Chemical group 0.000 claims 12
- 238000000034 method Methods 0.000 claims 8
- -1 cyano, hydroxy Chemical group 0.000 claims 7
- 125000000623 heterocyclic group Chemical group 0.000 claims 7
- 125000000753 cycloalkyl group Chemical group 0.000 claims 6
- 125000001424 substituent group Chemical group 0.000 claims 6
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 claims 5
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims 5
- 125000003545 alkoxy group Chemical group 0.000 claims 5
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 claims 5
- 229910052794 bromium Inorganic materials 0.000 claims 5
- 229910052801 chlorine Inorganic materials 0.000 claims 5
- 239000000460 chlorine Substances 0.000 claims 5
- 239000003085 diluting agent Substances 0.000 claims 5
- 229910052731 fluorine Inorganic materials 0.000 claims 5
- 239000011737 fluorine Substances 0.000 claims 5
- 125000001188 haloalkyl group Chemical group 0.000 claims 5
- 125000004076 pyridyl group Chemical group 0.000 claims 5
- 125000000714 pyrimidinyl group Chemical group 0.000 claims 5
- YWBFPKPWMSWWEA-UHFFFAOYSA-O triazolopyrimidine Chemical compound BrC1=CC=CC(C=2N=C3N=CN[N+]3=C(NCC=3C=CN=CC=3)C=2)=C1 YWBFPKPWMSWWEA-UHFFFAOYSA-O 0.000 claims 5
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims 4
- 239000002253 acid Substances 0.000 claims 4
- 229910052757 nitrogen Inorganic materials 0.000 claims 4
- KVGVQTOQSNJTJI-UHFFFAOYSA-N 8-azaxanthine Chemical compound O=C1NC(=O)NC2=C1NN=N2 KVGVQTOQSNJTJI-UHFFFAOYSA-N 0.000 claims 3
- 125000004093 cyano group Chemical group *C#N 0.000 claims 3
- 229910052739 hydrogen Inorganic materials 0.000 claims 3
- 239000001257 hydrogen Substances 0.000 claims 3
- 244000005700 microbiome Species 0.000 claims 3
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 3
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- IYXGSMUGOJNHAZ-UHFFFAOYSA-N Ethyl malonate Chemical compound CCOC(=O)CC(=O)OCC IYXGSMUGOJNHAZ-UHFFFAOYSA-N 0.000 claims 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 2
- 125000003342 alkenyl group Chemical group 0.000 claims 2
- 125000004666 alkoxyiminoalkyl group Chemical group 0.000 claims 2
- 125000000304 alkynyl group Chemical group 0.000 claims 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 2
- 150000001879 copper Chemical class 0.000 claims 2
- 125000001153 fluoro group Chemical group F* 0.000 claims 2
- 125000004438 haloalkoxy group Chemical group 0.000 claims 2
- 229910052760 oxygen Inorganic materials 0.000 claims 2
- 239000001301 oxygen Substances 0.000 claims 2
- 229920006395 saturated elastomer Polymers 0.000 claims 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 1
- 150000001412 amines Chemical class 0.000 claims 1
- 239000011230 binding agent Substances 0.000 claims 1
- 239000003054 catalyst Substances 0.000 claims 1
- 239000003795 chemical substances by application Substances 0.000 claims 1
- 125000001309 chloro group Chemical group Cl* 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 230000002140 halogenating effect Effects 0.000 claims 1
- 125000005842 heteroatom Chemical group 0.000 claims 1
- 150000002431 hydrogen Chemical class 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 125000005017 substituted alkenyl group Chemical group 0.000 claims 1
- 125000000547 substituted alkyl group Chemical group 0.000 claims 1
- 125000004426 substituted alkynyl group Chemical group 0.000 claims 1
- 125000005346 substituted cycloalkyl group Chemical group 0.000 claims 1
- 229910052717 sulfur Inorganic materials 0.000 claims 1
- 239000011593 sulfur Substances 0.000 claims 1
- 125000004434 sulfur atom Chemical group 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10325133A DE10325133A1 (de) | 2003-06-04 | 2003-06-04 | Triazolopyrimidine |
| PCT/EP2004/005876 WO2004108727A1 (de) | 2003-06-04 | 2004-06-01 | Triazolopyrimidine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006526587A JP2006526587A (ja) | 2006-11-24 |
| JP2006526587A5 true JP2006526587A5 (enExample) | 2007-08-02 |
Family
ID=33482458
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006508237A Pending JP2006526587A (ja) | 2003-06-04 | 2004-06-01 | トリアゾロピリミジン類 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20070275985A1 (enExample) |
| EP (1) | EP1641798A1 (enExample) |
| JP (1) | JP2006526587A (enExample) |
| KR (1) | KR20060015304A (enExample) |
| CN (1) | CN1802379A (enExample) |
| BR (1) | BRPI0410906A (enExample) |
| CO (1) | CO5721005A2 (enExample) |
| CR (1) | CR8074A (enExample) |
| DE (1) | DE10325133A1 (enExample) |
| EC (1) | ECSP056201A (enExample) |
| IL (1) | IL172098A0 (enExample) |
| MX (1) | MXPA05012951A (enExample) |
| WO (1) | WO2004108727A1 (enExample) |
| ZA (1) | ZA200509637B (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR052341A1 (es) * | 2004-12-17 | 2007-03-14 | Basf Ag | Compuestos de 7-amino-6-hetaril-1, 2, 4-triazolo[1, 5 - a]pirimidina, intermediarios para su preparacion, y su empleo en agentes fungicidas para combatir hongos fitopatogenos |
| US20080132412A1 (en) * | 2004-12-17 | 2008-06-05 | Basf Aktiengesellschaft | 7-Amino-6-Heteroaryl-1,2,4-Triazolo[1,5-A]Pyrimidines and Their Use for Controlling Harmful Fungi |
| TW200643022A (en) * | 2005-03-02 | 2006-12-16 | Basf Ag | 2-substituted 7-aminoazolopyrimidines, processes for their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
| WO2006122740A2 (de) * | 2005-05-17 | 2006-11-23 | Basf Aktiengesellschaft | 7-AMINO-6-HETARYLIMIDAZOLO[1,2-a]PYRIMIDIN-VERBINDUNGEN UND IHRE VERWENDUNG ZU BEKÄMPFUNG VON SCHADPILZEN |
| WO2007006723A1 (de) * | 2005-07-13 | 2007-01-18 | Basf Aktiengesellschaft | 7-amino-6-tetrazolyl-1,2,4-triazolo[1,5-a]pyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen |
| WO2007101870A1 (de) * | 2006-03-08 | 2007-09-13 | Basf Se | Substituierte triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| CN101153041B (zh) * | 2006-09-28 | 2010-05-12 | 中国科学院化学研究所 | 1,2,3-三唑并1,3-二氮杂环化合物及其制备方法与应用 |
| EP2131658A2 (en) * | 2007-01-30 | 2009-12-16 | Basf Se | Method for improving plant health |
| EP1952691A3 (en) * | 2007-01-31 | 2008-09-17 | Basf Se | Method for improving plant health by application of a triazolopyrimidine derivative |
| US9101131B2 (en) | 2007-12-03 | 2015-08-11 | Valent U.S.A., Corporation | Seed treatment formulations |
| JP5650539B2 (ja) * | 2007-12-03 | 2015-01-07 | バレント・ユーエスエイ・コーポレイションＶａｌｅｎｔ Ｕ．Ｓ．Ａ．， Ｃｏｒｐｏｒａｔｉｏｎ | 種子処理製剤および使用方法 |
| EP2204366A1 (de) | 2008-12-19 | 2010-07-07 | Bayer CropScience AG | Herbizid und insektizid wirksame phenylsubstituierte Pyridazinone |
| WO2011035878A1 (de) | 2009-09-25 | 2011-03-31 | Bayer Cropscience Ag | Herbizid wirksame phenylsubstituierte pyridazinone |
| WO2011045271A1 (de) | 2009-10-15 | 2011-04-21 | Bayer Cropscience Ag | Herbizid wirksame heterocyclylsubstituierte pyridazinone |
| RU2013114184A (ru) | 2010-09-01 | 2014-10-10 | Байер Интеллектуэль Проперти Гмбх | Гербицидно-активные кетосультамы и дикетопиридины |
| CN106810550A (zh) * | 2017-01-10 | 2017-06-09 | 湖南华腾制药有限公司 | 一种萘啶衍生物的制备方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU407902A1 (ru) * | 1971-11-16 | 1973-12-10 | Институт органической химии Украинской ССР | Способ получения диэтилового эфира 3,4,5,6-тетрахлорпиридил-2-малоновой кислоты |
| IL108731A (en) * | 1993-03-04 | 1997-03-18 | Shell Int Research | 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES |
| IL108747A (en) * | 1993-03-04 | 1999-03-12 | Shell Int Research | Mushroom-killing preparations containing a history of 6 metamorphoses of 5 - 7 Dihalo - 1, 2 - 4 Triazlo [A-1,5] Pyrimidine Certain such new compounds and their preparation |
| EE200000706A (et) * | 1998-05-26 | 2002-06-17 | Warner-Lambert Company | Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid |
| US6156925A (en) * | 1998-09-25 | 2000-12-05 | American Cyanamid Company | Process for the preparation of halogenated phenylmaloates |
| EP1204323B1 (en) * | 1999-08-18 | 2004-07-14 | Aventis CropScience GmbH | Fungicides |
| KR20030013475A (ko) * | 2000-06-30 | 2003-02-14 | 와이어쓰 | 항암제로서의 치환된 트리아졸로피리미딘 |
| DE10063115A1 (de) * | 2000-12-18 | 2002-06-27 | Bayer Ag | Triazolopyrimidine |
| CA2453639A1 (en) * | 2001-07-18 | 2003-01-30 | Basf Aktiengesellschaft | Substituted 6-(2-tolyl)-triazolopyrimidines as fungicides |
| JPWO2004011467A1 (ja) * | 2002-07-29 | 2005-12-15 | 北興化学工業株式会社 | トリアゾロピリミジン誘導体および農園芸用殺菌剤 |
-
2003
- 2003-06-04 DE DE10325133A patent/DE10325133A1/de not_active Withdrawn
-
2004
- 2004-06-01 WO PCT/EP2004/005876 patent/WO2004108727A1/de not_active Ceased
- 2004-06-01 MX MXPA05012951A patent/MXPA05012951A/es unknown
- 2004-06-01 EP EP04735570A patent/EP1641798A1/de not_active Ceased
- 2004-06-01 BR BRPI0410906-6A patent/BRPI0410906A/pt not_active IP Right Cessation
- 2004-06-01 US US10/559,102 patent/US20070275985A1/en not_active Abandoned
- 2004-06-01 KR KR1020057022521A patent/KR20060015304A/ko not_active Withdrawn
- 2004-06-01 JP JP2006508237A patent/JP2006526587A/ja active Pending
- 2004-06-01 CN CNA2004800154818A patent/CN1802379A/zh active Pending
-
2005
- 2005-11-04 CR CR8074A patent/CR8074A/es not_active Application Discontinuation
- 2005-11-22 IL IL172098A patent/IL172098A0/en unknown
- 2005-11-29 ZA ZA200509637A patent/ZA200509637B/en unknown
- 2005-11-29 CO CO05121068A patent/CO5721005A2/es not_active Application Discontinuation
- 2005-12-02 EC EC2005006201A patent/ECSP056201A/es unknown