CO5721005A2 - Triazolopirimidinas - Google Patents

Triazolopirimidinas

Info

Publication number
CO5721005A2
CO5721005A2 CO05121068A CO05121068A CO5721005A2 CO 5721005 A2 CO5721005 A2 CO 5721005A2 CO 05121068 A CO05121068 A CO 05121068A CO 05121068 A CO05121068 A CO 05121068A CO 5721005 A2 CO5721005 A2 CO 5721005A2
Authority
CO
Colombia
Prior art keywords
substituted
carbon atoms
halogen
cycloalkyl
alkyl
Prior art date
Application number
CO05121068A
Other languages
English (en)
Inventor
Olaf Gebauer
Ulrich Heinemann
Hans-Ludwig Elbe
Herbert Gayer
Stefan Herrmann
Jorg Nico Greul
Bernd-Wielan Kruger
Stefan Hellebrand
Ronald Ebbert
Neumann Ulrike Wachendorff
Peter Dahmen
Karl Heinz Kuck
Original Assignee
Bayer Cropscience Aktiengesellshaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Aktiengesellshaft filed Critical Bayer Cropscience Aktiengesellshaft
Publication of CO5721005A2 publication Critical patent/CO5721005A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

1.- Triazolopirimidinas de la formula en la queR1 significa alquilo, en caso dado substituido, alquenilo, en caso dado substituido, alquinilo, en caso dado substituido, cicloalquilo en caso dado substituido o significa heterociclilo en caso dado substituido,R2 significa hidrogeno o alquilo, oR1 y R2 significan, en conjunto, junto con el atomo de nitrogeno, con el que estan enlazados, un anillo heterociclico, en caso dado substituido,R3 significa piridilo, en caso dado substituido o pirimidilo en caso dado substituido, y X significa halogeno.2.- Triazolopirimidinas de la formula (I), de conformidad con la reivindicacion 1, en las queR1 significa alquilo con 1 a 6 atomos de carbono, que puede estar substituido de una a cinco veces, de forma igual o de formas diferentes, por halogeno, por ciano, por hidroxi, por alcoxi con 1 a 4 atomos de carbono y/o por cicloalquilo con 3 a 6 atomos de carbono, oR1 significa alquenilo con 2 a 6 atomos de carbono, que puede estar substituido de una a tres veces, de forma igual o de formas diferentes, por halogeno, por ciano, por hidroxi, por alcoxi con 1 a 4 atomos de carbono y/o por cicloalquilo con 3 a 6 atomos de carbono, oR1 significa alquinilo con 3 a 6 atomos de carbono, que puede estar substituido de una a tres veces, de forma igual o de formas diferentes, por halogeno, por ciano, por alcoxi con 1 a 4 atomos de carbono y/o por cicloalquilo con 3 a 6 atomos de carbono, o R1 significa cicloalquilo con 3 a 6 atomos de carbono, que puede estar substituido de una a tres veces, de forma igual o de formas diferentes, por halogeno y/o alquilo con 1 a 4 atomos de carbono, oR1 significa heterociclilo saturado o insaturado con 5 o 6 miembros en el anillo y con 1 a 3 heteroatomos, tales como nitrogeno, oxigeno y/o azufre, pudiendo estar substituido el heterociclilo una o dos veces por halogeno, ...
CO05121068A 2003-06-04 2005-11-29 Triazolopirimidinas CO5721005A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10325133A DE10325133A1 (de) 2003-06-04 2003-06-04 Triazolopyrimidine

Publications (1)

Publication Number Publication Date
CO5721005A2 true CO5721005A2 (es) 2007-01-31

Family

ID=33482458

Family Applications (1)

Application Number Title Priority Date Filing Date
CO05121068A CO5721005A2 (es) 2003-06-04 2005-11-29 Triazolopirimidinas

Country Status (14)

Country Link
US (1) US20070275985A1 (es)
EP (1) EP1641798A1 (es)
JP (1) JP2006526587A (es)
KR (1) KR20060015304A (es)
CN (1) CN1802379A (es)
BR (1) BRPI0410906A (es)
CO (1) CO5721005A2 (es)
CR (1) CR8074A (es)
DE (1) DE10325133A1 (es)
EC (1) ECSP056201A (es)
IL (1) IL172098A0 (es)
MX (1) MXPA05012951A (es)
WO (1) WO2004108727A1 (es)
ZA (1) ZA200509637B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006066818A2 (de) * 2004-12-17 2006-06-29 Basf Aktiengesellschaft 7-AMINO-6-HETARYL-1,2,4-TRIAZOLO[1,5-a]PYRIMIDIN-VERBINDUNGEN UND IHRE VERWENDUNG ZUR BEKÄMPFUNG VON SCHADPILZEN
JP2008524149A (ja) * 2004-12-17 2008-07-10 ビーエーエスエフ ソシエタス・ヨーロピア ７−アミノ−６−ヘテロアリール−１，２，４−トリアゾロ［１，５−ａ］ピリミジンおよび有害な菌類を防除するためのそれらの使用
TW200643022A (en) * 2005-03-02 2006-12-16 Basf Ag 2-substituted 7-aminoazolopyrimidines, processes for their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
WO2006122740A2 (de) * 2005-05-17 2006-11-23 Basf Aktiengesellschaft 7-AMINO-6-HETARYLIMIDAZOLO[1,2-a]PYRIMIDIN-VERBINDUNGEN UND IHRE VERWENDUNG ZU BEKÄMPFUNG VON SCHADPILZEN
WO2007006723A1 (de) * 2005-07-13 2007-01-18 Basf Aktiengesellschaft 7-amino-6-tetrazolyl-1,2,4-triazolo[1,5-a]pyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen
WO2007101870A1 (de) * 2006-03-08 2007-09-13 Basf Se Substituierte triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
CN101153041B (zh) * 2006-09-28 2010-05-12 中国科学院化学研究所 1,2,3-三唑并1,3-二氮杂环化合物及其制备方法与应用
WO2008092836A2 (en) * 2007-01-30 2008-08-07 Basf Se Method for improving plant health
EP1952691A3 (en) * 2007-01-31 2008-09-17 Basf Se Method for improving plant health by application of a triazolopyrimidine derivative
JP5650539B2 (ja) * 2007-12-03 2015-01-07 バレント・ユーエスエイ・コーポレイションＶａｌｅｎｔ Ｕ．Ｓ．Ａ．， Ｃｏｒｐｏｒａｔｉｏｎ 種子処理製剤および使用方法
US9101131B2 (en) 2007-12-03 2015-08-11 Valent U.S.A., Corporation Seed treatment formulations
EP2204366A1 (de) 2008-12-19 2010-07-07 Bayer CropScience AG Herbizid und insektizid wirksame phenylsubstituierte Pyridazinone
WO2011035878A1 (de) 2009-09-25 2011-03-31 Bayer Cropscience Ag Herbizid wirksame phenylsubstituierte pyridazinone
WO2011045271A1 (de) 2009-10-15 2011-04-21 Bayer Cropscience Ag Herbizid wirksame heterocyclylsubstituierte pyridazinone
JP5990170B2 (ja) 2010-09-01 2016-09-07 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 除草活性を有するケトスルタム類及びジケトピリジン類
CN106810550A (zh) * 2017-01-10 2017-06-09 湖南华腾制药有限公司 一种萘啶衍生物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU407902A1 (ru) * 1971-11-16 1973-12-10 Институт органической химии Украинской ССР Способ получения диэтилового эфира 3,4,5,6-тетрахлорпиридил-2-малоновой кислоты
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
IL108747A (en) * 1993-03-04 1999-03-12 Shell Int Research Mushroom-killing preparations containing a history of 6 metamorphoses of 5 - 7 Dihalo - 1, 2 - 4 Triazlo [A-1,5] Pyrimidine Certain such new compounds and their preparation
EP1080092B1 (en) * 1998-05-26 2008-07-23 Warner-Lambert Company LLC Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
AU7278500A (en) * 1999-08-18 2001-03-13 Aventis Cropscience Gmbh Fungicides
PL360027A1 (en) * 2000-06-30 2004-09-06 Wyeth Substituted-triazolopyrimidines as anticancer agents
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
KR20040015358A (ko) * 2001-07-18 2004-02-18 바스프 악티엔게젤샤프트 살진균제인 치환된 6-(2-톨릴)-트리아졸로피리미딘
JPWO2004011467A1 (ja) * 2002-07-29 2005-12-15 北興化学工業株式会社 トリアゾロピリミジン誘導体および農園芸用殺菌剤

Also Published As

Publication number Publication date
EP1641798A1 (de) 2006-04-05
CN1802379A (zh) 2006-07-12
US20070275985A1 (en) 2007-11-29
MXPA05012951A (es) 2006-02-13
DE10325133A1 (de) 2004-12-23
IL172098A0 (en) 2009-02-11
CR8074A (es) 2007-09-11
ZA200509637B (en) 2007-02-28
ECSP056201A (es) 2006-04-19
JP2006526587A (ja) 2006-11-24
KR20060015304A (ko) 2006-02-16
WO2004108727A1 (de) 2004-12-16
BRPI0410906A (pt) 2006-06-27

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