JP2004508330A5 - - Google Patents

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Publication number
JP2004508330A5
JP2004508330A5 JP2002524497A JP2002524497A JP2004508330A5 JP 2004508330 A5 JP2004508330 A5 JP 2004508330A5 JP 2002524497 A JP2002524497 A JP 2002524497A JP 2002524497 A JP2002524497 A JP 2002524497A JP 2004508330 A5 JP2004508330 A5 JP 2004508330A5
Authority
JP
Japan
Prior art keywords
phenyl
alkyl
pyridin
pyrazolo
piperidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2002524497A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004508330A (ja
JP4129391B2 (ja
Filing date
Publication date
Priority claimed from US09/927,188 external-priority patent/US6635633B2/en
Application filed filed Critical
Priority claimed from PCT/US2001/027480 external-priority patent/WO2002020013A2/en
Publication of JP2004508330A publication Critical patent/JP2004508330A/ja
Publication of JP2004508330A5 publication Critical patent/JP2004508330A5/ja
Application granted granted Critical
Publication of JP4129391B2 publication Critical patent/JP4129391B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2002524497A 2000-09-06 2001-09-05 置換ピラゾールを用いてアレルギーを治療する方法 Expired - Fee Related JP4129391B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23040700P 2000-09-06 2000-09-06
US09/927,188 US6635633B2 (en) 2000-08-14 2001-08-10 Substituted pyrazoles
PCT/US2001/027480 WO2002020013A2 (en) 2000-09-06 2001-09-05 A method for treating allergies using substituted pyrazoles

Publications (3)

Publication Number Publication Date
JP2004508330A JP2004508330A (ja) 2004-03-18
JP2004508330A5 true JP2004508330A5 (https=) 2005-08-18
JP4129391B2 JP4129391B2 (ja) 2008-08-06

Family

ID=26924202

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002524497A Expired - Fee Related JP4129391B2 (ja) 2000-09-06 2001-09-05 置換ピラゾールを用いてアレルギーを治療する方法

Country Status (14)

Country Link
EP (1) EP1315492B1 (https=)
JP (1) JP4129391B2 (https=)
CN (1) CN1321641C (https=)
AT (1) ATE402699T1 (https=)
AU (2) AU2001288731B8 (https=)
CA (1) CA2421510A1 (https=)
DE (1) DE60135130D1 (https=)
DK (1) DK1315492T3 (https=)
ES (1) ES2309088T3 (https=)
HK (1) HK1052881B (https=)
MX (1) MXPA03001962A (https=)
NZ (1) NZ524682A (https=)
PT (1) PT1315492E (https=)
WO (1) WO2002020013A2 (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004531456A (ja) * 2000-09-06 2004-10-14 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド 置換ピラゾールを用いてアレルギーを治療する方法
ES2201899B1 (es) * 2002-04-01 2005-06-01 Almirall Prodesfarma, S.A. Derivados de la azaindolilpiperidina como agentes antihistaminicos y antialergicos.
ES2201907B1 (es) 2002-05-29 2005-06-01 Almirall Prodesfarma, S.A. Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos.
KR20070034049A (ko) 2004-06-09 2007-03-27 글락소 그룹 리미티드 피롤로피리딘 유도체
LT3141252T (lt) 2009-06-17 2018-11-12 Vertex Pharmaceuticals Inc. Gripo virusų replikacijos inhibitoriai
RU2013132681A (ru) 2010-12-16 2015-01-27 Вертекс Фармасьютикалз Инкорпорейтед Ингибиторы репликации вирусов гриппа
UA118010C2 (uk) 2011-08-01 2018-11-12 Вертекс Фармасьютікалз Інкорпорейтед Інгібітори реплікації вірусів грипу
EP2742046A1 (en) 2011-08-12 2014-06-18 F.Hoffmann-La Roche Ag PYRAZOLO[3,4-c]PYRIDINE COMPOUNDS AND METHODS OF USE
JP6618901B2 (ja) 2013-11-13 2019-12-11 バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated インフルエンザウイルスの複製の阻害剤を調製する方法
LT3068776T (lt) 2013-11-13 2019-08-12 Vertex Pharmaceuticals Incorporated Gripo virusų replikacijos inhibitoriai
EP3294735B8 (en) 2015-05-13 2022-01-05 Vertex Pharmaceuticals Incorporated Inhibitors of influenza viruses replication
EP3294717B1 (en) 2015-05-13 2020-07-29 Vertex Pharmaceuticals Inc. Methods of preparing inhibitors of influenza viruses replication
MX2021003904A (es) 2018-10-05 2021-10-26 Annapurna Bio Inc Compuestos y composiciones para el tratamiento de afecciones asociadas con la actividad del receptor apj.
CN111518019B (zh) * 2019-02-01 2023-10-24 江苏豪森药业集团有限公司 一种棕榈酸帕里哌酮中间体的制备方法
CN112142744A (zh) * 2019-06-28 2020-12-29 上海瑛派药业有限公司 取代的稠合杂芳双环化合物作为激酶抑制剂及其应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE789948A (fr) * 1971-10-13 1973-04-11 Sandoz Sa Nouveaux derives du pyrazole, leur preparation et leur application comme medicaments
JPH0615542B2 (ja) * 1986-07-22 1994-03-02 吉富製薬株式会社 ピラゾロピリジン化合物
JP3907220B2 (ja) * 1994-06-30 2007-04-18 エーザイ・アール・アンド・ディー・マネジメント株式会社 複素環含有化合物
JP3964478B2 (ja) * 1995-06-30 2007-08-22 エーザイ・アール・アンド・ディー・マネジメント株式会社 ヘテロ環含有カルボン酸誘導体及びそれを含有する医薬
AU7553198A (en) * 1997-06-12 1998-12-30 Sumitomo Pharmaceuticals Company, Limited Pyrazole derivatives

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