JP2003532737A5 - - Google Patents

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Publication number
JP2003532737A5
JP2003532737A5 JP2001582354A JP2001582354A JP2003532737A5 JP 2003532737 A5 JP2003532737 A5 JP 2003532737A5 JP 2001582354 A JP2001582354 A JP 2001582354A JP 2001582354 A JP2001582354 A JP 2001582354A JP 2003532737 A5 JP2003532737 A5 JP 2003532737A5
Authority
JP
Japan
Prior art keywords
hydroxy
pregna
methoxy
triene
hydroxymethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001582354A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003532737A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/GB2001/002103 external-priority patent/WO2001085755A1/en
Publication of JP2003532737A publication Critical patent/JP2003532737A/ja
Publication of JP2003532737A5 publication Critical patent/JP2003532737A5/ja
Pending legal-status Critical Current

Links

JP2001582354A 2000-05-11 2001-05-11 ２位置換プレグナ−１，３，５（１０）−トリエン誘導体およびコラン−１，３，５（１０）−トリエン誘導体およびそれらの生物活性 Pending JP2003532737A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20346200P 2000-05-11 2000-05-11
US60/203,462 2000-05-11
PCT/GB2001/002103 WO2001085755A1 (en) 2000-05-11 2001-05-11 2-substituted pregna-1, 3, 5 (10) -triene and chola-1, 3, 5 (10)-triene derivatives and their biological activity

Publications (2)

Publication Number Publication Date
JP2003532737A JP2003532737A (ja) 2003-11-05
JP2003532737A5 true JP2003532737A5 (enExample) 2006-01-05

Family

ID=22754111

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001582354A Pending JP2003532737A (ja) 2000-05-11 2001-05-11 ２位置換プレグナ−１，３，５（１０）−トリエン誘導体およびコラン−１，３，５（１０）−トリエン誘導体およびそれらの生物活性

Country Status (16)

Country Link
EP (1) EP1287017B1 (enExample)
JP (1) JP2003532737A (enExample)
KR (1) KR100740354B1 (enExample)
CN (1) CN100338088C (enExample)
AT (1) ATE301130T1 (enExample)
AU (1) AU784563B2 (enExample)
CA (1) CA2408751A1 (enExample)
CZ (1) CZ298835B6 (enExample)
DE (1) DE60112438T2 (enExample)
DK (1) DK1287017T3 (enExample)
ES (1) ES2247102T3 (enExample)
IL (2) IL152728A0 (enExample)
NO (1) NO323857B1 (enExample)
NZ (1) NZ523042A (enExample)
WO (1) WO2001085755A1 (enExample)
ZA (1) ZA200209060B (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6908910B2 (en) 1993-08-06 2005-06-21 The Children's Medical Center Corporation Estrogenic compounds as anti-mitotic agents
US7135581B2 (en) 2000-08-18 2006-11-14 Entremed, Inc. Antiangiogenic agents
US6995278B2 (en) 2000-08-18 2006-02-07 Entre Med, Inc. Antiangiogenic agents
JP2004537499A (ja) * 2000-11-27 2004-12-16 エントレメッド インコーポレイテッド 抗血管新生薬
WO2002092100A1 (en) * 2001-05-11 2002-11-21 Marsden, John, Christopher 17-(c(ch3) (ch2) o-3c (r4, r5) n (r6, r7))-substituted 19-nor-pregna-1, 3, 5(10)-triene derivatives and their medical use
AU2004224053B2 (en) 2003-03-24 2011-06-09 Sterix Limited Oestrogen derivatives as inhibitors of steroid sulphatase
AU2004275693A1 (en) 2003-05-28 2005-04-07 Entremed, Inc. Antiangiogenic agents
JP2007529426A (ja) 2004-03-12 2007-10-25 エントレメッド インコーポレイテッド 抗血管新生薬
CA2646065C (en) 2006-03-20 2014-01-14 Entremed, Inc. Disease modifying anti-arthritic activity of 2-methoxyestradiol

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3562260A (en) * 1965-08-23 1971-02-09 Ormonoterapia Richter Spa 2-carbonyl-estratrienes and method of their preparation
JPS54112850A (en) * 1978-02-23 1979-09-04 Mitsubishi Chem Ind Ltd Steroid derivative and its preparation
JPS54112580A (en) * 1978-02-23 1979-09-03 Nec Corp Electroless discharge lamp
JPS54112849A (en) * 1978-02-23 1979-09-04 Mitsubishi Chem Ind Ltd Preparation of steroid derivative
JPS54117456A (en) * 1978-03-02 1979-09-12 Mitsubishi Chem Ind Ltd Alkoxysteroid derivative
JPS54117454A (en) * 1978-03-02 1979-09-12 Mitsubishi Chem Ind Ltd Acylsteroid derivative
JPS54117455A (en) * 1978-03-02 1979-09-12 Mitsubishi Chem Ind Ltd Novel 19-norsteroid derivative
GB9804861D0 (en) * 1998-03-06 1998-04-29 Res Inst Medicine Chem Chemical compounds
GB9910934D0 (en) * 1999-05-11 1999-07-14 Res Inst Medicine Chem Chemical compounds

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