JP2003503340A - 短時間型催眠薬またはその塩からなる二重持効性剤形 - Google Patents
短時間型催眠薬またはその塩からなる二重持効性剤形Info
- Publication number
- JP2003503340A JP2003503340A JP2001505891A JP2001505891A JP2003503340A JP 2003503340 A JP2003503340 A JP 2003503340A JP 2001505891 A JP2001505891 A JP 2001505891A JP 2001505891 A JP2001505891 A JP 2001505891A JP 2003503340 A JP2003503340 A JP 2003503340A
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Anesthesiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP99401605A EP1064937A1 (en) | 1999-06-28 | 1999-06-28 | Timed dual release dosage forms comprising a short acting hypnotic or a salt thereof |
| EP99401605.3 | 1999-06-28 | ||
| PCT/EP2000/006792 WO2001000181A2 (en) | 1999-06-28 | 2000-06-27 | Timed dual release dosage forms comprising a short acting hypnotic or a salt thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2003503340A true JP2003503340A (ja) | 2003-01-28 |
| JP2003503340A5 JP2003503340A5 (https=) | 2007-08-02 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001505891A Pending JP2003503340A (ja) | 1999-06-28 | 2000-06-27 | 短時間型催眠薬またはその塩からなる二重持効性剤形 |
Country Status (28)
| Country | Link |
|---|---|
| EP (2) | EP1064937A1 (https=) |
| JP (1) | JP2003503340A (https=) |
| KR (1) | KR20020015064A (https=) |
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| CA (1) | CA2370556C (https=) |
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| DE (1) | DE60011617T2 (https=) |
| DK (1) | DK1194132T3 (https=) |
| ES (1) | ES2222223T3 (https=) |
| HK (1) | HK1043057B (https=) |
| HU (1) | HU227810B1 (https=) |
| IL (1) | IL146928A0 (https=) |
| MX (1) | MXPA01013212A (https=) |
| NO (1) | NO20016283L (https=) |
| NZ (1) | NZ515997A (https=) |
| PL (1) | PL201777B1 (https=) |
| PT (1) | PT1194132E (https=) |
| SI (1) | SI1194132T1 (https=) |
| SK (1) | SK285347B6 (https=) |
| TR (1) | TR200103594T2 (https=) |
| TW (1) | TWI285118B (https=) |
| WO (1) | WO2001000181A2 (https=) |
| ZA (1) | ZA200110005B (https=) |
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| JP2006096729A (ja) * | 2004-09-30 | 2006-04-13 | Nippon Zoki Pharmaceut Co Ltd | 固形医薬製剤 |
| JP2008105969A (ja) * | 2006-10-24 | 2008-05-08 | Kobayashi Kako Kk | 酒石酸ゾルピデム組成物 |
| JP2008546830A (ja) * | 2005-06-28 | 2008-12-25 | サノフイ−アベンテイス | ｐＨ依存性の溶解度を有する有効成分の持続放出製剤 |
| JP2009532331A (ja) * | 2006-03-02 | 2009-09-10 | ワトソン ファーマスーティカルズ インコーポレーテッド | 鎮静剤および睡眠剤の経口放出制御製剤 |
| JP2010521437A (ja) * | 2007-03-15 | 2010-06-24 | ポリケム・エスエイ | 時間特異的遅延／パルス放出剤形 |
| JP2012510987A (ja) * | 2008-12-04 | 2012-05-17 | インテック ファーマ リミテッド | ザレプロン胃内滞留性薬剤送達システム |
| JP2012532866A (ja) * | 2009-07-07 | 2012-12-20 | サノビオン ファーマシューティカルズ インク | ６−（５−クロロ−２−ピリジル）−５−［（４−メチル−１−ピペラジニル）カルボニルオキシ］−７−オキソ−６，７−ジヒドロ−５ｈ−ピロロ［３，４−ｂ］ピラジンの配合物 |
| JP2013501763A (ja) * | 2009-08-12 | 2013-01-17 | デブルジャ・ゼ・タソシエ・ファルマ | 薬物誤用に対する新規の医薬製剤 |
| JP2013521332A (ja) * | 2010-03-05 | 2013-06-10 | ユニヴァーシティー オヴ ストラスクライド | パルス状薬剤放出 |
| JP2013545784A (ja) * | 2010-12-16 | 2013-12-26 | サノフイ | 誤用を防止することを目的とする経口投与用医薬組成物 |
| JP2014501739A (ja) * | 2010-12-16 | 2014-01-23 | サノフイ | ゾルピデムベースの口腔内崩壊医薬錠剤 |
| US9283192B2 (en) | 2010-03-05 | 2016-03-15 | University Of Strathclyde | Delayed prolonged drug delivery |
| JP2016536371A (ja) * | 2014-02-06 | 2016-11-24 | シーケンシャル メディシン リミテッド | 睡眠を補助する組成物及び方法 |
| US10137091B2 (en) | 2010-03-05 | 2018-11-27 | University Of Strathclyde | Immediate/delayed drug delivery |
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| EP1064938A1 (en) * | 1999-06-28 | 2001-01-03 | Sanofi-Synthelabo | Pharmaceutical dosage forms for controlled release producing at least a timed pulse |
| DE60003194T2 (de) * | 1999-08-26 | 2004-06-17 | Neurocrine Biosciences, Inc., San Diego | Sedativ hypnotische zusammensetzungen mit gesteuerter freisetzung und diesbezügliche verfahren |
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| US8329216B2 (en) | 2001-07-06 | 2012-12-11 | Endo Pharmaceuticals Inc. | Oxymorphone controlled release formulations |
| KR20030048026A (ko) | 2001-07-06 | 2003-06-18 | 펜웨스트 파머슈티칼즈 컴파니 | 옥시모르폰의 서방형 제제 |
| CN1610551A (zh) | 2001-07-06 | 2005-04-27 | 恩德制药公司 | 用作止痛剂的6－羟基羟吗啡酮的肠胃外给药 |
| JP4417110B2 (ja) * | 2001-12-19 | 2010-02-17 | 株式会社三和化学研究所 | 放出制御型成型品 |
| EP1941878A1 (en) * | 2002-01-10 | 2008-07-09 | Biovail Laboratories International Srl | Sedative non-benzodiazepine formulations |
| ES2301797T3 (es) * | 2002-01-10 | 2008-07-01 | Biovail Laboratories International Srl | Formulaciones sedantes no benzodiazepinicas. |
| US20030165566A1 (en) * | 2002-01-10 | 2003-09-04 | O'toole Edel | Sedative non-benzodiazepine formulations |
| CA2503121A1 (en) * | 2002-10-25 | 2004-05-13 | Collegium Pharmaceutical, Inc. | Pulsatile release compositions of milnacipran |
| GB0423964D0 (en) * | 2004-10-28 | 2004-12-01 | Jagotec Ag | Dosage form |
| AU2006322314A1 (en) * | 2005-11-18 | 2007-06-14 | Synthon B.V. | Zolpidem tablets |
| AR056633A1 (es) * | 2005-12-07 | 2007-10-17 | Gador Sa | Composiciones farmaceuticas de agentes hipnoticos de accion corta en forma de liberacion modificada y los procedimientos para preparar dichas formulaciones |
| KR20070091960A (ko) * | 2006-03-08 | 2007-09-12 | 주식회사종근당 | 졸피뎀 또는 그의 염을 포함하는 안전한 제어방출형 제제조성물 |
| AU2013202441B2 (en) * | 2006-04-26 | 2016-02-25 | Alphapharm Pty Ltd | Controlled release formulations comprising uncoated discrete unit(s) and an extended release matrix |
| NZ703464A (en) | 2006-04-26 | 2016-05-27 | Alphapharm Pty Ltd | Controlled release formulations comprising uncoated discrete unit(s) and an extended release matrix |
| EP1938805A1 (en) * | 2006-12-22 | 2008-07-02 | LEK Pharmaceuticals D.D. | Monolithic sustained release zolpidem tablets |
| WO2009021127A2 (en) * | 2007-08-07 | 2009-02-12 | Neurogen Corporation | Controlled released compositions |
| KR101601649B1 (ko) | 2008-04-18 | 2016-03-09 | 인텍 파마 리미티드 | 카르비도파／레보도파 위체류 약물 전달 |
| US20100068256A1 (en) | 2008-09-16 | 2010-03-18 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Ex vivo modifiable medicament release-substance |
| RU2384336C1 (ru) * | 2009-04-22 | 2010-03-20 | Маргарита Алексеевна Морозова | Фармацевтический состав для коррекции психосоматических проявлений |
| TWI505841B (zh) * | 2011-09-29 | 2015-11-01 | Taiwan Biotech Co Ltd | 治療睡眠障礙之控釋調配物 |
| RU2659200C1 (ru) * | 2017-07-24 | 2018-06-28 | Общество С Ограниченной Ответственностью "Валента - Интеллект" | Фармацевтический состав, содержащий алимемазина тартрат |
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Cited By (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006096729A (ja) * | 2004-09-30 | 2006-04-13 | Nippon Zoki Pharmaceut Co Ltd | 固形医薬製剤 |
| JP2008546830A (ja) * | 2005-06-28 | 2008-12-25 | サノフイ−アベンテイス | ｐＨ依存性の溶解度を有する有効成分の持続放出製剤 |
| JP2009532331A (ja) * | 2006-03-02 | 2009-09-10 | ワトソン ファーマスーティカルズ インコーポレーテッド | 鎮静剤および睡眠剤の経口放出制御製剤 |
| JP2008105969A (ja) * | 2006-10-24 | 2008-05-08 | Kobayashi Kako Kk | 酒石酸ゾルピデム組成物 |
| JP2010521437A (ja) * | 2007-03-15 | 2010-06-24 | ポリケム・エスエイ | 時間特異的遅延／パルス放出剤形 |
| JP2012510987A (ja) * | 2008-12-04 | 2012-05-17 | インテック ファーマ リミテッド | ザレプロン胃内滞留性薬剤送達システム |
| JP2012532866A (ja) * | 2009-07-07 | 2012-12-20 | サノビオン ファーマシューティカルズ インク | ６−（５−クロロ−２−ピリジル）−５−［（４−メチル−１−ピペラジニル）カルボニルオキシ］−７−オキソ−６，７−ジヒドロ−５ｈ−ピロロ［３，４−ｂ］ピラジンの配合物 |
| JP2013501763A (ja) * | 2009-08-12 | 2013-01-17 | デブルジャ・ゼ・タソシエ・ファルマ | 薬物誤用に対する新規の医薬製剤 |
| JP2013521332A (ja) * | 2010-03-05 | 2013-06-10 | ユニヴァーシティー オヴ ストラスクライド | パルス状薬剤放出 |
| US9283192B2 (en) | 2010-03-05 | 2016-03-15 | University Of Strathclyde | Delayed prolonged drug delivery |
| JP2016040309A (ja) * | 2010-03-05 | 2016-03-24 | ユニヴァーシティー オヴ ストラスクライド | パルス状薬剤放出 |
| US10137091B2 (en) | 2010-03-05 | 2018-11-27 | University Of Strathclyde | Immediate/delayed drug delivery |
| US11065205B2 (en) | 2010-03-05 | 2021-07-20 | Drug Delivery International Limited | Immediate/delayed drug delivery |
| JP2013545784A (ja) * | 2010-12-16 | 2013-12-26 | サノフイ | 誤用を防止することを目的とする経口投与用医薬組成物 |
| JP2014501739A (ja) * | 2010-12-16 | 2014-01-23 | サノフイ | ゾルピデムベースの口腔内崩壊医薬錠剤 |
| JP2016536371A (ja) * | 2014-02-06 | 2016-11-24 | シーケンシャル メディシン リミテッド | 睡眠を補助する組成物及び方法 |
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