JP2002541237A5 - - Google Patents

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Publication number
JP2002541237A5
JP2002541237A5 JP2000610819A JP2000610819A JP2002541237A5 JP 2002541237 A5 JP2002541237 A5 JP 2002541237A5 JP 2000610819 A JP2000610819 A JP 2000610819A JP 2000610819 A JP2000610819 A JP 2000610819A JP 2002541237 A5 JP2002541237 A5 JP 2002541237A5
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JP
Japan
Prior art keywords
composition
prodrug
pharmaceutically acceptable
acceptable salt
asp
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000610819A
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English (en)
Japanese (ja)
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JP2002541237A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2000/009319 external-priority patent/WO2000061542A1/en
Publication of JP2002541237A publication Critical patent/JP2002541237A/ja
Publication of JP2002541237A5 publication Critical patent/JP2002541237A5/ja
Pending legal-status Critical Current

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JP2000610819A 1999-04-09 2000-04-07 カスパーゼインヒビターおよびその使用 Pending JP2002541237A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US12854599P 1999-04-09 1999-04-09
US60/128,545 1999-04-09
US15837099P 1999-10-12 1999-10-12
US60/158,370 1999-10-12
PCT/US2000/009319 WO2000061542A1 (en) 1999-04-09 2000-04-07 Caspase inhibitors and the use thereof

Publications (2)

Publication Number Publication Date
JP2002541237A JP2002541237A (ja) 2002-12-03
JP2002541237A5 true JP2002541237A5 (enExample) 2007-06-14

Family

ID=26826691

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000610819A Pending JP2002541237A (ja) 1999-04-09 2000-04-07 カスパーゼインヒビターおよびその使用

Country Status (12)

Country Link
US (3) US6355618B1 (enExample)
EP (1) EP1177168B1 (enExample)
JP (1) JP2002541237A (enExample)
KR (1) KR20020005665A (enExample)
CN (1) CN1176941C (enExample)
AT (1) ATE363465T1 (enExample)
AU (1) AU4213500A (enExample)
BR (1) BR0009610A (enExample)
CA (1) CA2369619A1 (enExample)
DE (1) DE60035037T2 (enExample)
MX (1) MXPA01010127A (enExample)
WO (1) WO2000061542A1 (enExample)

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JP6836996B2 (ja) * 2015-02-25 2021-03-03 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ 新しいトリフルオロメチルプロパンアミド誘導体
CN106317161B (zh) * 2015-06-29 2020-05-15 深圳翰宇药业股份有限公司 一种氟甲基酮肽系列化合物的制备方法
CN108699106B (zh) * 2016-03-04 2021-11-30 豪夫迈·罗氏有限公司 作为htra1抑制剂的新型三氟甲基丙酰胺衍生物
CN108699105A (zh) 2016-03-04 2018-10-23 豪夫迈·罗氏有限公司 作为htra1抑制剂的新型二氟酮酰胺衍生物
US11186541B2 (en) * 2016-03-28 2021-11-30 The University Of Toledo Potent inhibitors of aspartate N-acetyl-transferase for the treatment of Canavan disease
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