JP2001505567A5 - - Google Patents

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Publication number
JP2001505567A5
JP2001505567A5 JP1998524218A JP52421898A JP2001505567A5 JP 2001505567 A5 JP2001505567 A5 JP 2001505567A5 JP 1998524218 A JP1998524218 A JP 1998524218A JP 52421898 A JP52421898 A JP 52421898A JP 2001505567 A5 JP2001505567 A5 JP 2001505567A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1998524218A
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English (en)
Japanese (ja)
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JP4422800B2 (ja
JP2001505567A (ja
Filing date
Publication date
Priority claimed from DE19649460A external-priority patent/DE19649460A1/de
Application filed filed Critical
Publication of JP2001505567A publication Critical patent/JP2001505567A/ja
Publication of JP2001505567A5 publication Critical patent/JP2001505567A5/ja
Application granted granted Critical
Publication of JP4422800B2 publication Critical patent/JP4422800B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP52421898A 1996-11-26 1997-11-14 心臓循環系疾患の処置のための新規な置換ピラゾール誘導体 Expired - Fee Related JP4422800B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19649460A DE19649460A1 (de) 1996-11-26 1996-11-26 Neue substituierte Pyrazolderivate
DE19649460.5 1996-11-26
PCT/EP1997/006366 WO1998023619A1 (de) 1996-11-26 1997-11-14 Neue substituierte pyrazolderivate zur behandlung von herzkreislauferkrankungen

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2009210476A Division JP2010013475A (ja) 1996-11-26 2009-09-11 新規な置換ピラゾール誘導体

Publications (3)

Publication Number Publication Date
JP2001505567A JP2001505567A (ja) 2001-04-24
JP2001505567A5 true JP2001505567A5 (cg-RX-API-DMAC10.html) 2005-05-12
JP4422800B2 JP4422800B2 (ja) 2010-02-24

Family

ID=7813100

Family Applications (2)

Application Number Title Priority Date Filing Date
JP52421898A Expired - Fee Related JP4422800B2 (ja) 1996-11-26 1997-11-14 心臓循環系疾患の処置のための新規な置換ピラゾール誘導体
JP2009210476A Ceased JP2010013475A (ja) 1996-11-26 2009-09-11 新規な置換ピラゾール誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2009210476A Ceased JP2010013475A (ja) 1996-11-26 2009-09-11 新規な置換ピラゾール誘導体

Country Status (25)

Country Link
EP (1) EP0944631B1 (cg-RX-API-DMAC10.html)
JP (2) JP4422800B2 (cg-RX-API-DMAC10.html)
CN (1) CN1122032C (cg-RX-API-DMAC10.html)
AR (1) AR010310A1 (cg-RX-API-DMAC10.html)
AT (1) ATE259812T1 (cg-RX-API-DMAC10.html)
AU (1) AU729642B2 (cg-RX-API-DMAC10.html)
BR (1) BR9714363A (cg-RX-API-DMAC10.html)
CA (1) CA2272584C (cg-RX-API-DMAC10.html)
CZ (1) CZ185099A3 (cg-RX-API-DMAC10.html)
DE (2) DE19649460A1 (cg-RX-API-DMAC10.html)
DK (1) DK0944631T3 (cg-RX-API-DMAC10.html)
EE (1) EE9900211A (cg-RX-API-DMAC10.html)
ES (1) ES2214646T3 (cg-RX-API-DMAC10.html)
HU (1) HUP0000562A3 (cg-RX-API-DMAC10.html)
ID (1) ID21881A (cg-RX-API-DMAC10.html)
IL (1) IL129998A0 (cg-RX-API-DMAC10.html)
MX (1) MXPA99004826A (cg-RX-API-DMAC10.html)
NO (1) NO992400D0 (cg-RX-API-DMAC10.html)
NZ (1) NZ335890A (cg-RX-API-DMAC10.html)
PT (1) PT944631E (cg-RX-API-DMAC10.html)
SK (1) SK67699A3 (cg-RX-API-DMAC10.html)
TR (1) TR199901172T2 (cg-RX-API-DMAC10.html)
TW (1) TW403746B (cg-RX-API-DMAC10.html)
WO (1) WO1998023619A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA9710573B (cg-RX-API-DMAC10.html)

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DE19920352A1 (de) * 1999-05-04 2000-11-09 Bayer Ag Substituiertes Pyrazolderivat
DE19943634A1 (de) 1999-09-13 2001-04-12 Bayer Ag Neuartige Dicarbonsäurederivate mit pharmazeutischen Eigenschaften
DE19943635A1 (de) 1999-09-13 2001-03-15 Bayer Ag Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften
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DE10021069A1 (de) * 2000-04-28 2001-10-31 Bayer Ag Substituiertes Pyrazolderivat
DE10057754A1 (de) 2000-11-22 2002-05-23 Bayer Ag Neue Sulfonamid-substituierte Pyrazolopyridinderivate
AR031176A1 (es) 2000-11-22 2003-09-10 Bayer Ag Nuevos derivados de pirazolpiridina sustituidos con piridina
WO2002042299A1 (de) 2000-11-22 2002-05-30 Bayer Aktiengesellschaft Neue lactam-substituierte pyrazolopyridinderivate
DE10057751A1 (de) 2000-11-22 2002-05-23 Bayer Ag Neue Carbamat-substituierte Pyrazolopyridinderivate
DE10109861A1 (de) 2001-03-01 2002-09-05 Bayer Ag Neuartige seitenkettenhalogenierte Aminodicarbonsäurederivate
DE10109858A1 (de) 2001-03-01 2002-09-05 Bayer Ag Neuartige halogensubstituierte Aminodicarbonsäurederivate
DE10110749A1 (de) * 2001-03-07 2002-09-12 Bayer Ag Substituierte Aminodicarbonsäurederivate
DE10122894A1 (de) 2001-05-11 2002-11-14 Bayer Ag Neue Sulfonat-substituierte Pyrazolopyridinderivate
DE10132416A1 (de) * 2001-07-04 2003-01-16 Bayer Ag Neue Morpholin-überbrückte Pyrazolopyridinderivate
DE10220570A1 (de) 2002-05-08 2003-11-20 Bayer Ag Carbamat-substituierte Pyrazolopyridine
DE10232572A1 (de) * 2002-07-18 2004-02-05 Bayer Ag Neue 2,5-disubstituierte Pyrimidinderivate
DE10244810A1 (de) * 2002-09-26 2004-04-08 Bayer Ag Neue Morpholin-überbrückte Indazolderivate
WO2005030121A2 (en) * 2003-06-30 2005-04-07 Hif Bio, Inc. Compounds, compositions and methods
DE102005050377A1 (de) 2005-10-21 2007-04-26 Bayer Healthcare Ag Heterocyclische Verbindungen und ihre Verwendung
DE102005050497A1 (de) 2005-10-21 2007-04-26 Bayer Healthcare Ag Difluorphenol-Derivate und ihre Verwendung
DE102005050375A1 (de) 2005-10-21 2007-04-26 Bayer Healthcare Ag Tetrazol-Derivate und ihre Verwendung
DE102005050376A1 (de) 2005-10-21 2007-05-31 Bayer Healthcare Ag Dicarbonsäure-Derivate und ihre Verwendung
DE102005050498A1 (de) 2005-10-21 2007-06-06 Bayer Healthcare Aktiengesellschaft Cyclopropylessigsäure-Derivate und ihre Verwendung
DE102006020327A1 (de) * 2006-04-27 2007-12-27 Bayer Healthcare Ag Heterocyclisch substituierte, anellierte Pyrazol-Derivate und ihre Verwendung
DE102006043443A1 (de) 2006-09-15 2008-03-27 Bayer Healthcare Ag Neue aza-bicyclische Verbindungen und ihre Verwendung
DE102007015035A1 (de) 2007-03-29 2008-10-02 Bayer Healthcare Ag Substituierte Dibenzoesäure-Derivate und ihre Verwendung
DE102007015034A1 (de) 2007-03-29 2008-10-02 Bayer Healthcare Ag Lactam-substituierte Dicarbonsäuren und ihre Verwendung
DE102007026392A1 (de) 2007-06-06 2008-12-11 Bayer Healthcare Ag Lösungen für die Perfusion und Konservierung von Organen und Geweben
DE102007028319A1 (de) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituierte Oxazolidinone und ihre Verwendung
DE102007028406A1 (de) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituierte Oxazolidinone und ihre Verwendung
DE102007028320A1 (de) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituierte Oxazolidinone und ihre Verwendung
DE102007028407A1 (de) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituierte Oxazolidinone und ihre Verwendung
SI2294066T1 (sl) 2008-04-28 2014-12-31 Janssen Pharmaceutica N.V. Benzoimidazoli kot inhibitorji prolil-hidroksilaze
EP2138178A1 (en) 2008-06-28 2009-12-30 Bayer Schering Pharma Aktiengesellschaft Oxazolidninones for the treatment fo chronic obstructive pulmonary disease (COPD) and/or asthma
DE102008063992A1 (de) 2008-12-19 2010-09-02 Lerner, Zinoviy, Dipl.-Ing. Neue aliphatisch substituierte Pyrazolopyridine und ihre Verwendung
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
UY33041A (es) 2009-11-27 2011-06-30 Bayer Schering Pharma Aktienegesellschaft Procedimiento para la preparaciòn de {4,6-diamino-2-[1-(2-fluorobencil)-1h-pirazolo[3,4-b]piridin-3-il]pirimidin-5-il}carbamato de metilo y su purificaciòn para el uso como principio activo farmacèutico
GB201004311D0 (en) 2010-03-15 2010-04-28 Proximagen Ltd New enzyme inhibitor compounds
DK2588465T3 (en) 2010-06-30 2017-05-01 Ironwood Pharmaceuticals Inc SGC stimulators
CN107266433A (zh) 2010-11-09 2017-10-20 铁木医药有限公司 sGC刺激剂
US9090610B2 (en) * 2011-04-21 2015-07-28 Bayer Intellectual Property Gmbh Fluoroalkyl-substituted pyrazolopyridines and use thereof
BR112014005793A2 (pt) 2011-09-14 2017-03-28 Proximagen Ltd compostos inibidores de enzimas
US9139564B2 (en) 2011-12-27 2015-09-22 Ironwood Pharmaceuticals, Inc. 2-benzyl, 3-(pyrimidin-2-yl) substituted pyrazoles useful as sGC stimulators
BR112014027952B1 (pt) 2012-05-10 2022-06-21 Bayer Pharma Aktiengesellschaft Anticorpos monoclonais humanos capazes de se ligarem ao fator de coagulação xi, seu uso, composição farmacêutica e medicamento os compreendendo, ácido nucleico que o codifica, bem como vetor
EP3094327A1 (en) 2014-01-13 2016-11-23 Ironwood Pharmaceuticals, Inc. USE OF sGC STIMULATORS FOR THE TREATMENT OF NEUROMUSCULAR DISORDERS
JP6748113B2 (ja) 2015-05-06 2020-08-26 バイエル・ファルマ・アクティエンゲゼルシャフト 全身性硬化症(SSc)に付随する指潰瘍(DU)を治療するための単独のまたはPDE5阻害剤と組み合わせたsGC刺激剤、sGC活性化剤の使用
CN113750102A (zh) 2015-07-23 2021-12-07 拜耳制药股份公司 可溶性鸟苷酸环化酶的刺激剂和/或活化剂及其用途
MX2018007152A (es) 2015-12-14 2018-08-15 Ironwood Pharmaceuticals Inc Uso de estimuladores de guanilato ciclasa soluble (sgc) para el tratamiento de la disfuncion del esfinter gastrointestinal.
WO2017121700A1 (de) * 2016-01-15 2017-07-20 Bayer Pharma Aktiengesellschaft 1,3-disubstituierte 1h-pyrazolo[3,4-b]pyridin- derivate und ihre verwendung als stimulatoren der löslichen guanylatcyclase
JP7237823B2 (ja) 2016-10-11 2023-03-13 バイエル ファーマ アクチエンゲゼルシャフト Sgcアクチベーターとミネラルコルチコイド受容体アンタゴニストとを含む組合せ
CA3039734A1 (en) 2016-10-11 2018-04-19 Bayer Pharma Aktiengesellschaft Combination containing sgc stimulators and mineralocorticoid receptor antagonists
US20190381039A1 (en) 2016-12-13 2019-12-19 Cyclerion Therapeutics, Inc. USE OF sGC STIMULATORS FOR THE TREATMENT OF ESOPHAGEAL MOTILITY DISORDERS
ES2924359T3 (es) 2017-04-11 2022-10-06 Sunshine Lake Pharma Co Ltd Compuestos de indazol sustituidos con flúor y usos de los mismos
BR112020022340A2 (pt) 2018-05-15 2021-02-02 Bayer Aktiengesellschaft benzamidas substituídas por 1,3-tiazol-2-il para o tratamento de doenças associadas com sensibilização de fibras nervosas
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