JP2000515866A5 - - Google Patents

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Publication number
JP2000515866A5
JP2000515866A5 JP1998508318A JP50831898A JP2000515866A5 JP 2000515866 A5 JP2000515866 A5 JP 2000515866A5 JP 1998508318 A JP1998508318 A JP 1998508318A JP 50831898 A JP50831898 A JP 50831898A JP 2000515866 A5 JP2000515866 A5 JP 2000515866A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1998508318A
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English (en)
Japanese (ja)
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JP4033494B2 (ja
JP2000515866A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/013244 external-priority patent/WO1998004569A1/en
Publication of JP2000515866A publication Critical patent/JP2000515866A/ja
Publication of JP2000515866A5 publication Critical patent/JP2000515866A5/ja
Application granted granted Critical
Publication of JP4033494B2 publication Critical patent/JP4033494B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP50831898A 1996-07-26 1997-07-25 ヌクレオチドアナログ Expired - Lifetime JP4033494B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US68683896A 1996-07-26 1996-07-26
US2270896P 1996-07-26 1996-07-26
US08/686,838 1996-07-26
US60/022,708 1996-07-26
PCT/US1997/013244 WO1998004569A1 (en) 1996-07-26 1997-07-25 Nucleotide analogs

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2007180398A Division JP2007297406A (ja) 1996-07-26 2007-07-09 ヌクレオチドアナログ

Publications (3)

Publication Number Publication Date
JP2000515866A JP2000515866A (ja) 2000-11-28
JP2000515866A5 true JP2000515866A5 (enExample) 2004-08-19
JP4033494B2 JP4033494B2 (ja) 2008-01-16

Family

ID=26696272

Family Applications (6)

Application Number Title Priority Date Filing Date
JP50831898A Expired - Lifetime JP4033494B2 (ja) 1996-07-26 1997-07-25 ヌクレオチドアナログ
JP2007180398A Withdrawn JP2007297406A (ja) 1996-07-26 2007-07-09 ヌクレオチドアナログ
JP2010233086A Withdrawn JP2011016847A (ja) 1996-07-26 2010-10-15 ヌクレオチドアナログ
JP2014083387A Withdrawn JP2014159450A (ja) 1996-07-26 2014-04-15 ヌクレオチドアナログ
JP2015091141A Withdrawn JP2015164934A (ja) 1996-07-26 2015-04-28 ヌクレオチドアナログ
JP2016212748A Withdrawn JP2017031212A (ja) 1996-07-26 2016-10-31 ヌクレオチドアナログ

Family Applications After (5)

Application Number Title Priority Date Filing Date
JP2007180398A Withdrawn JP2007297406A (ja) 1996-07-26 2007-07-09 ヌクレオチドアナログ
JP2010233086A Withdrawn JP2011016847A (ja) 1996-07-26 2010-10-15 ヌクレオチドアナログ
JP2014083387A Withdrawn JP2014159450A (ja) 1996-07-26 2014-04-15 ヌクレオチドアナログ
JP2015091141A Withdrawn JP2015164934A (ja) 1996-07-26 2015-04-28 ヌクレオチドアナログ
JP2016212748A Withdrawn JP2017031212A (ja) 1996-07-26 2016-10-31 ヌクレオチドアナログ

Country Status (4)

Country Link
JP (6) JP4033494B2 (enExample)
CA (1) CA2261619C (enExample)
TW (2) TW444020B (enExample)
WO (1) WO1998004569A1 (enExample)

Families Citing this family (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998004569A1 (en) * 1996-07-26 1998-02-05 Gilead Sciences, Inc. Nucleotide analogs
BR9811552A (pt) * 1997-07-25 2000-08-29 Gilead Sciences Inc Composições de análogos de nucleotìdeos
DK1243590T3 (da) * 1997-07-25 2005-07-25 Gilead Sciences Inc Nukleotid-analog sammensætning og syntesemetode
ATE288914T1 (de) * 1997-07-25 2005-02-15 Gilead Sciences Inc Nukleotid-analog zusamensetzung und synthese verfahren
BR9911457A (pt) * 1998-06-24 2001-12-11 Univ Emory Uso de 3'-azida-2', 3'-dideoxiuridina em combinaçãocom drogas anti-hiv adicionais para a manufaturade um medicamento para o tratamento de hiv
AP1466A (en) * 2000-07-21 2005-09-22 Gilead Sciences Inc Prodrugs of phosphonate nucleotide analogues and methods for selecting and making same.
UA80819C2 (en) 2002-04-26 2007-11-12 Gilead Sciences Inc Phosphonate analogs of compounds inhibiting hiv proteases, pharmaceutical composition on their basis and their use
KR20090053867A (ko) 2003-01-14 2009-05-27 길리애드 사이언시즈, 인코포레이티드 복합 항바이러스 치료를 위한 조성물 및 방법
US7427636B2 (en) 2003-04-25 2008-09-23 Gilead Sciences, Inc. Inosine monophosphate dehydrogenase inhibitory phosphonate compounds
US7432261B2 (en) 2003-04-25 2008-10-07 Gilead Sciences, Inc. Anti-inflammatory phosphonate compounds
WO2005002626A2 (en) 2003-04-25 2005-01-13 Gilead Sciences, Inc. Therapeutic phosphonate compounds
AU2004233897A1 (en) * 2003-04-25 2004-11-11 Gilead Sciences, Inc. Kinase inhibitor phosphonate conjugates
US7407965B2 (en) 2003-04-25 2008-08-05 Gilead Sciences, Inc. Phosphonate analogs for treating metabolic diseases
CN101410120A (zh) * 2003-04-25 2009-04-15 吉里德科学公司 抗炎的膦酸酯化合物
SG182849A1 (en) 2003-04-25 2012-08-30 Gilead Sciences Inc Antiviral phosphonate analogs
US7452901B2 (en) 2003-04-25 2008-11-18 Gilead Sciences, Inc. Anti-cancer phosphonate analogs
US7470724B2 (en) 2003-04-25 2008-12-30 Gilead Sciences, Inc. Phosphonate compounds having immuno-modulatory activity
US7300924B2 (en) 2003-04-25 2007-11-27 Gilead Sciences, Inc. Anti-infective phosphonate analogs
EA011948B1 (ru) 2003-06-16 2009-06-30 Инститьют Оф Оргэник Кемистри Энд Байокемистри, Экэдеми Оф Сайэнс Оф Зе Чек Рипаблик Фосфонатзамещенные пиримидиновые соединения (варианты), способ их получения (варианты), фармацевтическая композиция на их основе и способ лечения вирусной инфекции
US7432273B2 (en) 2003-10-24 2008-10-07 Gilead Sciences, Inc. Phosphonate analogs of antimetabolites
JP2007508845A (ja) 2003-10-24 2007-04-12 ギリアード サイエンシーズ, インコーポレイテッド 治療用化合物の同定のための方法および組成物
WO2005044279A1 (en) 2003-10-24 2005-05-19 Gilead Sciences, Inc. Purine nucleoside phosphonate conjugates
EP1715871A1 (en) * 2003-12-22 2006-11-02 Gilead Sciences, Inc. Kinase inhibitor phosphonate conjugates
ATE424400T1 (de) 2003-12-22 2009-03-15 Gilead Sciences Inc 4'-substituierte carbovir- und abacavir-derivate sowie verwandte verbindungen mit hiv- und hcv- antiviraler wirkung
TR201906416T4 (tr) 2004-07-27 2019-05-21 Gilead Sciences Inc Hiv inhibitörü bileşiklerin fosfonat analogları.
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
JP5323476B2 (ja) * 2005-06-13 2013-10-23 博瑞生物医葯技▲術▼(▲蘇▼州)有限公司 ヌクレオチド類縁体プロドラッグおよびその製剤
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same
JP5291700B2 (ja) 2007-04-13 2013-09-18 サザン リサーチ インスティテュート 血管新生阻害薬及び使用方法
AU2008253803A1 (en) * 2007-05-22 2008-11-27 Ultimorphix Technolgies B.V. Tenofovir disoproxil hemi-fumaric acid Co-crystal
WO2009064174A1 (en) * 2007-11-14 2009-05-22 Ultimorphix Technologies B.V. Polymorphic form of tenofovir disoproxil fumarate, method for its preparation and use
NZ588796A (en) * 2008-04-25 2012-07-27 Cipla Ltd Crystalline form of tenofovir disoproxil and a process for its preparation
BRPI0915878A2 (pt) 2008-07-08 2015-11-03 Gilead Sciences Inc sais ou hidratos de compostos inibidores de hiv, seu uso e composição farmacêutica que os compreende
CN102093422B (zh) 2009-12-10 2015-02-25 中国人民解放军军事医学科学院毒物药物研究所 无环核苷膦酸酯衍生物及其医药用途
BR112013028698A8 (pt) * 2011-05-10 2018-04-03 Okapi Sciences Nv Compostos para uso no tratamento de infecções retrovirais em felinos
AU2012296622C1 (en) 2011-08-16 2017-02-16 Gilead Sciences, Inc. Tenofovir alafenamide hemifumarate
CN103626802A (zh) * 2012-08-23 2014-03-12 重庆药友制药有限责任公司 一种制备替诺福韦的新方法
CN107312039B (zh) 2012-08-30 2019-06-25 江苏豪森药业集团有限公司 一种替诺福韦前药的制备方法
JP2015536940A (ja) 2012-10-29 2015-12-24 シプラ・リミテッド 抗ウイルス性ホスホネート類似体及びその製造方法
EP2860185A1 (en) 2013-10-09 2015-04-15 Zentiva, k.s. An improved process for the preparation of Tenofovir disoproxil and pharmaceutically acceptable salts thereof
EP2860184B1 (en) 2013-10-09 2018-08-29 Zentiva, k.s. Dihydrogenphosphate salt of Tenofovir disoproxil
TWI660965B (zh) * 2014-01-15 2019-06-01 美商基利科學股份有限公司 泰諾福韋之固體形式
SI3661937T1 (sl) 2017-08-01 2021-11-30 Gilead Sciences, Inc. Kristalinične oblike etil((S)-((((2R,5R)-5-(6-amino-9H-purin-9-IL)-4- fluoro-2,5-dihidrofuran-2-IL)oksi)metil)(fenoksi)fosforil)-L-alaninata (GS-9131) za zdravljenje virusnih okužb
CN107805202A (zh) * 2017-12-01 2018-03-16 内蒙古圣氏化学股份有限公司 一种氯甲基异丙基碳酸酯连续化反应装置及方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL84477A (en) * 1986-11-18 1995-12-08 Bristol Myers Squibb Co History of Phosphonomethoxyalkylene Purinopyrimidine and Pharmaceutical Preparations Containing Them
ES2118069T3 (es) * 1990-09-14 1998-09-16 Acad Of Science Czech Republic Profarmacos de fosfonatos.
GB9026164D0 (en) * 1990-12-01 1991-01-16 Beecham Group Plc Pharmaceuticals
WO1995007920A1 (en) * 1993-09-17 1995-03-23 Gilead Sciences, Inc. Nucleotide analogs
WO1998004569A1 (en) * 1996-07-26 1998-02-05 Gilead Sciences, Inc. Nucleotide analogs

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