JP2000503304A5 - - Google Patents

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Publication number
JP2000503304A5
JP2000503304A5 JP1997525466A JP52546697A JP2000503304A5 JP 2000503304 A5 JP2000503304 A5 JP 2000503304A5 JP 1997525466 A JP1997525466 A JP 1997525466A JP 52546697 A JP52546697 A JP 52546697A JP 2000503304 A5 JP2000503304 A5 JP 2000503304A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1997525466A
Other languages
English (en)
Japanese (ja)
Other versions
JP2000503304A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/000619 external-priority patent/WO1997025048A1/en
Publication of JP2000503304A publication Critical patent/JP2000503304A/ja
Publication of JP2000503304A5 publication Critical patent/JP2000503304A5/ja
Ceased legal-status Critical Current

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JP9525466A 1996-01-11 1997-01-10 新規シクロアルキル置換イミダゾール Ceased JP2000503304A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1001096P 1996-01-11 1996-01-11
US60/010,010 1996-01-11
PCT/US1997/000619 WO1997025048A1 (en) 1996-01-11 1997-01-10 Novel cycloalkyl substituted imidazoles

Publications (2)

Publication Number Publication Date
JP2000503304A JP2000503304A (ja) 2000-03-21
JP2000503304A5 true JP2000503304A5 (cg-RX-API-DMAC10.html) 2004-11-11

Family

ID=21743297

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9525466A Ceased JP2000503304A (ja) 1996-01-11 1997-01-10 新規シクロアルキル置換イミダゾール

Country Status (24)

Country Link
US (1) US6329526B1 (cg-RX-API-DMAC10.html)
EP (1) EP0889726B1 (cg-RX-API-DMAC10.html)
JP (1) JP2000503304A (cg-RX-API-DMAC10.html)
CN (1) CN1213305A (cg-RX-API-DMAC10.html)
AP (1) AP9700912A0 (cg-RX-API-DMAC10.html)
AR (1) AR005434A1 (cg-RX-API-DMAC10.html)
AT (1) ATE276248T1 (cg-RX-API-DMAC10.html)
AU (1) AU715315B2 (cg-RX-API-DMAC10.html)
BR (1) BR9708149A (cg-RX-API-DMAC10.html)
CZ (1) CZ218198A3 (cg-RX-API-DMAC10.html)
DE (1) DE69730704T2 (cg-RX-API-DMAC10.html)
ES (1) ES2229335T3 (cg-RX-API-DMAC10.html)
HU (1) HUP9901233A2 (cg-RX-API-DMAC10.html)
ID (1) ID18759A (cg-RX-API-DMAC10.html)
IL (1) IL125224A0 (cg-RX-API-DMAC10.html)
MA (1) MA24055A1 (cg-RX-API-DMAC10.html)
MX (1) MX9805628A (cg-RX-API-DMAC10.html)
NO (1) NO983182L (cg-RX-API-DMAC10.html)
NZ (1) NZ330889A (cg-RX-API-DMAC10.html)
PL (1) PL327939A1 (cg-RX-API-DMAC10.html)
TR (1) TR199801350T2 (cg-RX-API-DMAC10.html)
UY (1) UY24434A1 (cg-RX-API-DMAC10.html)
WO (1) WO1997025048A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA97173B (cg-RX-API-DMAC10.html)

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US6096899A (en) * 1998-04-14 2000-08-01 The Regents Of The University Of Michigan Cylic imidazole compounds having relatively low hydrogen content and relatively high nitrogen content and polymers formed therefrom
GB9809869D0 (en) * 1998-05-09 1998-07-08 Medical Res Council Inhibition of protein kinases
CN1548436A (zh) 1998-05-22 2004-11-24 ʷ��˿�������ȳ�ķ���޹�˾ 新的2-烷基取代咪唑化合物
US6858617B2 (en) 1998-05-26 2005-02-22 Smithkline Beecham Corporation Substituted imidazole compounds
WO2000010563A1 (en) 1998-08-20 2000-03-02 Smithkline Beecham Corporation Novel substituted triazole compounds
ATE258055T1 (de) 1998-11-04 2004-02-15 Smithkline Beecham Corp Pyridin-4-yl oder pyrimidin-4-yl substituierte pyrazine
US6239279B1 (en) 1998-12-16 2001-05-29 Smithkline Beecham Corporation Synthesis for 4-aryl-5-pyrimidine imidazole substituted derivatives
US6930101B1 (en) 1999-05-17 2005-08-16 The Regents Of The University Of California Thiazolopyrimidines useful as TNFα inhibitors
EP1223924A4 (en) * 1999-09-17 2004-07-14 Smithkline Beecham Corp USE OF CSAIDS AGAINST RHINOVIRUS INFECTION
EP1233950B1 (en) 1999-11-23 2005-10-05 Smithkline Beecham Corporation 3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/P39 kINASE INHIBITORS
AU1783201A (en) 1999-11-23 2001-06-04 Smithkline Beecham Corporation 3,4-dihydro-(1h)quinazolin-2-one compounds as csbp/p38 kinase inhibitors
US6759410B1 (en) 1999-11-23 2004-07-06 Smithline Beecham Corporation 3,4-dihydro-(1H)-quinazolin-2-ones and their use as CSBP/p38 kinase inhibitors
PT1175214E (pt) 1999-12-08 2005-04-29 Pharmacia Corp Composicoes de inibidor de ciclo-oxigenase-2 com um inicio rapido do seu efito terapeutico
US7235551B2 (en) 2000-03-02 2007-06-26 Smithkline Beecham Corporation 1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
US6673818B2 (en) 2001-04-20 2004-01-06 Pharmacia Corporation Fluoro-substituted benzenesulfonyl compounds for the treatment of inflammation
US7473695B2 (en) * 2001-10-22 2009-01-06 Mitsubishi Tanabe Pharma Corporation 4-imidazolin-2-one compounds
JP2005538066A (ja) 2002-07-09 2005-12-15 ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト 新規な抗コリン作用薬及びp38キナーゼ阻害剤を用いた新規な医薬組成物
US20050004098A1 (en) * 2003-03-20 2005-01-06 Britten Nancy Jean Dispersible formulation of an anti-inflammatory agent
US20040214753A1 (en) * 2003-03-20 2004-10-28 Britten Nancy Jean Dispersible pharmaceutical composition for treatment of mastitis and otic disorders
DK1608407T3 (da) * 2003-03-20 2006-12-04 Pharmacia Corp Dispergébar formulering af et antiinflammatorisk middel
US20050009931A1 (en) * 2003-03-20 2005-01-13 Britten Nancy Jean Dispersible pharmaceutical composition for treatment of mastitis and otic disorders
US7105467B2 (en) * 2003-07-08 2006-09-12 Pharmacore, Inc. Nickel catalyzed cross-coupling reactions between organomagnesium compounds and anisole derivatives
US7105707B2 (en) * 2003-12-17 2006-09-12 Pharmacore, Inc. Process for preparing alkynyl-substituted aromatic and heterocyclic compounds
US20060035893A1 (en) 2004-08-07 2006-02-16 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
WO2006062069A1 (ja) * 2004-12-06 2006-06-15 Santen Pharmaceutical Co., Ltd. p38MAPキナーゼ阻害剤を有効成分とする掻痒治療剤
PE20060777A1 (es) 2004-12-24 2006-10-06 Boehringer Ingelheim Int Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas
JP2007145819A (ja) * 2005-10-28 2007-06-14 Tanabe Seiyaku Co Ltd 医薬組成物
WO2007056016A2 (en) * 2005-11-02 2007-05-18 Kemia, Inc. Bisamide cytokine inhibitors
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
EP2111861A1 (en) 2008-04-21 2009-10-28 Ranbaxy Laboratories Limited Compositions of phosphodiesterase type IV inhibitors
EP3553169B1 (en) 2011-12-28 2021-11-03 Kyoto Prefectural Public University Corporation Normalization of culture of corneal endothelial cells
JP6730701B2 (ja) 2013-11-14 2020-07-29 学校法人同志社 細胞増殖促進または細胞障害抑制による角膜内皮治療薬
US10342786B2 (en) 2017-10-05 2019-07-09 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD
RS63581B1 (sr) 2017-10-05 2022-10-31 Fulcrum Therapeutics Inc Inhibitori p38 kinaze smanjuju ekspresiju dux4 i nizvodnih gena u cilju lečenja fshd
WO2022195579A1 (en) 2021-03-15 2022-09-22 Saul Yedgar Hyaluronic acid-conjugated dipalmitoyl phosphatidyl ethanolamine in combination with non-steroidal anti-inflammatory drugs (nsaids) for treating or alleviating inflammatory diseases

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TR199801361T2 (xx) 1996-01-11 1998-10-21 Smithkline Beecham Corporation Yeni ikameli imidazol bile�imleri.
US6096739A (en) 1996-03-25 2000-08-01 Smithkline Beecham Corporation Treatment for CNS injuries
JP2000507545A (ja) 1996-03-25 2000-06-20 スミスクライン・ビーチャム・コーポレイション Cns損傷についての新規な治療
CA2271893A1 (en) 1996-11-20 1998-05-28 Linda L. Chang Triaryl substituted imidazoles as glucagon antagonists

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