IT8049899A0 - Composti diazepinici per uso farmaceutico e loro procedimento di preparazione - Google Patents

Composti diazepinici per uso farmaceutico e loro procedimento di preparazione

Info

Publication number
IT8049899A0
IT8049899A0 IT8049899A IT4989980A IT8049899A0 IT 8049899 A0 IT8049899 A0 IT 8049899A0 IT 8049899 A IT8049899 A IT 8049899A IT 4989980 A IT4989980 A IT 4989980A IT 8049899 A0 IT8049899 A0 IT 8049899A0
Authority
IT
Italy
Prior art keywords
pharmaceutical use
preparation procedure
diazepine compounds
diazepine
compounds
Prior art date
Application number
IT8049899A
Other languages
English (en)
Other versions
IT1143047B (it
Inventor
Jiban K Chakrabarti
Terrence M Hotten
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of IT8049899A0 publication Critical patent/IT8049899A0/it
Application granted granted Critical
Publication of IT1143047B publication Critical patent/IT1143047B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
IT49899/80A 1979-10-16 1980-10-14 Composti diazepinici per uso farmaceutico e loro procedimento di preparazione IT1143047B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7935846 1979-10-16

Publications (2)

Publication Number Publication Date
IT8049899A0 true IT8049899A0 (it) 1980-10-14
IT1143047B IT1143047B (it) 1986-10-22

Family

ID=10508540

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49899/80A IT1143047B (it) 1979-10-16 1980-10-14 Composti diazepinici per uso farmaceutico e loro procedimento di preparazione

Country Status (33)

Country Link
US (3) US4404137A (it)
EP (1) EP0027390B1 (it)
JP (1) JPS5663987A (it)
KR (2) KR850000471B1 (it)
AR (2) AR228041A1 (it)
AT (1) AT373889B (it)
AU (1) AU538500B2 (it)
BE (1) BE885729A (it)
BG (2) BG34907A3 (it)
CA (1) CA1159056A (it)
CH (1) CH646700A5 (it)
CS (1) CS244409B2 (it)
DD (1) DD153692A5 (it)
DE (1) DE3068706D1 (it)
DK (1) DK437480A (it)
ES (1) ES8106905A1 (it)
FI (1) FI67550C (it)
FR (1) FR2467851A1 (it)
GB (1) GB8327127D0 (it)
GR (1) GR70720B (it)
HU (1) HU182213B (it)
IE (1) IE50358B1 (it)
IL (1) IL61264A (it)
IT (1) IT1143047B (it)
LU (1) LU82853A1 (it)
MX (1) MX6233E (it)
NZ (1) NZ195248A (it)
PH (2) PH16288A (it)
PL (2) PL135044B1 (it)
PT (1) PT71913B (it)
RO (2) RO81351B (it)
YU (1) YU261580A (it)
ZA (1) ZA806342B (it)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4404137A (en) * 1979-10-16 1983-09-13 Lilly Industries Limited Pyrazolo [3,4-b][1,5]benzodiazepine compounds
US4431589A (en) * 1980-12-11 1984-02-14 Lilly House Benzodiazepine compounds and their use as pharmaceuticals
US4596799A (en) * 1985-01-29 1986-06-24 Ciba-Geigy Corporation 9H-pyrrolo[2,1-c]-1,2,4-triazolo[4,3-a][1,4]benzodiazepines
TW219896B (it) * 1988-07-07 1994-02-01 Duphar Int Res
GB8819059D0 (en) * 1988-08-11 1988-09-14 Lilly Industries Ltd Benzodiazepine compounds & their use as pharmaceuticals
US5637584A (en) * 1995-03-24 1997-06-10 Eli Lilly And Company Solvate of olanzapine
US5631250A (en) * 1995-03-24 1997-05-20 Eli Lilly And Company Process and solvate of 2-methyl-thieno-benzodiazepine
US20050085463A1 (en) * 2003-01-23 2005-04-21 Weiner David M. Use of N-desmethylclozapine to treat human neuropsychiatric disease
US20050250767A1 (en) * 2003-01-23 2005-11-10 Weiner David M Use of N-desmethylclozapine to treat human neuropsychiatric disease
JP2006515628A (ja) * 2003-01-23 2006-06-01 アカディア ファーマシューティカルズ，インコーポレーテッド ヒト神経精神疾患を処置するためのｎ−デスメチルクロザピンの使用
ES2324713T3 (es) * 2003-12-22 2009-08-13 Acadia Pharmaceuticals Inc. Analogos de diaril(a,d)ciclohepteno amino-sustituidos como agonistas muscarinicos y metodos de tratamiento de trastornos neuropsiquiatricos.
CN1950346A (zh) * 2004-04-01 2007-04-18 阿卡蒂亚药品公司 N－去甲基氯氮平的晶形
WO2007053618A1 (en) * 2005-10-31 2007-05-10 Acadia Pharmaceuticals Inc. Prodrugs of muscarinic agonists and methods of treatment of neuropsychiatric disorders
JP5438482B2 (ja) * 2009-12-03 2014-03-12 Ｊｕｋｉ株式会社 ミシン、ミシンの縫製データ編集装置及びミシンの縫製データ編集プログラム

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3450694A (en) * 1966-02-23 1969-06-17 Abbott Lab Substituted benzoxazepines and benzothiazepines
US3758479A (en) * 1967-03-22 1973-09-11 Sandoz Ag Nitro and sulphamoyl substituted dibenzodiazepines
DE1795183B1 (de) * 1968-08-20 1972-07-20 Thomae Gmbh Dr K 5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-on-derivate und Arzneimittel
CA918659A (en) * 1969-07-31 1973-01-09 Yoshitomi Pharmaceutical Industries 11-(4-substituted-1-piperazinyl)-dibenzo (b,f) (1,4) thiazepines
US4115568A (en) * 1974-11-26 1978-09-19 Lilly Industries Limited Thieno[3,2-b]-[1,5]benzodiazepines
US4172831A (en) * 1974-11-26 1979-10-30 Lilly Industries Limited Thieno-benzodiazepines
US3953430A (en) * 1975-02-24 1976-04-27 American Cyanamid Company Substituted benzodiazepin-10-ones and method of use
US3951981A (en) * 1975-02-24 1976-04-20 American Cyanamid Company Substituted benzodiazepines and method of use
DE2707270A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Pyrazolo-diazepine und verfahren zu ihrer herstellung
DE2707269A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
US4097597A (en) * 1977-02-23 1978-06-27 Abbott Laboratories Dibenzo b,e! 1,4!diazepines
IT7851496A0 (it) * 1977-10-31 1978-10-13 Sandoz Ag Menti pirazinobenzossazepine loro preparazione e loro impiego quali medica
CH643263A5 (de) * 1979-05-11 1984-05-30 Sandoz Ag Benzodiazepine, ihre herstellung und verwendung.
NO802326L (no) * 1979-08-03 1981-02-04 Byk Gulden Lomberg Chem Fab Fremgangsmaate ved fremstilling av substituerte tetraazatricyklen
US4404137A (en) * 1979-10-16 1983-09-13 Lilly Industries Limited Pyrazolo [3,4-b][1,5]benzodiazepine compounds

Also Published As

Publication number Publication date
FI67550B (fi) 1984-12-31
FR2467851B1 (it) 1985-04-05
PL126824B1 (en) 1983-09-30
EP0027390B1 (en) 1984-07-25
RO81351A (ro) 1983-02-15
RO85822A (ro) 1984-11-25
FI67550C (fi) 1985-04-10
IL61264A0 (en) 1980-12-31
US4486591A (en) 1984-12-04
AU538500B2 (en) 1984-08-16
IT1143047B (it) 1986-10-22
GR70720B (it) 1983-01-18
DE3068706D1 (en) 1984-08-30
KR850001463A (ko) 1985-03-18
DK437480A (da) 1981-04-17
KR850000471B1 (ko) 1985-04-08
YU261580A (en) 1983-12-31
CH646700A5 (fr) 1984-12-14
BG35042A3 (en) 1983-01-16
PL227306A1 (it) 1981-09-18
JPS5663987A (en) 1981-05-30
KR850000472B1 (ko) 1985-04-08
RO85822B (ro) 1984-11-30
PH17759A (en) 1984-12-05
ATA510180A (de) 1983-07-15
MX6233E (es) 1985-01-14
KR830004300A (ko) 1983-07-09
AR228041A1 (es) 1983-01-14
PT71913A (en) 1980-11-01
CS244409B2 (en) 1986-07-17
PL231270A1 (it) 1981-12-23
PH16288A (en) 1983-09-05
IL61264A (en) 1985-08-30
EP0027390A1 (en) 1981-04-22
ES495948A0 (es) 1981-09-16
PT71913B (en) 1981-08-31
RO81351B (ro) 1983-02-28
US4404137A (en) 1983-09-13
HU182213B (en) 1983-12-28
AU6325280A (en) 1981-04-30
IE50358B1 (en) 1986-04-02
PL135044B1 (en) 1985-09-30
ZA806342B (en) 1982-05-26
CA1159056A (en) 1983-12-20
IE802135L (en) 1981-04-16
NZ195248A (en) 1983-11-18
US4542131A (en) 1985-09-17
FI803253L (fi) 1981-04-17
AT373889B (de) 1984-02-27
LU82853A1 (fr) 1982-05-10
GB8327127D0 (en) 1983-11-09
FR2467851A1 (fr) 1981-04-30
ES8106905A1 (es) 1981-09-16
BG34907A3 (en) 1983-12-15
AR228101A1 (es) 1983-01-14
DD153692A5 (de) 1982-01-27
BE885729A (fr) 1981-04-15

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