IT1171477B - Derivati del 4h-1,2,4-triazolo procedimento per la loro preparazione, loro impiego in quanto farmaci, composizioni che li contengono e prodotti intermedi ottenuti - Google Patents

Derivati del 4h-1,2,4-triazolo procedimento per la loro preparazione, loro impiego in quanto farmaci, composizioni che li contengono e prodotti intermedi ottenuti

Info

Publication number
IT1171477B
IT1171477B IT49147/81A IT4914781A IT1171477B IT 1171477 B IT1171477 B IT 1171477B IT 49147/81 A IT49147/81 A IT 49147/81A IT 4914781 A IT4914781 A IT 4914781A IT 1171477 B IT1171477 B IT 1171477B
Authority
IT
Italy
Prior art keywords
triazole
drugs
derivatives
procedure
preparation
Prior art date
Application number
IT49147/81A
Other languages
English (en)
Italian (it)
Other versions
IT8149147A0 (it
Inventor
Jean Meier
Francois Clemence
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IT8149147A0 publication Critical patent/IT8149147A0/it
Application granted granted Critical
Publication of IT1171477B publication Critical patent/IT1171477B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C243/24—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids
    • C07C243/38—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT49147/81A 1980-08-22 1981-08-21 Derivati del 4h-1,2,4-triazolo procedimento per la loro preparazione, loro impiego in quanto farmaci, composizioni che li contengono e prodotti intermedi ottenuti IT1171477B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8018354A FR2488891A1 (fr) 1980-08-22 1980-08-22 Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament

Publications (2)

Publication Number Publication Date
IT8149147A0 IT8149147A0 (it) 1981-08-21
IT1171477B true IT1171477B (it) 1987-06-10

Family

ID=9245357

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49147/81A IT1171477B (it) 1980-08-22 1981-08-21 Derivati del 4h-1,2,4-triazolo procedimento per la loro preparazione, loro impiego in quanto farmaci, composizioni che li contengono e prodotti intermedi ottenuti

Country Status (24)

Country Link
US (3) US4512997A (en17)
JP (1) JPS5770875A (en17)
AT (1) AT378957B (en17)
AU (1) AU543946B2 (en17)
BE (1) BE890035A (en17)
CA (1) CA1208226A (en17)
CH (1) CH649994A5 (en17)
DE (1) DE3133185A1 (en17)
DK (1) DK370781A (en17)
ES (2) ES504887A0 (en17)
FI (1) FI72971C (en17)
FR (1) FR2488891A1 (en17)
GB (1) GB2082581B (en17)
GR (1) GR75329B (en17)
HU (1) HU185647B (en17)
IE (1) IE51510B1 (en17)
IT (1) IT1171477B (en17)
LU (1) LU83576A1 (en17)
NL (1) NL8103903A (en17)
OA (2) OA06889A (en17)
PH (2) PH19890A (en17)
PT (1) PT73544B (en17)
SE (1) SE454173B (en17)
ZA (1) ZA815689B (en17)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2488891A1 (fr) * 1980-08-22 1982-02-26 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament
FR2539127B1 (fr) * 1983-01-10 1985-08-23 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicaments
FR2570699B1 (fr) * 1984-09-24 1987-08-28 Roussel Uclaf Nouveau procede de preparation de derives du 4h-1,2,4-triazole, nouveaux triazoles ainsi obtenus, leur application comme medicaments et les compositions pharmaceutiques les renfermant
US5278180A (en) * 1984-09-24 1994-01-11 Roussel Uclaf 4,5-bis(aryl) 4H-1,2,4-triazoles derivatives and analgesic use
RU2124010C1 (ru) * 1991-09-02 1998-12-27 Яманучи Фармасетикал Ко., Лтд. Триазолилзамещенное соединение третичного амина и фармацевтическая композиция
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
RU2131411C1 (ru) * 1997-11-20 1999-06-10 Институт химической физики РАН в Черноголовке Способ получения смеси олиготрифениламинов, способ получения 3-(4-бифенилил)-4- (4-трет-бутилфенил)-5-(4-диметиламинофенил)-1,2,4-триазола и электролюминесцентное устройство
US6362342B1 (en) * 1999-06-29 2002-03-26 Lion Bioscience Ag Triazole compounds and methods of making same
US6770621B2 (en) 2000-05-02 2004-08-03 Theravance, Inc. Polyacid glycopeptide derivatives
AU2003210916B9 (en) * 2002-02-07 2008-12-18 The Curators Of The University Of Missouri Opioid receptor active 4-(3-hydroxyphenyl) or 4-(3-alkoxyphenyl)-1,2,4-triazole compounds
KR102780240B1 (ko) 2017-04-26 2025-03-14 오티아이 루미오닉스 인크. 표면의 코팅을 패턴화하는 방법 및 패턴화된 코팅을 포함하는 장치
US11751415B2 (en) 2018-02-02 2023-09-05 Oti Lumionics Inc. Materials for forming a nucleation-inhibiting coating and devices incorporating same
US11730012B2 (en) 2019-03-07 2023-08-15 Oti Lumionics Inc. Materials for forming a nucleation-inhibiting coating and devices incorporating same
US12101987B2 (en) 2019-04-18 2024-09-24 Oti Lumionics Inc. Materials for forming a nucleation-inhibiting coating and devices incorporating same
JP7576337B2 (ja) 2019-05-08 2024-11-01 オーティーアイ ルミオニクス インコーポレーテッド 核生成抑制コーティングを形成するための材料およびそれを組み込んだデバイス

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1796403A (en) * 1931-03-17 Schaft
US3681374A (en) * 1970-08-11 1972-08-01 Asahi Chemical Ind Synthetic nacreous triazole crystals and method for production thereof
SU508198A3 (ru) * 1971-07-22 1976-03-25 Группо Лепетит С.П.А. (Фирма) Способ получени производных 1,2,4-триазола
AU7528974A (en) * 1973-11-13 1976-06-10 Commonwealth Scientific And Industrial Research Organization Triazoles
FR2269938A2 (en) * 1974-05-08 1975-12-05 Delalande Sa 5-Hydroxymethyl-3,4-diphenyl-1,2,4-triazoles - with anticholinergic, bronchodilator, antidepressant, analgesic, vasodilator activity, etc.
JPS56125376A (en) * 1980-03-07 1981-10-01 Mitsubishi Chem Ind Ltd Triazole derivative
FR2488891A1 (fr) * 1980-08-22 1982-02-26 Roussel Uclaf Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament

Also Published As

Publication number Publication date
PH21567A (en) 1987-12-11
US4512997A (en) 1985-04-23
HU185647B (en) 1985-03-28
ATA368281A (de) 1985-03-15
FI72971B (fi) 1987-04-30
PH19890A (en) 1986-08-13
CA1208226A (fr) 1986-07-22
OA07537A (fr) 1985-03-31
US4727084A (en) 1988-02-23
GB2082581A (en) 1982-03-10
AT378957B (de) 1985-10-25
US4659729A (en) 1987-04-21
IE811923L (en) 1982-02-22
LU83576A1 (fr) 1982-04-14
IT8149147A0 (it) 1981-08-21
GR75329B (en17) 1984-07-13
FR2488891B1 (en17) 1983-06-17
ES8306730A1 (es) 1983-06-01
ZA815689B (en) 1982-08-25
JPH0261463B2 (en17) 1990-12-20
OA06889A (fr) 1983-04-30
SE8104515L (sv) 1982-02-23
ES504887A0 (es) 1983-06-01
ES515419A0 (es) 1983-06-16
NL8103903A (nl) 1982-03-16
PT73544B (fr) 1983-07-14
BE890035A (fr) 1982-02-22
FR2488891A1 (fr) 1982-02-26
GB2082581B (en) 1985-02-13
DE3133185A1 (de) 1982-04-08
PT73544A (fr) 1981-09-01
ES8307227A1 (es) 1983-06-16
FI72971C (fi) 1987-08-10
AU543946B2 (en) 1985-05-09
FI812585L (fi) 1982-02-23
IE51510B1 (en) 1987-01-07
JPS5770875A (en) 1982-05-01
SE454173B (sv) 1988-04-11
CH649994A5 (fr) 1985-06-28
DK370781A (da) 1982-02-23
AU7442681A (en) 1982-02-25

Similar Documents

Publication Publication Date Title
IT8347820A0 (it) Derivati di 3-cheto delta 4,9 19nor-steroidi,procedimento per la loro preparazione,loro impiego come medicamenti,composizioni che li con tengono ed intermedi ottenuti
IT1171477B (it) Derivati del 4h-1,2,4-triazolo procedimento per la loro preparazione, loro impiego in quanto farmaci, composizioni che li contengono e prodotti intermedi ottenuti
IT1170286B (it) Derivati del labdano, procedimento per la loro preparazione, e composizioni farmaceutiche contenenti derivati del labdano
IL57178A0 (en) 1,3,4-triazole derivatives their preparation and pharmaceutical compositions containing them
IL58775A0 (en) Hydroxyethyl-azole compounds,their production and pharmaceutical compositions containing them
DE3160616D1 (en) Polyether compounds and their manufacture, resultant composition and the use of these products as medicaments or growth promoting agents in ruminants
IL69825A0 (en) Triazole derivatives,pharmaceutical compositions containing them and their use as fungicides
ZA80234B (en) New heterotricyclic derivatives, process for their preparation, their use as medicaments and the pharmaceutical compositions incorporating them
DE3166084D1 (en) Tricyclic cytosine derivatives for use in pharmaceutical preparations and process for their preparation
IT7967043A0 (it) Derivati di aza i biciclo 2 2 2 octano prodotti intermedi procedimento per la loro preparazione e loro applicazione come medicinali
DE3063905D1 (en) Compounds having antitumour properties, process for their preparation, these compounds for use as antitumour agents and pharmaceutical compositions containing them
ES478048A1 (es) Procedimiento para la obtencion de difenil-imidazolil-meta- nos sustituidos.
IT1196411B (it) Derivati ergolinici,loro preparazione e composizioni terapeutiche che li contengono
IT7948011A0 (it) Procedimento per la preparazione di derivati di 2-fenilimminoimidazolidine composizioni farmaceutiche che li contengono e prodotto ottenuto
IL62229A (en) 3-substituted-5-amino-1,2,4-triazole derivatives,their preparation and pharmaceutical compositions containing them
JPS55105654A (en) Novel dehydropeptide compounds*their manufacture and their medical use
BE884353A (fr) Nouveaux derives 1-substitues de 3-cycloalcoyl-sulfonyl-pyrrolidine-2, 5-diones, compositions fongicides les contenant et procede pour la preparation des ingredients actifs
IT1228130B (it) Derivati dell'1,1,2-trifenilpropano e dell'1,1,2-trifenilpropene, procedimento per la loro preparazione e composizioni farmaceutiche contenenti i composti
DE2966639D1 (en) Benzodiazepine derivatives, process for their preparation and pharmaceutical compositions containing them
DE2960227D1 (en) Dichlorobenzodioxole derivatives, process for their preparation and their use as synergetic agents in insecticidal and acaricidal compositions
IT8022601A0 (it) Derivati 3h-naft[1.2-d]-imidazolici il procedimento per la loro preparazione,il loro uso come agenti antiinfiammatori e le composizioni farmaceutiche che li contengono
IT1168171B (it) Derivati del 2-idrossimetil-chinossalin-1,4-biossido, procedimento per la loro preparazione e composizioni contenenti gli stessi
IL56617A0 (en) Benzimidazole derivatives,their manufacture and pharmaceutical compositions containing
IT8123055A1 (it) Derivati del piridazino/4,5-b /chinossalin-5,10-biossido, procedimento per prepararli e composizioni che li contengono
DE2965098D1 (en) 1.2.4-triazolidine-3.5-dione derivatives, process for their preparation and pharmaceutical compositions containing them