IS6304A - Kínasólínefnasambönd og lyfjafræðilegar efnasamsetningar sem innihalda þau - Google Patents

Kínasólínefnasambönd og lyfjafræðilegar efnasamsetningar sem innihalda þau

Info

Publication number
IS6304A
IS6304A IS6304A IS6304A IS6304A IS 6304 A IS6304 A IS 6304A IS 6304 A IS6304 A IS 6304A IS 6304 A IS6304 A IS 6304A IS 6304 A IS6304 A IS 6304A
Authority
IS
Iceland
Prior art keywords
pharmaceutical compositions
compositions containing
quinazoline compounds
quinazoline
compounds
Prior art date
Application number
IS6304A
Other languages
English (en)
Inventor
Austen Mortlock Andrew
John Keen Nicholas
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9922156.6A external-priority patent/GB9922156D0/en
Priority claimed from GBGB9922152.5A external-priority patent/GB9922152D0/en
Priority claimed from GBGB9922159.0A external-priority patent/GB9922159D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IS6304A publication Critical patent/IS6304A/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/582Recycling of unreacted starting or intermediate materials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IS6304A 1999-09-21 2002-03-18 Kínasólínefnasambönd og lyfjafræðilegar efnasamsetningar sem innihalda þau IS6304A (is)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9922156.6A GB9922156D0 (en) 1999-09-21 1999-09-21 Chemical compounds
GBGB9922152.5A GB9922152D0 (en) 1999-09-21 1999-09-21 Chemical compounds
GBGB9922159.0A GB9922159D0 (en) 1999-09-21 1999-09-21 Chemical compounds
PCT/GB2000/003556 WO2001021594A1 (en) 1999-09-21 2000-09-18 Quinazoline compounds and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
IS6304A true IS6304A (is) 2002-03-18

Family

ID=27269803

Family Applications (1)

Application Number Title Priority Date Filing Date
IS6304A IS6304A (is) 1999-09-21 2002-03-18 Kínasólínefnasambönd og lyfjafræðilegar efnasamsetningar sem innihalda þau

Country Status (20)

Country Link
US (1) US7081461B1 (is)
EP (1) EP1218356A1 (is)
JP (1) JP2003509497A (is)
KR (1) KR20020032608A (is)
CN (1) CN1391561A (is)
AU (1) AU763242B2 (is)
BG (1) BG106491A (is)
BR (1) BR0014133A (is)
CA (1) CA2384282A1 (is)
CZ (1) CZ20021010A3 (is)
EE (1) EE200200149A (is)
HK (1) HK1046688A1 (is)
HU (1) HUP0204413A3 (is)
IL (1) IL148489A0 (is)
IS (1) IS6304A (is)
NO (1) NO20021401L (is)
PL (1) PL354923A1 (is)
SK (1) SK3832002A3 (is)
TR (1) TR200200749T2 (is)
WO (1) WO2001021594A1 (is)

Families Citing this family (65)

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SK2142003A3 (en) 2000-08-21 2003-07-01 Astrazeneca Ab Quinazoline derivatives, process for their preparation, pharmaceutical composition comprising same and their use
US6939866B2 (en) 2000-10-13 2005-09-06 Astrazeneca Ab Quinazoline derivatives
WO2002030924A1 (en) 2000-10-13 2002-04-18 Astrazeneca Ab Quinazoline derivatives with anti-tumour activity
WO2002036587A2 (en) 2000-11-01 2002-05-10 Cor Therapeutics, Inc. Process for the production of 4-quinazolinylpiperazin-1-carboxylic acid phenylamides
DE60229046D1 (de) 2001-04-19 2008-11-06 Astrazeneca Ab Chinazolin derivate
EP1408980A4 (en) 2001-06-21 2004-10-20 Ariad Pharma Inc NEW QUINAZOLINES AND THEIR USE
EP1447405A4 (en) 2001-10-17 2005-01-12 Kirin Brewery QUINOLINE OR QUINAZOLINE DERIVATIVES INHIBITING THE AUTOPHOSPHORYLATION OF FIBROBLAST GROWTH FACTOR RECEPTORS
WO2003044176A2 (en) * 2001-11-19 2003-05-30 Interleukin Genetics, Inc. Functional polymorphisms of the interleukin-1 locus affecting transcription and susceptibility to inflammatory and infectious diseases
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ATE429230T1 (de) * 2002-07-09 2009-05-15 Astrazeneca Ab Chinazoline derivative und ihre anwendung in der krebsbehandlung
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CA2592900A1 (en) 2005-01-03 2006-07-13 Myriad Genetics Inc. Nitrogen containing bicyclic compounds and therapeutical use thereof
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JO2787B1 (en) 2005-04-27 2014-03-15 امجين إنك, Alternative amide derivatives and methods of use
GB0509224D0 (en) * 2005-05-05 2005-06-15 Chroma Therapeutics Ltd Inhibitors of intracellular enzymatic activity
US7732613B2 (en) 2005-09-14 2010-06-08 Bristol-Myers Squibb Company Met kinase inhibitors
US8119655B2 (en) 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors
US7977359B2 (en) 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
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US8648087B2 (en) 2005-11-15 2014-02-11 Array Biopharma, Inc. N4-phenyl-quinazoline-4-amine derivatives and related compounds as ErbB type I receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases
CN101003514A (zh) * 2006-01-20 2007-07-25 上海艾力斯医药科技有限公司 喹唑啉衍生物、其制备方法及用途
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US8088782B2 (en) 2008-05-13 2012-01-03 Astrazeneca Ab Crystalline 4-(3-chloro-2-fluoroanilino)-7 methoxy-6-{[1-(N-methylcarbamoylmethyl)piperidin-4-yl]oxy}quinazoline difumarate form A
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CN101857588B (zh) * 2010-06-08 2013-11-27 东南大学 4-芳香胺基喹唑啉类衍生物及其用途
CN102850280B (zh) * 2011-06-30 2015-06-10 陕西师范大学 6,7-二烷氧基-4-取代苯基氨基喹唑啉类化合物及其制备方法
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Also Published As

Publication number Publication date
CA2384282A1 (en) 2001-03-29
HUP0204413A2 (en) 2003-05-28
AU7432500A (en) 2001-04-24
TR200200749T2 (tr) 2002-06-21
JP2003509497A (ja) 2003-03-11
BG106491A (bg) 2002-12-29
BR0014133A (pt) 2002-06-11
PL354923A1 (en) 2004-03-22
HUP0204413A3 (en) 2003-07-28
US7081461B1 (en) 2006-07-25
AU763242B2 (en) 2003-07-17
CZ20021010A3 (cs) 2002-06-12
CN1391561A (zh) 2003-01-15
NO20021401D0 (no) 2002-03-20
SK3832002A3 (en) 2002-11-06
EE200200149A (et) 2003-04-15
IL148489A0 (en) 2002-09-12
HK1046688A1 (zh) 2003-01-24
KR20020032608A (ko) 2002-05-03
EP1218356A1 (en) 2002-07-03
NO20021401L (no) 2002-05-21
WO2001021594A1 (en) 2001-03-29

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