IN2014DN04588A - - Google Patents

Info

Publication number
IN2014DN04588A
IN2014DN04588A IN4588DEN2014A IN2014DN04588A IN 2014DN04588 A IN2014DN04588 A IN 2014DN04588A IN 4588DEN2014 A IN4588DEN2014 A IN 4588DEN2014A IN 2014DN04588 A IN2014DN04588 A IN 2014DN04588A
Authority
IN
India
Prior art keywords
4alkyl
salt
compound
formula
Prior art date
Application number
Other languages
English (en)
Inventor
Philippe Robert Schils Didier
Elisabeth Stappers Alfred
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35822492&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014DN04588(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of IN2014DN04588A publication Critical patent/IN2014DN04588A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IN4588DEN2014 2005-05-26 2006-05-24 IN2014DN04588A (en17)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05104531 2005-05-26
US68599305P 2005-05-31 2005-05-31
PCT/EP2006/062606 WO2006125809A1 (en) 2005-05-26 2006-05-24 Process for preparing 4-[(1,6-dihydro-6-oxo-2-pyrimidinyl)amino benzonitrile

Publications (1)

Publication Number Publication Date
IN2014DN04588A true IN2014DN04588A (en17) 2015-07-10

Family

ID=35822492

Family Applications (1)

Application Number Title Priority Date Filing Date
IN4588DEN2014 IN2014DN04588A (en17) 2005-05-26 2006-05-24

Country Status (19)

Country Link
US (2) US8101752B2 (en17)
EP (1) EP1888537B1 (en17)
JP (2) JP5148483B2 (en17)
CN (1) CN101248051B (en17)
AU (1) AU2006251163C1 (en17)
BR (1) BRPI0611038B8 (en17)
CA (1) CA2609716C (en17)
DK (1) DK1888537T3 (en17)
ES (1) ES2437202T3 (en17)
HR (1) HRP20131133T1 (en17)
IN (1) IN2014DN04588A (en17)
ME (1) ME01612B (en17)
MX (1) MX2007014881A (en17)
PL (1) PL1888537T3 (en17)
PT (1) PT1888537E (en17)
RS (1) RS53062B (en17)
RU (1) RU2458056C2 (en17)
SI (1) SI1888537T1 (en17)
WO (1) WO2006125809A1 (en17)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006125809A1 (en) * 2005-05-26 2006-11-30 Tibotec Pharmaceuticals Ltd Process for preparing 4-[(1,6-dihydro-6-oxo-2-pyrimidinyl)amino benzonitrile
WO2012125993A1 (en) 2011-03-17 2012-09-20 Teva Pharmaceutical Industries Ltd. Solid state forms of rilpivirine base, and rilipivirine salts
WO2013135684A1 (en) 2012-03-13 2013-09-19 Octapharma Ag Improved process for production of fibrinogen and fibrinogen produced thereby
CN103058936B (zh) * 2013-01-23 2016-01-06 宁波九胜创新医药科技有限公司 4-[(4-氯-2-嘧啶基)氨基]苯腈的制备方法
CN103193719B (zh) * 2013-04-08 2015-07-22 宁波九胜创新医药科技有限公司 一种4-[(4-羟基-2-嘧啶基)氨基]苯腈的制备方法
CN114933567B (zh) * 2022-04-29 2023-07-11 武汉工程大学 一种2-甲硫基-4-嘧啶酮的制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE63502B1 (en) 1989-04-21 1995-05-03 Zeneca Ltd Aminopyrimidine derivatives useful for treating cardiovascular disorders
RU2037483C1 (ru) * 1989-07-20 1995-06-19 Мерк Патент Гмбх Способ получения замещенных ароматических нитрилов
DE3923979A1 (de) 1989-07-20 1991-01-24 Merck Patent Gmbh Verfahren zur herstellung von aromatischen nitrilen
WO1999050250A1 (en) * 1998-03-27 1999-10-07 Janssen Pharmaceutica N.V. Hiv inhibiting pyrimidine derivatives
EE05086B1 (et) * 1998-11-10 2008-10-15 Janssen Pharmaceutica N.V. Primidiini derivaadid, nende valmistamismeetod ja kasutamine, farmatseutiline kompositsioon ja selle valmistamismeetod, kombinatsioon ning saadus
BRPI0014271B1 (pt) * 1999-09-24 2021-06-22 Janssen Pharmaceutica N.V. Partícula consistindo em uma dispersão de sólidos, uso da dita partícula, dispersão de sólidos, forma de dosagem farmacêutica, bem como processos de preparação de dita partícula, dispersão e forma de dosagem
EP1282607B1 (en) * 2000-05-08 2015-11-11 Janssen Pharmaceutica NV Prodrugs of hiv replication inhibiting pyrimidines
JO3429B1 (ar) * 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv مشتقات برميدينات مثبطة فيروس الايدز
MXPA04004178A (es) * 2001-11-01 2004-09-06 Janssen Pharmaceutica Nv Heteroarilaminas como inhibidores de glucogeno cintasa cinasa 3beta.
AU2003266413B2 (en) * 2002-08-09 2009-04-02 Janssen Pharmaceutica N.V. Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile
AU2004286933B2 (en) * 2003-09-30 2010-11-18 Janssen Pharmaceutica N.V. Benzoimidazole compounds
WO2006125809A1 (en) * 2005-05-26 2006-11-30 Tibotec Pharmaceuticals Ltd Process for preparing 4-[(1,6-dihydro-6-oxo-2-pyrimidinyl)amino benzonitrile

Also Published As

Publication number Publication date
CN101248051B (zh) 2013-07-17
US8101752B2 (en) 2012-01-24
EP1888537B1 (en) 2013-09-11
DK1888537T3 (da) 2013-12-09
HK1123551A1 (en) 2009-06-19
WO2006125809A1 (en) 2006-11-30
AU2006251163B2 (en) 2012-03-08
RS53062B (en) 2014-04-30
JP2008545680A (ja) 2008-12-18
RU2007148968A (ru) 2009-07-10
US20120083606A1 (en) 2012-04-05
HRP20131133T1 (hr) 2014-01-03
US20080171878A1 (en) 2008-07-17
US8618291B2 (en) 2013-12-31
ES2437202T3 (es) 2014-01-09
BRPI0611038B8 (pt) 2022-10-25
RU2458056C2 (ru) 2012-08-10
BRPI0611038B1 (pt) 2022-02-08
ME01612B (me) 2014-09-20
JP2013040194A (ja) 2013-02-28
CN101248051A (zh) 2008-08-20
AU2006251163A1 (en) 2006-11-30
EP1888537A1 (en) 2008-02-20
PT1888537E (pt) 2013-11-26
JP5148483B2 (ja) 2013-02-20
CA2609716C (en) 2014-10-14
SI1888537T1 (sl) 2014-01-31
BRPI0611038A2 (pt) 2010-08-10
CA2609716A1 (en) 2006-11-30
MX2007014881A (es) 2008-02-15
JP5580385B2 (ja) 2014-08-27
AU2006251163C1 (en) 2012-07-12
PL1888537T3 (pl) 2014-02-28

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