IN2006DE01793A - - Google Patents
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- Publication number
- IN2006DE01793A IN2006DE01793A IN1793DE2006A IN2006DE01793A IN 2006DE01793 A IN2006DE01793 A IN 2006DE01793A IN 1793DE2006 A IN1793DE2006 A IN 1793DE2006A IN 2006DE01793 A IN2006DE01793 A IN 2006DE01793A
- Authority
- IN
- India
- Prior art keywords
- sup
- formula
- preparing
- esters
- dihalomethylpyrazoles
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/30—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10349500A DE10349500A1 (de) | 2003-10-23 | 2003-10-23 | Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2006DE01793A true IN2006DE01793A (zh) | 2007-08-10 |
Family
ID=34529740
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN1793DE2006 IN2006DE01793A (zh) | 2003-10-23 | 2006-04-03 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US7358387B2 (zh) |
| EP (1) | EP1678119B1 (zh) |
| JP (1) | JP4725977B2 (zh) |
| KR (1) | KR101116686B1 (zh) |
| CN (1) | CN100422141C (zh) |
| AT (1) | ATE494274T1 (zh) |
| BR (1) | BRPI0415855B1 (zh) |
| DE (2) | DE10349500A1 (zh) |
| DK (1) | DK1678119T3 (zh) |
| IL (1) | IL175024A (zh) |
| IN (1) | IN2006DE01793A (zh) |
| MX (1) | MXPA06004339A (zh) |
| TW (1) | TWI363050B (zh) |
| WO (1) | WO2005042468A1 (zh) |
Families Citing this family (61)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10352082A1 (de) * | 2003-10-23 | 2005-05-25 | Bayer Cropscience Ag | Hexylcarboxanilide |
| DE102006039909A1 (de) * | 2006-08-25 | 2008-03-13 | Bayer Cropscience Ag | Verfahren zum Herstellen von 3-Dihalomethyl-pyrazol-4-carbonsäurederivaten |
| US20100010216A1 (en) * | 2006-12-28 | 2010-01-14 | Mitsui Chemicals Agro, Inc | 2-fluorinated acyl-3-aminoacrylonitrile derivative and method for producing the same |
| EP1997808A1 (en) * | 2007-05-31 | 2008-12-03 | Syngeta Participations AG | Process for the production of pyrazoles |
| EP2150536A1 (en) * | 2007-05-31 | 2010-02-10 | Syngeta Participations AG | Process for the production of pyrazoles |
| EP2164831B1 (de) | 2007-06-01 | 2013-07-17 | Basf Se | Verfahren zur herstellung n-substituierter (3-dihalomethyl-1-methyl-pyrazol-4-yl)carboxamide |
| ES2369215T3 (es) * | 2007-06-15 | 2011-11-28 | Basf Se | Procedimiento para la obtención de compuestos de pirazol substituidos con difluormetilo. |
| EP2008996A1 (en) * | 2007-06-27 | 2008-12-31 | Syngeta Participations AG | Process for the production of pyrazoles |
| EP2042482A1 (de) * | 2007-09-26 | 2009-04-01 | Bayer CropScience AG | Verfahren zur Herstellung von 2-Dihalogenacyl-3-amino-acrylsäure-Derivaten |
| EP2072497A1 (de) | 2007-12-21 | 2009-06-24 | Bayer CropScience AG | Verfahren zum Herstellen von 2-Fluoracyl-3-amino-acrylsäure-Derivaten |
| EP2133341A1 (de) * | 2008-02-25 | 2009-12-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten |
| EP2100883A1 (de) * | 2008-03-10 | 2009-09-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten |
| US8344156B2 (en) | 2008-03-18 | 2013-01-01 | Mitsui Chemicals Agro, Inc. | Method for producing fluorine-containing acylacetic acid derivative, method for producing fluorine-containing pyrazolecarboxylic acid ester derivative, and method for producing fluorine-containing pyrazolecarboxylic acid derivative |
| JP2009227643A (ja) * | 2008-03-25 | 2009-10-08 | Mitsui Chemicals Agro Inc | 含フッ素アルキルカルボン酸誘導体を利用した含フッ素ピラゾール誘導体の製造方法 |
| EP2297111B1 (de) * | 2008-05-02 | 2012-06-20 | Basf Se | Verfahren zur herstellung halogensubstituierter 2-(aminomethyliden)-3-oxobuttersäureester |
| BRPI0911898A2 (pt) * | 2008-05-02 | 2015-10-13 | Basf Se | processo para preparar compostos, e, composto. |
| CN102015654B (zh) | 2008-05-05 | 2014-03-12 | 巴斯夫欧洲公司 | 制备1，3，4-取代的吡唑化合物的方法 |
| US7601864B1 (en) * | 2008-05-08 | 2009-10-13 | Ufc Corporation | Method for synthesizing 4,4-dihalogen-2-(dialkylamino)methylene-3-oxy-alkylbutyrate and derivatives thereof |
| KR20110031501A (ko) * | 2008-07-21 | 2011-03-28 | 바스프 에스이 | 1,3-이치환된 피라졸카르복실산 에스테르의 제조 방법 |
| EP2320909B8 (en) | 2008-07-25 | 2016-03-30 | VIIV Healthcare Company | Chemical compounds |
| JP5228817B2 (ja) * | 2008-11-12 | 2013-07-03 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| RU2527451C2 (ru) | 2008-12-11 | 2014-08-27 | Вайв Хелткер Компани | Синтез карбамоилпиридоновых ингибиторов интегразы вич и промежуточных соединений |
| EP2376453B1 (en) | 2008-12-11 | 2019-11-20 | VIIV Healthcare Company | Intermediates for carbamoylpyridone hiv integrase inhibitors |
| TWI518084B (zh) | 2009-03-26 | 2016-01-21 | 鹽野義製藥股份有限公司 | 哌喃酮與吡啶酮衍生物之製造方法 |
| AR077503A1 (es) * | 2009-07-28 | 2011-08-31 | Syngenta Participations Ag | Procesos relacionados con la alquilacion de pirazoles |
| US8362273B2 (en) | 2009-11-05 | 2013-01-29 | Basf Se | Process for preparing aminale and their use for preparing 1,3-disubstituted pyrazole compounds |
| WO2011054732A1 (en) | 2009-11-05 | 2011-05-12 | Basf Se | Process for preparing 1,3-disubstituted pyrazole compounds |
| TWI582097B (zh) | 2010-03-23 | 2017-05-11 | Ｖｉｉｖ醫療保健公司 | 製備胺甲醯吡啶酮衍生物及中間體之方法 |
| ES2615729T3 (es) * | 2010-08-10 | 2017-06-08 | Syngenta Participations Ag | Proceso para preparar 3-haloalquilpirazoles |
| JP5605104B2 (ja) * | 2010-09-10 | 2014-10-15 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5830957B2 (ja) * | 2011-06-22 | 2015-12-09 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| CN103635461B (zh) * | 2011-06-22 | 2016-01-20 | 中央硝子株式会社 | 吡唑化合物的制造方法 |
| JP5793983B2 (ja) * | 2011-06-22 | 2015-10-14 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5915004B2 (ja) * | 2011-06-22 | 2016-05-11 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5790195B2 (ja) * | 2011-06-22 | 2015-10-07 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| EP2623496A1 (de) | 2012-02-01 | 2013-08-07 | Bayer CropScience AG | Verfahren zur Herstellung von 3,5-bis (fluoralkyl)-pyrazol-4-carbonsäure-Derivaten und 3,5-bis(fluoralkyl)-pyrazolen |
| CN102731402A (zh) * | 2012-06-29 | 2012-10-17 | 上海康鹏化学有限公司 | 3-三氟甲基吡唑-4-羧酸和3-二氟甲基吡唑-4-羧酸的制备方法 |
| US8871947B2 (en) | 2013-02-04 | 2014-10-28 | KingChem LLC | Preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid ester |
| MX2015016119A (es) | 2013-05-22 | 2016-03-31 | Bayer Cropscience Ag | Metodo para preparar derivados de 3,5-bis(fluoroalquil)pirazol. |
| WO2014187773A1 (en) | 2013-05-22 | 2014-11-27 | Bayer Cropscience Ag | PROCESS FOR PREPARING 3,5-BIS(FLUOROALKYL)PYRAZOLE DERIVATIVES FROM α,α-DIHALOAMINES |
| TWI647215B (zh) * | 2013-11-11 | 2019-01-11 | 德商拜耳作物科學股份有限公司 | 自α,α－二鹵胺製備３,５－雙鹵烷基吡唑衍生物之方法 |
| US9139507B2 (en) | 2013-12-09 | 2015-09-22 | KingChem LLC. | Process for the preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylate and its analogs |
| CN105980362A (zh) | 2014-01-10 | 2016-09-28 | 旭硝子株式会社 | 含醚性氧原子的全氟烷基取代吡唑环化合物及其制造方法 |
| EP3122727B1 (en) * | 2014-03-24 | 2018-01-31 | Bayer CropScience Aktiengesellschaft | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from alpha , alpha-dihaloamines and ketimines |
| EP3015458A1 (en) | 2014-11-03 | 2016-05-04 | Bayer CropScience AG | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines |
| ES2672581T3 (es) | 2014-06-11 | 2018-06-15 | Bayer Cropscience Aktiengesellschaft | Proceso para la preparación de 3,5-bis(haloalquil)pirazoles por medio de la acilación de cetiminas |
| ES2672577T3 (es) | 2014-06-11 | 2018-06-15 | Bayer Cropscience Aktiengesellschaft | Proceso para preparar derivados de 3,5-bis(haloalquil)pirazol por medio de la acilación de Hidrazonas |
| EP2987782A1 (en) | 2014-08-22 | 2016-02-24 | Solvay SA | Distillation process comprising at least two distillation steps to obtain purified halogenated carboxylic acid halide, and use of the purified halogenated carboxylic acid halide |
| WO2016079126A1 (en) | 2014-11-17 | 2016-05-26 | Solvay Sa | Distillation process comprising at least two distillation steps to obtain purified halogenated carboxylic acid halide, and use of the purified halogenated carboxylic acid halide |
| CN104529899A (zh) * | 2014-12-19 | 2015-04-22 | 浙江泰达作物科技有限公司 | 高区域选择性制备1-烷基-3-卤代烷基吡唑衍生物的方法 |
| CN105541716B (zh) * | 2015-03-26 | 2024-02-23 | Ａｇｃ株式会社 | 吡唑衍生物的制造方法 |
| KR20160120009A (ko) | 2015-04-07 | 2016-10-17 | (주)부흥산업사 | 4,4-디플루오로-((2-디알킬아미노)메틸렌)-3-옥소부탄산 알킬에스테르의 새로운 제조방법 |
| MX2017017140A (es) | 2015-06-26 | 2018-03-09 | Bayer Cropscience Ag | Proceso para la preparacion de pirazoles sustituidos que contienen grupos haloalcoxi-y haloalquiltio a partir de a,a-dihaloalquilaminas y quetiminas. |
| EP3178813A1 (en) | 2015-12-09 | 2017-06-14 | Basf Se | Method for preparing halogenated 3-oxocarboxylates carrying a 2-alkoxymethylidene or a 2-dialkylaminomethylidene group |
| WO2017194517A1 (en) * | 2016-05-10 | 2017-11-16 | Solvay Sa | Composition comprising 3-(haloalkyl or formyl)-1h-pyrazole-4-carboxylic acids or esters, its manufacture and its use for the preparation of carboxamides |
| JP7044766B2 (ja) | 2016-09-21 | 2022-03-30 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | ３－フルオロアルキル－５－ピラゾールカルボキシレート類及び３－フルオロアルキル－５－ピラゾールカルボン酸類を調製する方法 |
| JP2020532524A (ja) | 2017-09-04 | 2020-11-12 | ソルヴェイ（ソシエテ アノニム） | ジフルオロアセチルクロリドの製造方法及び製造中間体 |
| CN111116364B (zh) * | 2019-12-30 | 2022-11-11 | 浙江本立科技股份有限公司 | 2-多卤代乙酰基-3-烷氧基丙烯酸酯的制备方法 |
| CN113912541A (zh) * | 2021-10-29 | 2022-01-11 | 南通宝凯药业有限公司 | 一种3-二氟甲基-1-甲基-1h-吡唑-4-羧酸的制备方法 |
| CN114195715B (zh) * | 2021-12-31 | 2024-05-10 | 福建永晶科技股份有限公司 | 1-甲基-3-二氟甲基-4-吡唑酸和1-甲基-3-三氟甲基-4-吡唑酸的制备方法 |
| CN117447401B (zh) * | 2023-12-26 | 2024-04-19 | 山东国邦药业有限公司 | 一种二氟吡唑酸的合成方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5093347A (en) * | 1991-01-28 | 1992-03-03 | Monsanto Company | 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use |
| US5223526A (en) * | 1991-12-06 | 1993-06-29 | Monsanto Company | Pyrazole carboxanilide fungicides and use |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| KR20000035081A (ko) * | 1998-11-10 | 2000-06-26 | 마크 에스. 아들러 | 2-(트리할로아세틸)-3-(치환된 아미노)-2-프로페노에이트 제조방법 |
| KR20010078067A (ko) * | 2000-01-28 | 2001-08-20 | 고사이 아끼오 | 디할로-화합물 및 비타민 ａ 유도체의 제조 방법 |
| DE10161978A1 (de) * | 2001-12-17 | 2003-06-26 | Bayer Ag | Verfahren zur Herstellung von 2-Halogenacyl-3-amino-acrylsäure-derivate |
-
2003
- 2003-10-23 DE DE10349500A patent/DE10349500A1/de not_active Withdrawn
-
2004
- 2004-10-12 KR KR1020067009068A patent/KR101116686B1/ko active IP Right Grant
- 2004-10-12 AT AT04790277T patent/ATE494274T1/de active
- 2004-10-12 JP JP2006535992A patent/JP4725977B2/ja active Active
- 2004-10-12 DE DE502004012095T patent/DE502004012095D1/de active Active
- 2004-10-12 WO PCT/EP2004/011376 patent/WO2005042468A1/de active Application Filing
- 2004-10-12 BR BRPI0415855-5B1A patent/BRPI0415855B1/pt active IP Right Grant
- 2004-10-12 EP EP04790277A patent/EP1678119B1/de active Active
- 2004-10-12 CN CNB2004800312031A patent/CN100422141C/zh active Active
- 2004-10-12 MX MXPA06004339A patent/MXPA06004339A/es active IP Right Grant
- 2004-10-12 DK DK04790277.0T patent/DK1678119T3/da active
- 2004-10-12 US US10/576,059 patent/US7358387B2/en active Active
- 2004-10-22 TW TW093132065A patent/TWI363050B/zh active
-
2006
- 2006-04-03 IN IN1793DE2006 patent/IN2006DE01793A/en unknown
- 2006-04-20 IL IL175024A patent/IL175024A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| JP2007509850A (ja) | 2007-04-19 |
| US7358387B2 (en) | 2008-04-15 |
| CN100422141C (zh) | 2008-10-01 |
| IL175024A0 (en) | 2006-08-20 |
| TW200526550A (en) | 2005-08-16 |
| BRPI0415855B1 (pt) | 2013-11-05 |
| KR101116686B1 (ko) | 2012-02-22 |
| KR20060109901A (ko) | 2006-10-23 |
| CN1871204A (zh) | 2006-11-29 |
| DK1678119T3 (da) | 2011-05-02 |
| DE502004012095D1 (de) | 2011-02-17 |
| EP1678119B1 (de) | 2011-01-05 |
| BRPI0415855A (pt) | 2007-01-09 |
| IL175024A (en) | 2011-05-31 |
| JP4725977B2 (ja) | 2011-07-13 |
| TWI363050B (en) | 2012-05-01 |
| WO2005042468A1 (de) | 2005-05-12 |
| MXPA06004339A (es) | 2006-06-05 |
| DE10349500A1 (de) | 2005-06-02 |
| US20060252944A1 (en) | 2006-11-09 |
| EP1678119A1 (de) | 2006-07-12 |
| ATE494274T1 (de) | 2011-01-15 |
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