IL96996A - Preparation of 4-) Argolin - 8-Ilalkyl (Piprazine-2,6-discussions - Google Patents

Preparation of 4-) Argolin - 8-Ilalkyl (Piprazine-2,6-discussions

Info

Publication number
IL96996A
IL96996A IL9699691A IL9699691A IL96996A IL 96996 A IL96996 A IL 96996A IL 9699691 A IL9699691 A IL 9699691A IL 9699691 A IL9699691 A IL 9699691A IL 96996 A IL96996 A IL 96996A
Authority
IL
Israel
Prior art keywords
formula
compound
group
methyl
carbon atoms
Prior art date
Application number
IL9699691A
Other languages
English (en)
Hebrew (he)
Other versions
IL96996A0 (en
Inventor
Sergio Mantegani
Gabriella Traquandi
Tiziano Bandira
Enzo Brambilla
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB909001774A external-priority patent/GB9001774D0/en
Priority claimed from GB909025849A external-priority patent/GB9025849D0/en
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of IL96996A0 publication Critical patent/IL96996A0/xx
Publication of IL96996A publication Critical patent/IL96996A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
    • C07D457/12—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/02—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL9699691A 1990-01-25 1991-01-22 Preparation of 4-) Argolin - 8-Ilalkyl (Piprazine-2,6-discussions IL96996A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB909001774A GB9001774D0 (en) 1990-01-25 1990-01-25 Process for preparing ergoline derivatives
GB909025849A GB9025849D0 (en) 1990-11-28 1990-11-28 Process for preparing ergoline derivatives

Publications (2)

Publication Number Publication Date
IL96996A0 IL96996A0 (en) 1992-03-29
IL96996A true IL96996A (en) 1994-11-28

Family

ID=26296553

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9699691A IL96996A (en) 1990-01-25 1991-01-22 Preparation of 4-) Argolin - 8-Ilalkyl (Piprazine-2,6-discussions

Country Status (21)

Country Link
US (1) US5210194A (sv)
EP (1) EP0464178B1 (sv)
JP (1) JPH04504582A (sv)
KR (1) KR920701205A (sv)
AT (1) ATE131167T1 (sv)
AU (1) AU644625B2 (sv)
CA (1) CA2049053A1 (sv)
DE (1) DE69115138T2 (sv)
DK (1) DK0464178T3 (sv)
ES (1) ES2083564T3 (sv)
FI (1) FI96113C (sv)
GR (1) GR3019125T3 (sv)
HU (1) HU208971B (sv)
IE (1) IE72142B1 (sv)
IL (1) IL96996A (sv)
MY (1) MY106383A (sv)
NO (1) NO178373C (sv)
NZ (1) NZ236852A (sv)
PT (1) PT96557B (sv)
RU (1) RU2074857C1 (sv)
WO (1) WO1991011447A1 (sv)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4033496A1 (de) * 1990-10-20 1992-04-23 Sandoz Ag Neue ergolinderivate, ihre herstellung und verwendung
ATE204278T1 (de) * 1992-12-24 2001-09-15 Pharmacia & Upjohn Spa Serotoninergische ergolin derivate
GB9407637D0 (en) 1994-04-18 1994-06-08 Erba Carlo Spa Serotoninergic abeo-ergoline derivatives
GB9603226D0 (en) * 1996-02-15 1996-04-17 Pharmacia Spa Heterocyclyl-ergoline derivatives
US6060483A (en) * 1996-06-27 2000-05-09 Pharmacia & Upjohn S.P.A. Antineurodegenerative ergoline derivatives
ATE424414T1 (de) 2001-06-08 2009-03-15 Sod Conseils Rech Applic Chimere somatostatin-dopamin-analoga
TWI523863B (zh) 2012-11-01 2016-03-01 艾普森藥品公司 體抑素－多巴胺嵌合體類似物
WO2014070965A2 (en) 2012-11-01 2014-05-08 Ipsen Pharma S.A.S Somatostatin analogs and dimers thereof

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3763161A (en) * 1970-07-13 1973-10-02 Du Pont Tetrasubstituted dicyanopyrazines and related compounds
JPS58172012A (ja) * 1982-04-01 1983-10-08 Clarion Co Ltd 同一放送識別受信機
PH21123A (en) * 1983-04-28 1987-07-27 Erba Farmitalia Ergoline derivatives
US4806538A (en) * 1984-11-02 1989-02-21 Fujisawa Pharmaceutical Co., Ltd. Piperazine compound as PAF-antagonist
GB8501078D0 (en) * 1985-01-16 1985-02-20 Erba Farmitalia Piperazin-1-yl-ergo-line derivatives
DE3517247A1 (de) * 1985-05-13 1986-11-13 Gerhard Prof. Dr.-Ing. 8012 Ottobrunn Flachenecker Antennendiversity-empfangsanlage zur elimination von empfangsstoerungen
US4871736A (en) * 1986-11-25 1989-10-03 The Ohio State University Stereoisomeric tricyclic bis(dioxopiperazines) and pharmaceutical compositions
US4733402A (en) * 1987-04-23 1988-03-22 Signatron, Inc. Adaptive filter equalizer systems
DE3814899A1 (de) * 1988-05-03 1989-11-16 Hirschmann Richard Gmbh Co Empfangsverfahren und empfangs-antennensystem fuer mobilen empfang
NO175659C (no) * 1988-07-06 1994-11-09 Sumitomo Electric Industries Kommunikasjonssystem med multippelmottagning og mottagerapparat for diversitetssignaler
DE3926336C2 (de) * 1989-08-09 2001-03-29 Heinz Lindenmeier Antennendiversity-Empfangsanlage zur Elimination von Empfangsstörungen beim mobilen Empfang von Fernsehsignalen

Also Published As

Publication number Publication date
NZ236852A (en) 1992-05-26
PT96557B (pt) 1998-07-31
MY106383A (en) 1995-05-30
ATE131167T1 (de) 1995-12-15
NO913647L (no) 1991-09-16
NO178373B (no) 1995-12-04
IE910244A1 (en) 1991-07-31
HU208971B (en) 1994-02-28
CA2049053A1 (en) 1991-07-26
AU7078891A (en) 1991-08-21
DE69115138D1 (de) 1996-01-18
RU2074857C1 (ru) 1997-03-10
ES2083564T3 (es) 1996-04-16
NO913647D0 (no) 1991-09-16
EP0464178A1 (en) 1992-01-08
US5210194A (en) 1993-05-11
HUT58092A (en) 1992-01-28
GR3019125T3 (en) 1996-05-31
JPH04504582A (ja) 1992-08-13
FI96113B (sv) 1996-01-31
PT96557A (pt) 1991-10-15
KR920701205A (ko) 1992-08-11
WO1991011447A1 (en) 1991-08-08
AU644625B2 (en) 1993-12-16
IE72142B1 (en) 1997-03-26
DE69115138T2 (de) 1996-05-09
EP0464178B1 (en) 1995-12-06
NO178373C (no) 1996-03-13
FI914458A0 (sv) 1991-09-23
FI96113C (sv) 1996-05-10
IL96996A0 (en) 1992-03-29
DK0464178T3 (da) 1996-01-02

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