IL79222A0 - 2-oxy-4h-3,1-benzoxazin-4-one derivatives and related compounds,their preparation and pharmaceutical compositions containing them - Google Patents

2-oxy-4h-3,1-benzoxazin-4-one derivatives and related compounds,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL79222A0
IL79222A0 IL79222A IL7922286A IL79222A0 IL 79222 A0 IL79222 A0 IL 79222A0 IL 79222 A IL79222 A IL 79222A IL 7922286 A IL7922286 A IL 7922286A IL 79222 A0 IL79222 A0 IL 79222A0
Authority
IL
Israel
Prior art keywords
benzoxazin
oxy
derivatives
preparation
pharmaceutical compositions
Prior art date
Application number
IL79222A
Other languages
English (en)
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of IL79222A0 publication Critical patent/IL79222A0/xx
Priority to IL94245A priority Critical patent/IL94245A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
    • C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07F9/6533—Six-membered rings
    • C07F9/65335—Six-membered rings condensed with carbocyclic rings or carbocyclic ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IL79222A 1985-06-25 1986-06-24 2-oxy-4h-3,1-benzoxazin-4-one derivatives and related compounds,their preparation and pharmaceutical compositions containing them IL79222A0 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL94245A IL94245A0 (en) 1985-06-25 1990-05-01 2-carbalkoxyamino substituted benzoic acid derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/748,631 US4665070A (en) 1985-06-25 1985-06-25 2-oxy-4H-3,1-benzoxazin-4-ones and pharmaceutical use

Publications (1)

Publication Number Publication Date
IL79222A0 true IL79222A0 (en) 1986-09-30

Family

ID=25010264

Family Applications (1)

Application Number Title Priority Date Filing Date
IL79222A IL79222A0 (en) 1985-06-25 1986-06-24 2-oxy-4h-3,1-benzoxazin-4-one derivatives and related compounds,their preparation and pharmaceutical compositions containing them

Country Status (13)

Country Link
US (1) US4665070A (xx)
EP (1) EP0206323A1 (xx)
JP (1) JPS6230770A (xx)
KR (1) KR900004319B1 (xx)
AU (2) AU599320B2 (xx)
CA (1) CA1270487A (xx)
DK (1) DK297486A (xx)
ES (4) ES8802223A1 (xx)
FI (1) FI862691A (xx)
HU (1) HU196772B (xx)
IL (1) IL79222A0 (xx)
NO (1) NO163486C (xx)
ZA (1) ZA864715B (xx)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4745116A (en) * 1985-06-25 1988-05-17 Syntex (U.S.A.) Inc. 2-oxy-4H-3,1-benzoxazin-4-ones and related compounds and pharmaceutical use
CA1309556C (en) * 1987-06-09 1992-10-27 Masayuki Kokubo 4h-3,1-benzoxazin-4-one compounds and pharmaceutical composition thereoffor the inhibition of serine proteases
US5204462A (en) * 1990-03-30 1993-04-20 Japan Tobacco, Inc. 4h-3,1-benzoxazin-4-one derivative
US5985872A (en) * 1995-05-24 1999-11-16 G.D. Searle & Co. 2-amino-benzoxazinones for the treatment of viral infections
FR2763944B1 (fr) * 1997-06-03 2000-12-15 Centre Nat Rech Scient Nouveaux derives de coumarines, leurs procedes de preparation et leur application comme medicaments en tant qu'inhibiteurs de proteases
AU2826099A (en) * 1998-03-24 1999-10-18 Novo Nordisk A/S Heterocyclic compounds regulating clotting
US6180625B1 (en) 1998-03-24 2001-01-30 Novo Nordisk A/S Heterocyclic compounds regulating clotting
AU1375000A (en) * 1998-11-26 2000-06-13 Novo Nordisk A/S Heterocyclic compounds regulating clotting
AR022204A1 (es) * 1999-01-08 2002-09-04 Norgine Bv Compuesto, proceso para su preparacion, composicion farmaceutica y producto comestible que lo comprende.
GB9900416D0 (en) * 1999-01-08 1999-02-24 Alizyme Therapeutics Ltd Inhibitors
JP2003509538A (ja) * 1999-09-10 2003-03-11 ザ、プロクター、エンド、ギャンブル、カンパニー 酵素インヒビター
EP1628674A2 (en) * 2003-05-06 2006-03-01 Cytovia, Inc. Protease inhibitors for coronaviruses and sars-cov and the use thereof
MX297306B (es) 2006-11-22 2012-03-22 Ajinomoto Kk Procedimiento para la produccion de derivados de fenilalanina que tienen estructuras de base de quinazolinodiona e intermediarios para la produccion.
JP2010254623A (ja) * 2009-04-24 2010-11-11 Takeda Chem Ind Ltd ベンゾオキサジノン化合物の結晶

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU173974B (hu) * 1971-08-30 1979-10-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija proizvodnykh 3,1-benzoksazin-4-ona

Also Published As

Publication number Publication date
KR870000310A (ko) 1987-02-17
ES8801808A1 (es) 1988-03-01
AU599320B2 (en) 1990-07-19
ES8801806A1 (es) 1988-03-01
HUT41750A (en) 1987-05-28
AU5915086A (en) 1987-01-08
ES557731A0 (es) 1988-03-01
FI862691A (fi) 1986-12-26
DK297486D0 (da) 1986-06-24
HU196772B (en) 1989-01-30
ES8801807A1 (es) 1988-03-01
JPS6230770A (ja) 1987-02-09
KR900004319B1 (ko) 1990-06-22
EP0206323A1 (en) 1986-12-30
ES556514A0 (es) 1988-05-01
NO862534L (no) 1986-12-29
NO862534D0 (no) 1986-06-24
ES557732A0 (es) 1988-03-01
NO163486C (no) 1990-06-13
FI862691A0 (fi) 1986-06-24
ZA864715B (en) 1988-02-24
CA1270487A (en) 1990-06-19
NO163486B (no) 1990-02-26
US4665070A (en) 1987-05-12
AU4912090A (en) 1990-05-31
DK297486A (da) 1986-12-26
ES557730A0 (es) 1988-03-01
ES8802223A1 (es) 1988-05-01

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